Cobalt-catalyzed isocyanide insertion cyclization to dihydrobenzoimidazotriazins
暂无分享,去创建一个
[1] Anand H Shinde,et al. Nickel-Catalyzed Aerobic Oxidative Isocyanide Insertion: Access to Benzimidazoquinazoline Derivatives via a Sequential Double Annulation Cascade (SDAC) Strategy. , 2017, The Journal of organic chemistry.
[2] Y. Liu,et al. Discovery of 4-(4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)benzamides as novel, highly potent and selective, orally bioavailable inhibitors of Tyrosine Threonine Kinase, TTK. , 2016, Bioorganic & medicinal chemistry letters.
[3] A. Bazgir,et al. Synthesis of benzoimidazoquinazolines by cobalt-catalyzed isocyanide insertion–cyclization , 2016 .
[4] J. Skolnick,et al. Ligand binding studies, preliminary structure-activity relationship and detailed mechanistic characterization of 1-phenyl-6,6-dimethyl-1,3,5-triazine-2,4-diamine derivatives as inhibitors of Escherichia coli dihydrofolate reductase. , 2015, European journal of medicinal chemistry.
[5] H. Stark,et al. (2-Arylethenyl)-1,3,5-triazin-2-amines as a novel histamine H4 receptor ligands. , 2015, European journal of medicinal chemistry.
[6] Vijay Luxami,et al. Triazine as a promising scaffold for its versatile biological behavior. , 2015, European journal of medicinal chemistry.
[7] Andrej Perdih,et al. 4,6-Substituted-1,3,5-triazin-2(1H)-ones as monocyclic catalytic inhibitors of human DNA topoisomerase IIα targeting the ATP binding site. , 2015, Bioorganic & medicinal chemistry.
[8] Xuesen Fan,et al. Synthesis of Pyrazolo[5,1-a]isoindoles and Pyrazolo[5,1-a]isoindole-3-carboxamides through One-Pot Cascade Reactions of 1-(2-Bromophenyl)buta-2,3-dien-1-ones with Isocyanide and Hydrazine or Acetohydrazide. , 2015, The Journal of organic chemistry.
[9] W. Chui,et al. Synthesis and biological activity of fluorinated 7-benzylamino-2-phenyl-1,2,4-triazolo[1,5-a][1,3,5]triazin-5-amines , 2015 .
[10] Guigen Li,et al. Synthesis of 3-Iminoindol-2-amines and Cyclic Enaminones via Palladium-Catalyzed Isocyanide Insertion-Cyclization. , 2015, The Journal of organic chemistry.
[11] Tian-Qi Wei,et al. Cobalt-Catalyzed Intermolecular Oxidative Isocyanide Insertion with Two Amines: An Approach to Guanidines , 2015 .
[12] M. Kumawat,et al. Discovery of novel 1,3,5-triazine-thiazolidine-2,4-diones as dipeptidyl peptidase-4 inhibitors with antibacterial activity targeting the S1 pocket for the treatment of type 2 diabetes , 2015 .
[13] Niren Murthy. In vivo delivery of transcription factors with chemically modified oligonucleotides , 2014 .
[14] Tian-Qi Wei,et al. NiCl2-catalyzed cascade reaction of isocyanides with functionalized anilines , 2014 .
[15] C. Cai,et al. One-pot synthesis of 2-amino-4(3H)-quinazolinones via ring-opening of isatoic anhydride and palladium-catalyzed oxidative isocyanide-insertion. , 2014, Organic & biomolecular chemistry.
[16] J. Zhao,et al. Direct Access to Isoindolinone Derivatives by Palladium-Catalyzed C–H Activation and Isocyanide Insertion by Using Molecular Oxygen as the Sole Oxidant , 2014, Synthesis.
[17] T. Tang,et al. Divergent synthesis of 6H-isoindolo[2,1-a]indol-6-ones and indenoindolones: an investigation of Pd-catalyzed isocyanide insertion , 2014 .
[18] Baishan Jiang,et al. Facile synthesis of 2-amino-3-bromoquinolines by palladium-catalyzed isocyanide insertion and cyclization of gem-dibromovinylanilines , 2014 .
[19] Tian-Qi Wei,et al. Cobalt(II)-Catalyzed Isocyanide Insertion Reaction with Amines under Ultrasonic Conditions: A Divergent Synthesis of Ureas, Thioureas and Azaheterocycles , 2014 .
[20] Gitte Van Baelen,et al. Synthesis of Pyridopyrimidines by Palladium-Catalyzed Isocyanide Insertion , 2014 .
[21] Shun-Yi Wang,et al. Palladium-Catalyzed Cascade Reactions of Isocyanides with Enaminones: Synthesis of 4-Aminoquinoline Derivatives , 2014 .
[22] Y. S. Prabhakar,et al. Discovery of triazine mimetics as potent antileishmanial agents. , 2013, ACS medicinal chemistry letters.
[23] Hong Chen,et al. Synthesis of chromeno[2,3-d]imidazol-9(1H)-ones via tandem reactions of 3-iodochromones with amidines involving copper-catalyzed C-H functionalization and C-O bond formation. , 2013, Organic letters.
[24] Jianguo Yang,et al. Cascade synthesis of azoquinazolinones by Cu(I)-catalyzed C–N coupling/C–H activation/C–N formation reactions under O2 , 2013 .
[25] Jie Wu,et al. Recent advances in isocyanide insertion chemistry. , 2013, Chemical Society reviews.
[26] Liming Hu,et al. Copper-catalyzed N-arylation and aerobic oxidative C–H/C–H coupling: one-pot synthesis of indoloimidazoquinoline derivatives , 2013 .
[27] Shun-Yi Wang,et al. Cobalt-catalyzed oxidative isocyanide insertion to amine-based bisnucleophiles: diverse synthesis of substituted 2-aminobenzimidazoles, 2-aminobenzothiazoles, and 2-aminobenzoxazoles. , 2013, Chemistry.
[28] Jihui Li,et al. Copper catalyzed N-arylation of amidines with aryl boronic acids and one-pot synthesis of benzimidazoles by a Chan-Lam-Evans N-arylation and C-H activation/C-N bond forming process. , 2012, Organic letters.
[29] T. Bush,et al. Discovery and optimization of potent and selective imidazopyridine and imidazopyridazine mTOR inhibitors. , 2012, Bioorganic & medicinal chemistry letters.
[30] Jongdoo Lim,et al. Triazine dendrimers as drug delivery systems: from synthesis to therapy. , 2012, Advanced drug delivery reviews.
[31] Daniel J. Freeman,et al. Structure-based design of a novel series of potent, selective inhibitors of the class I phosphatidylinositol 3-kinases. , 2012, Journal of medicinal chemistry.
[32] Qiang Zhu,et al. Palladium-catalyzed intramolecular C(sp2)-H amidination by isonitrile insertion provides direct access to 4-aminoquinazolines from N-arylamidines. , 2011, Organic letters.
[33] S. Katiyar,et al. Synthesis and cytotoxicity evaluation of (tetrahydro-beta-carboline)-1,3,5-triazine hybrids as anticancer agents. , 2010, European journal of medicinal chemistry.
[34] A. Konstas,et al. 24-hour intraocular pressures with brimonidine purite versus dorzolamide added to latanoprost in primary open-angle glaucoma subjects. , 2005, Ophthalmology.
[35] P. Bednarski,et al. Synthesis and anticancer activity of novel 2-amino-4-(4-phenylpiperazino)- 1,3,5-triazine derivatives. , 2004, Acta poloniae pharmaceutica.
[36] W. Schnick,et al. Melem (2,5,8-triamino-tri-s-triazine), an important intermediate during condensation of melamine rings to graphitic carbon nitride: synthesis, structure determination by X-ray powder diffractometry, solid-state NMR, and theoretical studies. , 2003, Journal of the American Chemical Society.
[37] E. Novellino,et al. Design, synthesis and biological evaluation of novel N-alkyl- and N-acyl-(7-substituted-2-phenylimidazo[1,2-a][1,3,5]triazin-4-yl)amines (ITAs) as novel A(1) adenosine receptor antagonists. , 2002, Journal of medicinal chemistry.
[38] M. Jhon,et al. Synthesis and electrorheological characteristics of microencapsulated polyaniline particles with melamine-formaldehyde resins , 2001 .
[39] T. Kappe,et al. Synthesis and in vitro anti‐HIV Activity of Certain 2‐(1H‐Benzimidazol‐2‐ylamino)pyrimidin‐4(3H)‐ones and Related Derivatives , 1997, Archiv der Pharmazie.
[40] Changjin Zhu,et al. Copper-catalyzed N-arylation and aerobic oxidation: one-pot synthesis of tetrahydroisoquinolino[2,1-a]quinazolinone derivatives , 2014 .
[41] H. Abdel-ghany,et al. Synthesis and biological activity of dihydroimidazole and 3,4-dihydrobenzo[4,5]imidazo[1,2-a][1,3,5]triazins. , 2012, European journal of medicinal chemistry.
[42] W. Chui,et al. Synthesis of 2-amino-s-triazino[1,2-a]benzimidazoles as potential antifolates from 2-guanidino- and 2-guanidino-5-methylbenzimidazoles , 2006 .
[43] Dieter Martin,et al. Cyansäureester. 31. Umsetzungen von 2‐Guanidino‐benzimidazol mit elektrophilen Reagentien , 1981 .