论文信息 - Preparation of Useful Buiding-Blocks for the Synthesis of 7-Azanorbornylprostanoids

Preparation of Useful Buiding-Blocks for the Synthesis of 7-Azanorbornylprostanoids

Abstract The Diels-Alder adduct 4 of an N-protected pyrrole with dimethyl acetylenedicarboxylate can be transformed to 5 and 6 by short sequences which differenciate the two ester groups; these compounds are interesting starting materials for the synthesis of potential thromboxane A2 antagonists as well as other bio-active compounds.

G. Balme | J. Goré | K. Fégy | C. Traversa

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