A mild and efficient route to 2-benzyl tryptamine derivatives via ring-opening of β-carbolines

[1]  Sunil K. Sharma,et al.  Water as an efficient medium for the synthesis of tetrahydro -β-carbolines via Pictet-Spengler reactions , 2007 .

[2]  D. Sames,et al.  Catalytic C-H arylation of SEM-protected azoles with palladium complexes of NHCs and phosphines. , 2006, Organic letters.

[3]  M. Brown,et al.  Direct palladium-catalyzed C-2 and C-3 arylation of indoles: a mechanistic rationale for regioselectivity. , 2005, Journal of the American Chemical Society.

[4]  J. Cook,et al.  A general strategy for the synthesis of vincamajine-related indole alkaloids: stereocontrolled total synthesis of (+)-dehydrovoachalotine, (-)-vincamajinine, and (-)-11-methoxy-17-epivincamajine as well as the related quebrachidine diol, vincamajine diol, and vincarinol. , 2005, Journal of Organic Chemistry.

[5]  D. Sames,et al.  Direct C-arylation of free (NH)-indoles and pyrroles catalyzed by Ar-Rh(III) complexes assembled in situ. , 2005, Journal of the American Chemical Society.

[6]  D. Sames,et al.  Direct C-H bond arylation: selective palladium-catalyzed C2-arylation of N-substituted indoles. , 2004, Organic letters.

[7]  Weiqin Jiang,et al.  Furoyl and benzofuroyl pyrroloquinolones as potent and selective PDE5 inhibitors for treatment of erectile dysfunction. , 2003, Journal of medicinal chemistry.

[8]  J. Poupaert,et al.  Antioxidant activity of pinoline analogues in the LDL oxidation model , 2002 .

[9]  M. Paal,et al.  Efficient synthesis of 3-(4,5-dihydro-1H-imidazole-2-yl)-1H-indoles , 2001 .

[10]  H. Tokuyama,et al.  Radical Cyclization of 2-Alkenylthioanilides: A Novel Synthesis of 2,3-Disubstituted Indoles , 1999 .

[11]  M. Nakagawa,et al.  CHIRAL AUXILIARY APPROACH TO THE ASYMMETRIC PICTET-SPENGLER REACTION OF TRYPTAMINES , 1999 .

[12]  L. Chu,et al.  SYNTHESIS OF 2-ARYLTRYPTAMINES WITH PALLADIUM CATALYZED CROSS-COUPLING OF 2-BROMOTRYPTAMINES AND ARYLBORONIC ACIDS , 1997 .

[13]  James Lin,et al.  Derivatives of 5-amidine indole as inhibitors of thrombin catalytic activity , 1996 .

[14]  S. Labadie,et al.  Palladium-Mediated Benzylation of Dimetalated 1-Butylindole-3-carboxylic Acid , 1995 .

[15]  H. Araki,et al.  Synthesis and Pharmacological Evaluation of 1, 2, 3, 4-Tetrahydro-β-carboline Derivatives , 1995 .

[16]  S. Labadie,et al.  Indol-2-yltributylstannane: A Versatile Reagent for 2-Substituted Indoles , 1994 .

[17]  K. Maruoka,et al.  Regioselective Fischer indole synthesis mediated by organoaluminum amides , 1993 .

[18]  J. Mérour,et al.  Synthesis and Reactions of 1-Acetyl-2-benzylidene-3-oxo-2,3-dihydroindoles , 1989 .

[19]  S. Ram,et al.  Ammonium Formate in Organic Synthesis: A Versatile Agent in Catalytic Hydrogen Transfer Reductions , 1988 .