Discovery of an Orally Efficacious Imidazo[5,1-f][1,2,4]triazine Dual Inhibitor of IGF-1R and IR.
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D. Werner | P. Gokhale | E. May | K. Foreman | Hanqing Dong | Kam W. Siu | R. Wild | J. Pachter | E. Buck | M. Mulvihill | Radoslaw S. Laufer | Lixin Feng | A. Steinig | Kathryn M. Stolz | Yan Yao | An-Hu Li | Meizhong Jin | Mridula Kadalbajoo | Andrew Kleinberg | A. Cooke | M. Bittner | D. Landfair