Discovery of 6-(2,4-Dichlorophenyl)-5-[4-[(3S)-1-(3-fluoropropyl)pyrrolidin-3-yl]oxyphenyl]-8,9-dihydro-7H-benzo[7]annulene-2-carboxylic acid (SAR439859), a Potent and Selective Estrogen Receptor Degrader (SERD) for the Treatment of Estrogen Receptor Positive Breast Cancer.
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M. Mathieu | C. García-echeverría | M. Levit | A. Rak | F. Vallée | Hong Cheng | C. Muller | Fangxian Sun | V. Certal | G. Mccort | M. Tabart | P. Vicat | Y. El-Ahmad | F. Halley | Fabienne Thompson | V. Steier | A. Hebert | M. Bouaboula | P. Abecassis | V. Loyau | L. Schio | L. Bertin | Laurence Fabien | Maysoun Shomali | M. Brollo | Christelle Perrault | Florence Gruss-Leleu | Fabienne Pilorge | Bruno Filoche-Rommé | Patrick Richepin | T. Bénard | Gilles Lebourg | Audrey Louboutin | Pascal Desmazeau | A. Courjaud | Chrystelle Girardet | Sylvie Beccari | Jacques Le-Roux | C. Terrier | C. Ginesty | Laurent Schio | Véronique Loyau