Synthesis of metallo-β-lactamase inhibitors
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[1] J. Frère,et al. Trifluoromethyl alcohol and ketone inhibitors of metallo-β-lactamases , 1996 .
[2] C. Schofield,et al. Reaction of ruppert's reagent (TMS-CF3) with Oxazolidinones: Synthesis of protected α-amino trifluoromethylketones , 1995 .
[3] J. Frère,et al. The 3‐D structure of a zinc metallo‐beta‐lactamase from Bacillus cereus reveals a new type of protein fold. , 1995 .
[4] J. Frère,et al. Beta‐lactamases and bacterial resistance to antibiotics , 1995, Molecular microbiology.
[5] P. Warner,et al. Non-peptidic inhibitors of human leukocyte elastase. 1. The design and synthesis of pyridone-containing inhibitors. , 1994, Journal of medicinal chemistry.
[6] Bert L. Vallee,et al. Zinc: biological functions and coordination motifs , 1993 .
[7] C. Free,et al. Activated ketone based inhibitors of human renin. , 1993, Journal of medicinal chemistry.
[8] D. Payne,et al. Metallo-beta-lactamases--a new therapeutic challenge. , 1993, Journal of medical microbiology.
[9] M. A. McClinton,et al. Trifluoromethylations and related reactions in organic chemistry , 1992 .
[10] P. Edwards. A method for the stereoselective synthesis of peptidyl trifluoromethyl ketones , 1992 .
[11] P. Mui,et al. Inhibition of human leukocyte elastase (HLE) by N-substituted peptidyl trifluoromethyl ketones. , 1992, Journal of medicinal chemistry.
[12] D. Dess,et al. A useful 12-I-5 triacetoxyperiodinane (the Dess-Martin periodinane) for the selective oxidation of primary or secondary alcohols and a variety of related 12-I-5 species , 1991 .
[13] D. Bonnet-Delpon,et al. Preparation of trifluoromethyl ketones and related fluorinated ketones , 1991 .
[14] N. Peet,et al. Synthesis of peptidyl fluoromethyl ketones and peptidyl alpha-keto esters as inhibitors of porcine pancreatic elastase, human neutrophil elastase, and rat and human neutrophil cathepsin G. , 1990, Journal of medicinal chemistry.
[15] J. Riordan,et al. Angiotensin-converting enzyme: new concepts concerning its biological role. , 1989, Biochemistry.
[16] D. M. Graves,et al. Oxidation of fluoroalkyl-substituted carbinols by the Dess-Martin reagent , 1989 .
[17] A. Gołębiowski,et al. Optically active N-protected .alpha.-amino aldehydes in organic synthesis , 1989 .
[18] K. Fukushima,et al. Phenylalanine derivatives enhancing intestinal absorption of insulin in mice. , 1988, Chemical & pharmaceutical bulletin.
[19] Brian W. Matthews,et al. Structural basis of the action of thermolysin and related zinc peptidases , 1988 .
[20] M. Kolb,et al. Synthesis of fluorinated α-amino ketones part I: α-benzamidoalkyl mono- di- and trifluoromethyl ketones , 1986 .
[21] B. Imperiali,et al. A versatile synthesis of peptidyl fluoromethyl ketones , 1986 .
[22] M. Kolb. Synthesis of fluorinated a-amino ketones. Part II: a-acylaminoalkyl a', a'-difluoroalkyl ketones , 1986 .
[23] D. Burton,et al. A remarkably simple preparation of (trifluoromethyl)cadmium and -zinc reagents directly from difluorodihalomethanes , 1985 .
[24] M. Gelb,et al. Fluoro ketone inhibitors of hydrolytic enzymes. , 1985, Biochemistry.
[25] P. G. Gassman,et al. Pentafluoroethyllithium. Generation and use in synthesis , 1985 .
[26] I. Ruppert,et al. Die ersten CF3-substituierten organyl(chlor)silane , 1984 .
[27] S. Nahm,et al. N-methoxy-n-methylamides as effective acylating agents , 1982 .
[28] R. Hiskey,et al. Azomethine Chemistry. II. Formation of Peptides from Oxazolidine-5-ones , 1963 .
[29] E. Ronwin. Direct Acylation of α-Amino Acids and Dipeptides , 1953 .