Effects of the psychotomimetic benzomorphan N-allylnormetazocine (SKF 10,047) on prepulse inhibition of startle in mice
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[1] G. Collingridge,et al. Pharmacological Investigations of the Dissociative ‘Legal Highs’ Diphenidine, Methoxphenidine and Analogues , 2016, PloS one.
[2] S. Powell,et al. The novel ketamine analog methoxetamine produces dissociative-like behavioral effects in rodents , 2016, Psychopharmacology.
[3] F. Vollenweider,et al. Acute Effects of Lysergic Acid Diethylamide in Healthy Subjects , 2015, Biological Psychiatry.
[4] J. McLaughlin,et al. Physical Presence of Nor-Binaltorphimine in Mouse Brain over 21 Days after a Single Administration Corresponds to Its Long-Lasting Antagonistic Effect on κ-Opioid Receptors , 2013, The Journal of Pharmacology and Experimental Therapeutics.
[5] Matthew W. Johnson,et al. Dose-related effects of salvinorin A in humans: dissociative, hallucinogenic, and memory effects , 2013, Psychopharmacology.
[6] B. Cohen,et al. Dose-Related Behavioral, Subjective, Endocrine, and Psychophysiological Effects of the κ Opioid Agonist Salvinorin A in Humans , 2012, Biological Psychiatry.
[7] B. Cohen,et al. Long-acting κ opioid antagonists nor-BNI, GNTI and JDTic: pharmacokinetics in mice and lipophilicity , 2012, BMC pharmacology.
[8] Peter H. Addy. Acute and post-acute behavioral and psychological effects of salvinorin A in humans , 2011, Psychopharmacology.
[9] Matthew W. Johnson,et al. Human psychopharmacology and dose-effects of salvinorin A, a kappa opioid agonist hallucinogen present in the plant Salvia divinorum. , 2011, Drug and alcohol dependence.
[10] V. Chefer,et al. The effects of kappa-opioid receptor ligands on prepulse inhibition and CRF-induced prepulse inhibition deficits in the rat , 2010, Psychopharmacology.
[11] M. Geyer,et al. LSD but not lisuride disrupts prepulse inhibition in rats by activating the 5-HT2A receptor , 2009, Psychopharmacology.
[12] M. Geyer,et al. Prepulse inhibition of the startle reflex and its attentional modulation in the human S-ketamine and N,N-dimethyltryptamine (DMT) models of psychosis , 2007, Journal of psychopharmacology.
[13] Yuko Fujita,et al. Phencyclidine-Induced Cognitive Deficits in Mice are Improved by Subsequent Subchronic Administration of Fluvoxamine: Role of Sigma-1 Receptors , 2007, Neuropsychopharmacology.
[14] M. Hiramatsu,et al. Improvement of memory impairment by (+)- and (−)-pentazocine via sigma, but not kappa opioid receptors , 2005, Brain Research.
[15] G. Gessa,et al. Kappa Opioid Receptor Activation Disrupts Prepulse Inhibition of the Acoustic Startle in Rats , 2005, Biological Psychiatry.
[16] M. Geyer,et al. Parametric determinants in pre-stimulus modification of acoustic startle: interaction with ketamine , 2005, Psychopharmacology.
[17] E. Butelman,et al. Effects of the plant-derived hallucinogen salvinorin A on basal dopamine levels in the caudate putamen and in a conditioned place aversion assay in mice: agonist actions at kappa opioid receptors , 2005, Psychopharmacology.
[18] M. Geyer,et al. Dopaminergic stimulation disrupts sensorimotor gating in the rat , 2004, Psychopharmacology.
[19] D. Segal,et al. Evidence for multiple opiate receptor involvement in different phencyclidine-induced unconditioned behaviors in rats , 2004, Psychopharmacology.
[20] E. T. Iwamoto. Comparison of the pharmacologic effects of N-allylnormetazocine and phencyclidine: Sensitization, cross-sensitization, and opioid antagonist activity , 2004, Psychopharmacology.
[21] C. Haertzen. Subjective effects of narcotic antagonists cyclazocine and nalorphine on the Addiction Research Center Inventory (ARCI) , 2004, Psychopharmacologia.
[22] Teruo Hayashi,et al. Understanding the molecular mechanism of sigma-1 receptors: towards a hypothesis that sigma-1 receptors are intracellular amplifiers for signal transduction. , 2003, Current medicinal chemistry.
[23] J. Wiley,et al. Affinity and specificity of N-methyl-D-aspartate channel blockers affect their ability to disrupt prepulse inhibition of acoustic startle in rats , 2003, Psychopharmacology.
[24] Meyer B. Jackson,et al. The Sigma Receptor as a Ligand-Regulated Auxiliary Potassium Channel Subunit , 2002, Neuron.
[25] Franz X Vollenweider,et al. A systems model of altered consciousness: integrating natural and drug-induced psychoses , 2001, Brain Research Bulletin.
[26] G. Bigelow,et al. Enadoline, a selective kappa opioid agonist: comparison with butorphanol and hydromorphone in humans , 2001, Psychopharmacology.
[27] G. Pasternak,et al. Molecular cloning and pharmacological characterization of the rat sigma1 receptor. , 2001, Biochemical pharmacology.
[28] Erica Duncan,et al. Clinical and Sensorimotor Gating Effects of Ketamine in Normals , 2001, Neuropsychopharmacology.
[29] Teruo Hayashi,et al. Regulating ankyrin dynamics: Roles of sigma-1 receptors. , 2001, Proceedings of the National Academy of Sciences of the United States of America.
[30] M. Tanaka,et al. Effects of sigma(1) receptor ligand, MS-377 on apomorphine- or phencyclidine-induced disruption of prepulse inhibition of acoustic startle in rats. , 2000, European journal of pharmacology.
[31] M A Geyer,et al. Disruption of prepulse inhibition and increases in locomotor activity by competitive N-methyl-D-aspartate receptor antagonists in rats. , 1999, The Journal of pharmacology and experimental therapeutics.
[32] S. Kulkarni,et al. Sigma (σ1) receptor mediated antidepressant‐like effects of neurosteroids in the Porsolt forced swim test , 1998 .
[33] M. Decker,et al. Effects of phencyclidne (PCP) and (+)MK-801 on sensorimotor gating in CD-1 mice , 1998, Progress in Neuro-Psychopharmacology and Biological Psychiatry.
[34] S. Kulkarni,et al. Sigma (sigma1) receptor mediated anti-depressant-like effects of neurosteroids in the Porsolt forced swim test. , 1998, Neuroreport.
[35] Effects of phencyclidine (PCP) and (+)MK-801 on sensorimotor gating in CD-1 mice. , 1998, Progress in neuro-psychopharmacology & biological psychiatry.
[36] V. Ganapathy,et al. Cloning and structural analysis of the cDNA and the gene encoding the murine type 1 sigma receptor. , 1997, Biochemical and biophysical research communications.
[37] J. Witkin,et al. Dizocilpine-like discriminative stimulus effects of competitive NMDA receptor antagonists in mice , 1997, Psychopharmacology.
[38] E. Kempner,et al. Purification, molecular cloning, and expression of the mammalian sigma1-binding site. , 1996, Proceedings of the National Academy of Sciences of the United States of America.
[39] Y. Minabe,et al. Interactions of selective serotonin reuptake inhibitors with subtypes of sigma receptors in rat brain. , 1996, European journal of pharmacology.
[40] G. Pasternak,et al. (−)-Pentazocine analgesia in mice: interactions with a σ receptor system , 1995 .
[41] M. Pontecorvo,et al. NPC 16377, a potent and selective sigma-ligand. II. Behavioral and neuroprotective profile. , 1993, The Journal of pharmacology and experimental therapeutics.
[42] S. Holtzman. Discriminative stimulus effects of the PCP/σ-ligand (+)-N-Allylnormetazocine in monkeys , 1993, Pharmacology Biochemistry and Behavior.
[43] S. Holtzman. Discriminative stimulus effects of the PCP/sigma-ligand (+)-N-allylnormetazocine in monkeys. , 1993, Pharmacology, biochemistry, and behavior.
[44] J. Woods,et al. Tolerance to the cataleptic effect of the N-methyl-D-aspartate (NMDA) receptor antagonists in pigeons: cross-tolerance between PCP-like compounds and competitive NMDA antagonists. , 1992, The Journal of pharmacology and experimental therapeutics.
[45] S. Mascarella,et al. Enantiomeric N-substituted N-normetazocines: a comparative study of affinities at sigma, PCP, and mu opioid receptors. , 1992, Journal of medicinal chemistry.
[46] D. Javitt,et al. Recent advances in the phencyclidine model of schizophrenia. , 1991, The American journal of psychiatry.
[47] T. Cicero,et al. Affinity of drugs and peptides for U-69,593-sensitive and -insensitive kappa opiate binding sites: the U-69,593-insensitive site appears to be the beta endorphin-specific epsilon receptor. , 1990, The Journal of pharmacology and experimental therapeutics.
[48] J. Vignon,et al. In vivo labeling of phencyclidine (PCP) receptors with 3H‐TCP in the mouse brain , 1990, Journal of neuroscience research.
[49] J. Musacchio. The psychotomimetic effects of opiates and the sigma receptor. , 1990, Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology.
[50] E. Wong,et al. Evidence against an involvement of the haloperidol‐sensitive σ recognition site in the discriminative stimulus properties of (+)‐N‐allylnormetazocine ((+)‐SKF 10,047) , 1990, British journal of pharmacology.
[51] G. Ma,et al. Effects of phencyclidine and phencyclidine biologs on sensorimotor gating in the rat. , 1989 .
[52] W. Bowen,et al. Synthesis and evaluation of optically pure [3H]‐(+)‐pentazocine, a highly potent and selective radioligand for σ receptors , 1989 .
[53] D. Sanger,et al. The discriminative stimulus effects of MK-801: Generalization to other N-methyl-D-aspartate receptor antagonists , 1989, Journal of psychopharmacology.
[54] R. Balster. Substitution and antagonism in rats trained to discriminate (+)-N-allylnormetazocine from saline. , 1989, The Journal of pharmacology and experimental therapeutics.
[55] W. Bowen,et al. Synthesis and evaluation of optically pure [3H]-(+)-pentazocine, a highly potent and selective radioligand for sigma receptors. , 1989, FEBS letters.
[56] M. Geyer,et al. Effects of phencyclidine and phencyclidine biologs on sensorimotor gating in the rat. , 1989, Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology.
[57] S. M. Owens,et al. Structure-activity relationships of arylcyclohexylamines as discriminative stimuli in pigeons. , 1988, The Journal of pharmacology and experimental therapeutics.
[58] P. Portoghese,et al. Nor-binaltorphimine, a highly selective kappa-opioid antagonist in analgesic and receptor binding assays. , 1988, The Journal of pharmacology and experimental therapeutics.
[59] E. Domino,et al. Sigma and Phencyclidine: Like Compounds As Molecular Probes in Biology , 1988 .
[60] E. London,et al. Steroid binding at sigma receptors suggests a link between endocrine, nervous, and immune systems. , 1988, Science.
[61] L. Dykstra,et al. Discriminative stimulus effects of N-allylnormetazocine in rats trained to discriminate a kappa from a sigma agonist. , 1987, Life sciences.
[62] C. Haertzen,et al. Human psychopharmacology of ketocyclazocine as compared with cyclazocine, morphine and placebo. , 1986, The Journal of pharmacology and experimental therapeutics.
[63] L. Iversen,et al. The anticonvulsant MK-801 is a potent N-methyl-D-aspartate antagonist. , 1986, Proceedings of the National Academy of Sciences of the United States of America.
[64] H. Emrich,et al. Psychotomimesis mediated by kappa opiate receptors , 1986, Science.
[65] S. Snyder,et al. Pharmacological and autoradiographic discrimination of sigma and phencyclidine receptor binding sites in brain with (+)-[3H]SKF 10,047, (+)-[3H]-3-[3-hydroxyphenyl]-N-(1-propyl)piperidine and [3H]-1-[1-(2-thienyl)cyclohexyl]piperidine. , 1986, The Journal of pharmacology and experimental therapeutics.
[66] K. Rice,et al. Differentiation of [3H]phencyclidine and ( + )‐[3H]SKF‐10,047 binding sites in rat cerebral cortex , 1985, FEBS letters.
[67] B. Johnson,et al. Sigma opioid receptor: characterization and co-identity with the phencyclidine receptor. , 1985, The Journal of pharmacology and experimental therapeutics.
[68] S. Tam,et al. (+)-[^3H]SKF-10,047, (+)[^3H]ethylketocyclazocine, μ,κ,δ and phencyclidine binding sites in guinea pig brain membranes , 1985 .
[69] E. J. Simon,et al. Characterization of specific binding sites for [3H](d)-N-allylnormetazocine in rat brain membranes. , 1985, Molecular pharmacology.
[70] S. Tam,et al. Sigma opiates and certain antipsychotic drugs mutually inhibit (+)-[3H] SKF 10,047 and [3H]haloperidol binding in guinea pig brain membranes. , 1984, Proceedings of the National Academy of Sciences of the United States of America.
[71] J. Stonham,et al. The Effect of Naloxone on Pentazocine Induced Hallucinations , 1984, Journal of the Royal Army Medical Corps.
[72] A. H. Tang,et al. Discriminative stimulus properties of nalorphine in the rhesus monkeys. , 1983, The Journal of pharmacology and experimental therapeutics.
[73] S. Tam. Naloxone-inaccessible sigma receptor in rat central nervous system. , 1983, Proceedings of the National Academy of Sciences of the United States of America.
[74] A. Tomie,et al. Effects of SKF-10047 in the phencyclidine-dependent rat: evidence for common receptor mechanisms. , 1983, Drug and alcohol dependence.
[75] T. Su. Evidence for sigma opioid receptor: binding of [3H]SKF-10047 to etorphine-inaccessible sites in guinea-pig brain. , 1982, The Journal of pharmacology and experimental therapeutics.
[76] H. Shannon. Phencyclidine-like discriminative stimuli of (+)- and (-)-N-allylnormetazocine in rats. , 1982, European journal of pharmacology.
[77] A. Herz,et al. Non-opioid psychotomimetic-like discriminative stimulus properties of N-allylnormetazocine (SKF 10,047) in the rat. , 1982, European journal of pharmacology.
[78] K. Brady,et al. Stereoisomers of N-allylnormetazocine: phencyclidine-like behavioral effects in squirrel monkeys and rats. , 1982, Science.
[79] R. Zukin,et al. Demonstration of [3H]cyclazocine binding to multiple opiate receptor sites. , 1981, Molecular pharmacology.
[80] H. Merz,et al. N-[(Tetrahydrofuryl)alkyl] and N-(alkoxyalkyl) derivatives of (-)-normetazocine, compounds with differentiated opioid action profiles. , 1979, Journal of medicinal chemistry.
[81] C. Coursey. The Psychotomimetic Side Effects of Pentazocine , 1978 .
[82] W. Beaver,et al. Twin Crossover Relative Potency Analgesic Assays in Man. II. Morphine Vs. 8‐Methoxycyclazocine , 1977, Journal of clinical pharmacology.
[83] W. Beaver,et al. Twin Crossover Relative Potency Analgesic Assays in Man. I. Morphine Vs. Morphine , 1977, Journal of clinical pharmacology.
[84] J. Thompson,et al. The effects of morphine- and nalorphine- like drugs in the nondependent and morphine-dependent chronic spinal dog. , 1976, The Journal of pharmacology and experimental therapeutics.
[85] W. Forrest,et al. Analgesic and other effects of the d‐ and l‐isomers of pentazocine , 1969, Clinical pharmacology and therapeutics.
[86] D. Jasinski,et al. Antagonism of the subjective, behavioral, pupillary, and respiratory depressant effects of cyclazocine by naloxone , 1968, Clinical pharmacology and therapeutics.
[87] L. Lasagna,et al. THE ANALGESIC EFFICACY AND RESPIRATORY EFFECTS IN MAN OF A BENZOMORPHAN "NARCOTIC ANTAGONIST" , 1964 .
[88] A. Keats,et al. Narcotic Antagonists as Analgesics: Clinical Aspects , 1964 .
[89] L. Harris,et al. Narcotic Antagonists as Analgesics , 1962, Science.
[90] A. Keats,et al. Subjective effects of nalorphine in hospitalized patients. , 1957, The Journal of pharmacology and experimental therapeutics.
[91] R. Huggins,et al. SOME EFFECTS OF N–ALLYLNORMORPHINE ON NORMAL SUBJECTS AND A REVIEW OF THE LITERATURE , 1955, Anesthesiology.
[92] L. Lasagna,et al. The analgesic effectiveness of nalorphine and nalorphine-morphine combinations in man. , 1954, The Journal of pharmacology and experimental therapeutics.
[93] L. Lasagna. Nalorphine (n-allylnormorphine); practical and theoretical considerations. , 1954, A.M.A. archives of internal medicine.
[94] A. Wikler,et al. N-Allylnormorphine: effects of single doses and precipitation of acute abstinence syndromes during addiction to morphine; methadone or heroin in man (post addicts). , 1953, The Journal of pharmacology and experimental therapeutics.