Influence of Polymer Molecular Weight on Drug-Polymer Solubility: A Comparison between Experimentally Determined Solubility in PVP and Prediction Derived from Solubility in Monomer.
暂无分享,去创建一个
Thomas Rades | René Holm | Peter Langguth | Per Holm | T. Rades | P. Holm | R. Holm | P. Langguth | M. Knopp | N. E. Olesen | Niels Erik Olesen | Matthias Manne Knopp
[1] JULIAN F. Johnson,et al. Influence of molecular weight and molecular weight distribution on mechanical properties of polymers , 1982 .
[2] M. Descamps,et al. A new protocol to determine the solubility of drugs into polymer matrixes. , 2013, Molecular pharmaceutics.
[3] G. Van den Mooter,et al. Review: physical chemistry of solid dispersions. , 2009, The Journal of pharmacy and pharmacology.
[4] Ford Jl,et al. The current status of solid dispersions. , 1986 .
[5] Lian Yu,et al. Solubility of Small-Molecule Crystals in Polymers: d-Mannitol in PVP, Indomethacin in PVP/VA, and Nifedipine in PVP/VA , 2009, Pharmaceutical Research.
[6] Bradley D Anderson,et al. Molecular dynamics simulation of amorphous indomethacin-poly(vinylpyrrolidone) glasses: solubility and hydrogen bonding interactions. , 2013, Journal of pharmaceutical sciences.
[7] F. Haaf,et al. Polymers of N-Vinylpyrrolidone: Synthesis, Characterization and Uses , 1985 .
[8] Lynne S. Taylor,et al. Spectroscopic Characterization of Interactions Between PVP and Indomethacin in Amorphous Molecular Dispersions , 1997, Pharmaceutical Research.
[9] Raymond C Rowe,et al. Handbook of Pharmaceutical Excipients , 1994 .
[10] P Augustijns,et al. Physical stabilisation of amorphous ketoconazole in solid dispersions with polyvinylpyrrolidone K25. , 2001, European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences.
[11] Simon Bates,et al. Evaluation of Drug-Polymer Miscibility in Amorphous Solid Dispersion Systems , 2009, Pharmaceutical Research.
[12] J Hadgraft,et al. Crystallization of hydrocortisone acetate: influence of polymers. , 2001, International journal of pharmaceutics.
[13] JULIAN F. Johnson,et al. Mechanical Properties of Polymers: The Influence of Molecular Weight and Molecular Weight Distribution , 1972 .
[14] Patrick J. Marsac,et al. Theoretical and Practical Approaches for Prediction of Drug–Polymer Miscibility and Solubility , 2006, Pharmaceutical Research.
[15] James S. Taylor,et al. Ideal copolymers and the second‐order transitions of synthetic rubbers. i. non‐crystalline copolymers , 2007 .
[16] Thomas Rades,et al. Emerging trends in the stabilization of amorphous drugs. , 2013, International journal of pharmaceutics.
[17] Peter York,et al. Mechanisms of dissolution of frusemide pvp solid dispersions , 1987 .
[18] S. Thakral,et al. Prediction of drug-polymer miscibility through the use of solubility parameter based Flory-Huggins interaction parameter and the experimental validation: PEG as model polymer. , 2013, Journal of pharmaceutical sciences.
[19] J. Torrado,et al. Preparation, dissolution and characterization of albendazole solid dispersions , 1996 .
[20] Wagh Vinod Tukaram. Solid Dispersions as Strategy to Improve Oral Bioavailability of Poor Water Soluble Drugs , 2013 .
[21] A. Ravve,et al. Principles of Polymer Chemistry , 1995 .
[22] M. Otsuka,et al. Determination of indomethacin polymorphic contents by chemometric near-infrared spectroscopy and conventional powder X-ray diffractometry. , 2001, The Analyst.
[23] R. Jachowicz. Dissolution rates of partially water-soluble drugs from solid dispersion systems. I. Prednisolone , 1987 .
[24] J. Ford. The current status of solid dispersions. , 1986, Pharmaceutica acta Helvetiae.
[25] V. Caron,et al. A comparison of spray drying and milling in the production of amorphous dispersions of sulfathiazole/polyvinylpyrrolidone and sulfadimidine/polyvinylpyrrolidone. , 2011, Molecular pharmaceutics.
[26] Lian Yu,et al. Solubilities of crystalline drugs in polymers: an improved analytical method and comparison of solubilities of indomethacin and nifedipine in PVP, PVP/VA, and PVAc. , 2010, Journal of pharmaceutical sciences.
[27] M. Summers,et al. The effect of wetting agents on the dissolution of indomethacin solid dispersion systems , 1986 .
[28] Amrit Paudel,et al. Theoretical and experimental investigation on the solid solubility and miscibility of naproxen in poly(vinylpyrrolidone). , 2010, Molecular pharmaceutics.
[29] E. Squillante,et al. Solid dispersion of carbamazepine in PVP K30 by conventional solvent evaporation and supercritical methods. , 2004, International journal of pharmaceutics.
[30] George Zografi,et al. Physical Properties of Solid Molecular Dispersions of Indomethacin with Poly(vinylpyrrolidone) and Poly(vinylpyrrolidone-co-vinyl-acetate) in Relation to Indomethacin Crystallization , 1999, Pharmaceutical Research.
[31] Patrick J. Marsac,et al. Estimation of Drug–Polymer Miscibility and Solubility in Amorphous Solid Dispersions Using Experimentally Determined Interaction Parameters , 2008, Pharmaceutical Research.
[32] N. Rodríguez-Hornedo,et al. Significance of controlling crystallization mechanisms and kinetics in pharmaceutical systems. , 1999, Journal of pharmaceutical sciences.
[33] T. Rades,et al. Evaluation of drug-polymer solubility curves through formal statistical analysis: comparison of preparation techniques. , 2015, Journal of pharmaceutical sciences.
[34] Bruno C. Hancock,et al. Crystallization of indomethacin from the amorphous state below and above its glass transition temperature. , 1994, Journal of pharmaceutical sciences.
[35] Feng Qian,et al. Drug-polymer solubility and miscibility: Stability consideration and practical challenges in amorphous solid dispersion development. , 2010, Journal of pharmaceutical sciences.
[36] N. Lordi,et al. Thermal Analysis Studies of Glass Dispersion Systems , 1984 .
[37] W. Higuchi,et al. Dissolution rates of high energy polyvinylpyrrolidone (PVP)-sulfathiazole coprecipitates. , 1969, Journal of pharmaceutical sciences.
[38] Bruno C. Hancock,et al. Characteristics and significance of the amorphous state in pharmaceutical systems. , 1997, Journal of pharmaceutical sciences.
[39] J Dressman,et al. Improving drug solubility for oral delivery using solid dispersions. , 2000, European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V.
[40] Patrick Augustijns,et al. Physico-chemical characterization of solid dispersions of temazepam with polyethylene glycol 6000 and PVP K30 , 1998 .
[41] Ravi M Shanker,et al. Solubility advantage of amorphous pharmaceuticals: I. A thermodynamic analysis. , 2010, Journal of pharmaceutical sciences.