Discovery of 2-chloro-N-(4-methoxyphenyl)-N-methylquinazolin-4-amine (EP128265, MPI-0441138) as a potent inducer of apoptosis with high in vivo activity.
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Mark B. Anderson | S. Kasibhatla | V. Baichwal | S. Cai | Kevin W. Jessing | J. Drewe | Songchun Jiang | Hong Zhang | B. Tseng | G. Mather | C. Pleiman | J. Willardsen | N. Sirisoma | A. Pervin | R. Hussain | Khanh C Hoang