2-Substituted tryptamines: agents with selectivity for 5-HT(6) serotonin receptors.
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B. Roth | S. Hufeisen | R. Glennon | J. Savage | R A Glennon | M Lee | J B Rangisetty | M Dukat | B L Roth | J E Savage | A McBride | L Rauser | S Hufeisen | D K Lee | M. Dukat | L. Rauser | Mase Lee | D. Lee | A. McBride | J. B. Rangisetty | M. Lee | Bryan L. Roth | Laura Rauser | Jason E. Savage | Sandy Hufeisen | David H. Lee
[1] E. Shaw. The Synthesis of Tryptamines Related to Serotonin , 1955 .
[2] M. Yoshioka,et al. Central distribution and function of 5-HT6 receptor subtype in the rat brain. , 1998, Life sciences.
[3] A. Brown,et al. (+/-) 3-Amino-6-carboxamido-1,2,3,4-tetrahydrocarbazole: a conformationally restricted analogue of 5-carboxamidotryptamine with selectivity for the serotonin 5-HT1D receptor. , 1993, Journal of medicinal chemistry.
[4] F. Monsma,et al. Determination of the role of the 5-ht6 receptor in the rat brain: a study using antisense oligonucleotides. , 1995, The Journal of pharmacology and experimental therapeutics.
[5] G. Fillion,et al. Characterization of 5-ht6 receptor and expression of 5-ht6 mRNA in the rat brain during ontogenetic development , 1998, Naunyn-Schmiedeberg's Archives of Pharmacology.
[6] L. Lanfumey,et al. Immuno-localization of serotonin 5-HT6 receptor-like material in the rat central nervous system , 1997, Brain Research.
[7] D. Sibley,et al. Binding of typical and atypical antipsychotic agents to 5-hydroxytryptamine-6 and 5-hydroxytryptamine-7 receptors. , 1994, The Journal of pharmacology and experimental therapeutics.
[8] F. Monsma,et al. Effects of altered 5-ht6 expression in the rat: functional studies using antisense oligonucleotides , 1995, Behavioural Brain Research.
[9] D. Sibley,et al. Cloning, Characterization, and Chromosomal Localization of a Human 5‐HT6 Serotonin Receptor , 1996, Journal of neurochemistry.
[10] Gavin Kilpatrick,et al. 5-HT 3 Receptors , 1993 .
[11] 5-HT6 serotonin receptor binding of indolealkylamines: A preliminary structure-affinity investigation , 1999 .
[12] A. Brown,et al. 5-Chloro-N-(4-methoxy-3-piperazin-1-yl- phenyl)-3-methyl-2-benzothiophenesulfon- amide (SB-271046): a potent, selective, and orally bioavailable 5-HT6 receptor antagonist. , 1999, Journal of medicinal chemistry.
[13] J. Schwartz,et al. A novel rat serotonin (5-HT6) receptor: molecular cloning, localization and stimulation of cAMP accumulation. , 1993, Biochemical and biophysical research communications.
[14] L. Lanfumey,et al. Antibodies and Antisense Oligonucleotide for Probing the Distribution and Putative Functions of Central 5-HT6Receptors , 1999, Neuropsychopharmacology.
[15] R. Glennon,et al. Binding of O-Alkyl Derivatives of Serotonin at Human 5-HT1Dβ Receptors , 1996 .
[16] A. Sleight,et al. The 5-hydroxytryptamine6 receptor-selective radioligand [3H]Ro 63-0563 labels 5-hydroxytryptamine receptor binding sites in rat and porcine striatum. , 1998, Molecular pharmacology.
[17] A. Sleight,et al. The 5-hydroxytryptamine 6 receptor: localisation and function , 1998 .
[18] A. Sleight,et al. Characterization of Ro 04‐6790 and Ro 63‐0563: potent and selective antagonists at human and rat 5‐HT6 receptors , 1998, British journal of pharmacology.
[19] R. Glennon,et al. Serotonin receptors and their ligands: A lack of selective agents , 1991, Pharmacology Biochemistry and Behavior.
[20] L. C. Clark,et al. Synthesis of O- and N-Methylated Derivatives of 5-Hydroxytryptamine , 1958 .
[21] D. Sibley,et al. Cloning and expression of a novel serotonin receptor with high affinity for tricyclic psychotropic drugs. , 1993, Molecular pharmacology.
[22] D. Sibley,et al. Clozapine: Selective Labeling of Sites Resembling 5HT6 Serotonin Receptors May Reflect Psychoactive Profile , 1995, Molecular medicine.