A single amino acid change makes a rat neuronal sodium channel highly sensitive to pyrethroid insecticides

[1]  T. M. Brown,et al.  Altered properties of neuronal sodium channels associated with genetic resistance to pyrethroids. , 1999, Molecular pharmacology.

[2]  W. Catterall,et al.  Voltage Sensor–Trapping Enhanced Activation of Sodium Channels by β-Scorpion Toxin Bound to the S3–S4 Loop in Domain II , 1998, Neuron.

[3]  S. Y. Wang,et al.  Point mutations in segment I-S6 render voltage-gated Na+ channels resistant to batrachotoxin. , 1998, Proceedings of the National Academy of Sciences of the United States of America.

[4]  P. Usherwood,et al.  Functional analysis of a rat sodium channel carrying a mutation for insect knock‐down resistance (kdr) to pyrethroids , 1997, FEBS letters.

[5]  R. Reenan,et al.  Functional Expression of Drosophila para Sodium Channels Modulation by the Membrane Protein TipE and Toxin Pharmacology , 1997 .

[6]  W. Catterall,et al.  Molecular Determinants of High Affinity Binding of α-Scorpion Toxin and Sea Anemone Toxin in the S3-S4 Extracellular Loop in Domain IV of the Na+ Channel α Subunit* , 1996, The Journal of Biological Chemistry.

[7]  T. Narahashi,et al.  Modulation of sodium channels of rat cerebellar Purkinje neurons by the pyrethroid tetramethrin. , 1996, The Journal of pharmacology and experimental therapeutics.

[8]  T. Narahashi,et al.  Differential effects of the pyrethroid tetramethrin on tetrodotoxin-sensitive and tetrodotoxin-resistant single sodium channels , 1996, Brain Research.

[9]  J. Bloomquist Ion channels as targets for insecticides. , 1996, Annual review of entomology.

[10]  P. Deák,et al.  Cloning and functional analysis of tipE, a novel membrane protein that enhances drosophila para sodium channel function , 1995, Cell.

[11]  W. Catterall,et al.  Molecular determinants of state-dependent block of Na+ channels by local anesthetics. , 1994, Science.

[12]  T. Narahashi,et al.  Differential mechanism of action of the pyrethroid tetramethrin on tetrodotoxin-sensitive and tetrodotoxin-resistant sodium channels. , 1994, The Journal of pharmacology and experimental therapeutics.

[13]  A. L. Goldin,et al.  Site-directed mutagenesis of the putative pore region of the rat IIA sodium channel. , 1993, Molecular pharmacology.

[14]  W. Catterall,et al.  Cellular and molecular biology of voltage-gated sodium channels. , 1992, Physiological reviews.

[15]  X. Zong,et al.  Relation between veratridine reaction dynamics and macroscopic Na current in single cardiac cells , 1992, The Journal of general physiology.

[16]  F. Conti,et al.  Mapping the site of block by tetrodotoxin and saxitoxin of sodium channel II , 1991, FEBS letters.

[17]  I. Denholm,et al.  Characterization of the structure-activity relationship of kdr and two variants of super-kdr to pyrethroids in the housefly (Musca domestica L.) , 1987 .

[18]  J. Casida,et al.  Two classes of pyrethroid action in the cockroach , 1981 .