The Optimisation of a Novel, Weak Bromo and Extra Terminal Domain (BET) Bromodomain Fragment Ligand to a Potent and Selective Second Bromodomain (BD2) Inhibitor.
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P. Grandi | A. Michon | I. Wall | James M. Woolven | P. Bamborough | R. Prinjha | C. Chung | S. Atkinson | E. Demont | I. Rioja | Simon Taylor | R. Copley | M. Lindon | D. Mitchell | L. A. Harrison | Cassie Messenger | James R. J. Gray | Alex Preston | Laurie J. Gordon | Jonathan T. Seal | Thomas G. Hayhow | Robert J. Watson | H. Aylott