International Union of Pharmacology. LXIV. Estrogen Receptors
暂无分享,去创建一个
V. Craig Jordan | John A. Katzenellenbogen | Karin Dahlman-Wright | S. Fuqua | K. Dahlman-Wright | J. Gustafsson | J. Katzenellenbogen | K. Korach | V. Jordan | V. Jordan | A. Maggi | M. Muramatsu | M. Parker | Adriana Maggi | Malcolm G. Parker | Masami Muramatsu | Kenneth S. Korach | V. Cavaillès | Jan-Åke Gustafsson | Vincent Cavailles | Suzanne A. Fuqua | Malcolm G. Parker
[1] W. Gradishar,et al. Selective estrogen receptor modulators and prevention of invasive breast cancer. , 2006, JAMA.
[2] Norman Wolmark,et al. Effects of tamoxifen vs raloxifene on the risk of developing invasive breast cancer and other disease outcomes: the NSABP Study of Tamoxifen and Raloxifene (STAR) P-2 trial. , 2006, JAMA.
[3] K. Korach,et al. 17beta-estradiol induces apoptosis in the developing rodent prostate independently of ERalpha or ERbeta. , 2006, Endocrinology.
[4] K. Korach,et al. 17β-Estradiol Induces Apoptosis in the Developing Rodent Prostate Independently of ERα or ERβ , 2006 .
[5] V. Jordan,et al. Selective estrogen receptor modulators (SERMs): mechanisms of anticarcinogenesis and drug resistance. , 2005, Mutation research.
[6] D. McDonnell,et al. Coregulators in nuclear estrogen receptor action: from concept to therapeutic targeting. , 2005, Molecular interventions.
[7] Byung-Mu Lee,et al. Assessment of Estrogenic and Androgenic Activities of Tetramethrin in Vitro and in Vivo Assays , 2005, Journal of toxicology and environmental health. Part A.
[8] R. Millikan,et al. The estrogen receptor-α A908G (K303R) mutation occurs at a low frequency in invasive breast tumors: results from a population-based study , 2005, Breast Cancer Research.
[9] Miguel A Hernán,et al. Recent use of oral contraceptives and the risk of multiple sclerosis. , 2005, Archives of neurology.
[10] F. Naftolin,et al. Is the Estrogen Controversy Over? Deconstructing the Women's Health Initiative Study: A Critical Evaluation of the Evidence , 2005, Annals of the New York Academy of Sciences.
[11] W. Boon,et al. Estrogen, a fundamental player in energy homeostasis , 2005, The Journal of Steroid Biochemistry and Molecular Biology.
[12] C. Burke. Endometrial cancer and tamoxifen. , 2005, Clinical journal of oncology nursing.
[13] R. Bhat,et al. Identification of pathway-selective estrogen receptor ligands that inhibit NF-kappaB transcriptional activity. , 2005, Proceedings of the National Academy of Sciences of the United States of America.
[14] J. Lindgren,et al. Effects of anti-estrogens on bone in castrated and intact female rats , 1987, Breast Cancer Research and Treatment.
[15] Yukun Cui,et al. Phosphorylation of Estrogen Receptor α Blocks Its Acetylation and Regulates Estrogen Sensitivity , 2004, Cancer Research.
[16] K. Korach,et al. Estrogen receptor-alpha mediates the detrimental effects of neonatal diethylstilbestrol (DES) exposure in the murine reproductive tract. , 2004, Toxicology.
[17] Toremifene and tamoxifen are equally effective for early-stage breast cancer: first results of International Breast Cancer Study Group Trials 12-93 and 14-93. , 2004, Annals of oncology : official journal of the European Society for Medical Oncology.
[18] J. Gustafsson,et al. Estrogen Receptor-Beta Regulates Epithelial Cell Differentiation in the Mouse Ventral Prostate , 2004, Hormone Research in Paediatrics.
[19] J. Gustafsson,et al. Estrogen receptor β regulates epithelial cellular differentiation in the mouse ventral prostate , 2004 .
[20] E. Tokunaga,et al. No Hypersensitive Estrogen Receptor-α Mutation (K303R) in Japanese Breast Carcinomas , 2004, Breast Cancer Research and Treatment.
[21] G. B. Lopes,et al. Effects of estrogen plus progestin on health-related quality of life. , 2004, The New England journal of medicine.
[22] J. Kemper,et al. Differential regulation of the human progesterone receptor gene through an estrogen response element half site and Sp1 sites , 2004, The Journal of Steroid Biochemistry and Molecular Biology.
[23] C. Bailey,et al. Role of ovarian hormones in the long-term control of glucose homeostasis , 1980, Diabetologia.
[24] E. Tokunaga,et al. No hypersensitive estrogen receptor-alpha mutation (K303R) in Japanese breast carcinomas. , 2004, Breast cancer research and treatment.
[25] R. Brinton. Impact of Estrogen Therapy on Alzheimer’s Disease , 2004, CNS drugs.
[26] Wade V Welshons,et al. Phosphorylation of estrogen receptor alpha blocks its acetylation and regulates estrogen sensitivity. , 2004, Cancer research.
[27] M Nilsson,et al. Association of estrogen receptor β gene polymorphisms with bulimic disease in women , 2004, Molecular Psychiatry.
[28] K. Korach,et al. Estrogen receptor knockout mice as a model for endocrine research. , 2004, ILAR journal.
[29] Dennis B. Lubahn,et al. Estrogen Receptor α Mediates Estrogen’s Immune Protection in Autoimmune Disease , 2003, The Journal of Immunology.
[30] N. Sicotte,et al. Immune Modulation in Multiple Sclerosis Patients Treated with the Pregnancy Hormone Estriol 1 , 2003, The Journal of Immunology.
[31] E. Lam,et al. Expression of estrogen receptor beta isoforms in normal breast epithelial cells and breast cancer: regulation by methylation. , 2003, Oncogene.
[32] D. Labuda,et al. Human estrogen receptor beta 548 is not a common variant in three distinct populations. , 2003, Endocrinology.
[33] J. Gustafsson,et al. Update on estrogen signaling , 2003, FEBS letters.
[34] B. Bhavnani. Estrogens and menopause: pharmacology of conjugated equine estrogens and their potential role in the prevention of neurodegenerative diseases such as Alzheimer’s , 2003, The Journal of Steroid Biochemistry and Molecular Biology.
[35] J. Lovejoy. The menopause and obesity. , 2003, Primary care.
[36] V. Jordan,et al. The estrogen receptor: a model for molecular medicine. , 2003, Clinical cancer research : an official journal of the American Association for Cancer Research.
[37] S. Malhotra,et al. Effect of hormone replacement therapy on cardiovascular disease: current opinion , 2003, Expert opinion on pharmacotherapy.
[38] D. Lubahn,et al. Estrogen receptor alpha mediates estrogen's immune protection in autoimmune disease. , 2003, Journal of immunology.
[39] E. Barrett-Connor,et al. Baseline characteristics of participants in the Raloxifene Use for The Heart (RUTH) trial. , 2002, The American journal of cardiology.
[40] G. Patrinos,et al. DNA hypermethylation: when tumour suppressor genes go silent , 2002, Human Genetics.
[41] J. Gustafsson,et al. pS2 Gene expression in HepG2 cells: complex regulation through crosstalk between the estrogen receptor alpha, an estrogen-responsive element, and the activator protein 1 response element. , 2002, Molecular pharmacology.
[42] P. Chambon,et al. Estrogen Receptor-&agr; Mediates the Protective Effects of Estrogen Against Vascular Injury , 2002, Circulation research.
[43] David A. Agard,et al. Structural characterization of a subtype-selective ligand reveals a novel mode of estrogen receptor antagonism , 2002, Nature Structural Biology.
[44] Myles Brown,et al. Molecular Determinants for the Tissue Specificity of SERMs , 2002, Science.
[45] E. Bleecker,et al. Estrogen-receptor polymorphisms and effects of estrogen replacement on high-density lipoprotein cholesterol in women with coronary disease. , 2002, The New England journal of medicine.
[46] J. Gustafsson,et al. Abnormal Vascular Function and Hypertension in Mice Deficient in Estrogen Receptor β , 2002, Science.
[47] R. Baron,et al. Deletion of estrogen receptors reveals a regulatory role for estrogen receptors-beta in bone remodeling in females but not in males. , 2002, Bone.
[48] Martin Koš,et al. 0888-8809/01/$03.00/0 Molecular Endocrinology 15(12):2057–2063 Printed in U.S.A. Copyright © 2001 by The Endocrine Society Minireview: Genomic Organization of the Human ER � Gene Promoter Region , 2022 .
[49] V. Speirs,et al. Expression of alternatively spliced estrogen receptor alpha mRNAs is increased in breast cancer tissues , 2001, The Journal of Steroid Biochemistry and Molecular Biology.
[50] B. Katzenellenbogen,et al. Estrogen receptor-beta potency-selective ligands: structure-activity relationship studies of diarylpropionitriles and their acetylene and polar analogues. , 2001, Journal of medicinal chemistry.
[51] K. Korach,et al. Estrogen Receptor-α Knockout Mice Exhibit Resistance to the Developmental Effects of Neonatal Diethylstilbestrol Exposure on the Female Reproductive Tract , 2001 .
[52] K. Belguise,et al. Characterization of the Physical Interaction between Estrogen Receptor α and JUN Proteins* , 2001, The Journal of Biological Chemistry.
[53] G. Lazennec. ER Inhibits Proliferation and Invasion of Breast Cancer Cells , 2001 .
[54] A. Lucas,et al. ERβ Inhibits Proliferation and Invasion of Breast Cancer Cells. , 2001, Endocrinology.
[55] D. Lubahn,et al. Estrogen receptor‐ and aromatase‐deficient mice provide insight into the roles of estrogen within the ovary and uterus * , 2001, Molecular reproduction and development.
[56] S. Safe,et al. Differential activation of wild-type and variant forms of estrogen receptor α by synthetic and natural estrogenic compounds using a promoter containing three estrogen-responsive elements , 2001, The Journal of Steroid Biochemistry and Molecular Biology.
[57] B. Katzenellenbogen,et al. Direct Acetylation of the Estrogen Receptor α Hinge Region by p300 Regulates Transactivation and Hormone Sensitivity* , 2001, The Journal of Biological Chemistry.
[58] M. Helder,et al. Is GnRH self-priming an obligatory feature of the reproductive cycle? , 2001, Human reproduction.
[59] S. Safe. Transcriptional activation of genes by 17 beta-estradiol through estrogen receptor-Sp1 interactions. , 2001, Vitamins and hormones.
[60] F. Gannon,et al. Minireview: genomic organization of the human ERalpha gene promoter region. , 2001, Molecular endocrinology.
[61] K. Belguise,et al. Characterization of the physical interaction between estrogen receptor alpha and JUN proteins. , 2001, The Journal of biological chemistry.
[62] K. Korach,et al. Estrogen receptor-alpha knockout mice exhibit resistance to the developmental effects of neonatal diethylstilbestrol exposure on the female reproductive tract. , 2001, Developmental biology.
[63] A. Lucas,et al. ER beta inhibits proliferation and invasion of breast cancer cells. , 2001, Endocrinology.
[64] Y. Miyoshi,et al. Quantitative analysis of estrogen receptor‐β mRNA and its variants in human breast cancers , 2000, International journal of cancer.
[65] B. Katzenellenbogen,et al. Pyrazole ligands: structure-affinity/activity relationships and estrogen receptor-alpha-selective agonists. , 2000, Journal of medicinal chemistry.
[66] Satoshi Inoue,et al. Association of estrogen receptor β (ESR2) gene polymorphism with blood pressure , 2000, Journal of Human Genetics.
[67] F. Gannon,et al. Identification of a new isoform of the human estrogen receptor‐alpha (hER‐α) that is encoded by distinct transcripts and that is able to repress hER‐α activation function 1 , 2000 .
[68] J. Gustafsson,et al. Functional Differences between the Amino-Terminal Domains of Estrogen Receptors α and β , 2000 .
[69] S. Hilsenbeck,et al. A hypersensitive estrogen receptor-alpha mutation in premalignant breast lesions. , 2000, Cancer research.
[70] C. Klinge,et al. Estrogen receptor interaction with co-activators and co-repressors☆ , 2000, Steroids.
[71] E. Mazzon,et al. 17β-Estradiol Antiinflammatory Activity in Carrageenan-Induced Pleurisy. , 2000, Endocrinology.
[72] Y. Ouchi,et al. Association of Estrogen Receptor β Gene Polymorphism with Bone Mineral Density , 2000 .
[73] F. Gannon,et al. Identification of a new isoform of the human estrogen receptor-alpha (hER-alpha) that is encoded by distinct transcripts and that is able to repress hER-alpha activation function 1. , 2000, The EMBO journal.
[74] R. Dahiya,et al. Cloning and characterization of human estrogen receptor beta promoter. , 2000, Biochemical and biophysical research communications.
[75] Y. Ouchi,et al. Association of estrogen receptor beta (ESR2) gene polymorphism with blood pressure. , 2000, Journal of human genetics.
[76] Y. Ouchi,et al. Association of estrogen receptor beta gene polymorphism with bone mineral density. , 2000, Biochemical and biophysical research communications.
[77] E. Mazzon,et al. 17beta-estradiol antiinflammatory activity in carrageenan-induced pleurisy. , 2000, Endocrinology.
[78] J. Gustafsson,et al. Functional differences between the amino-terminal domains of estrogen receptors alpha and beta. , 2000, Molecular pharmacology.
[79] R. Karas,et al. The protective effects of estrogen on the cardiovascular system. , 2002, The New England journal of medicine.
[80] P. Mecocci,et al. Association of the estrogen receptor alpha gene polymorphisms with sporadic Alzheimer's disease. , 1999, Biochemical and biophysical research communications.
[81] L. Moore,et al. Expression of wild-type estrogen receptor beta and variant isoforms in human breast cancer. , 1999, Cancer research.
[82] B. Ponder,et al. A Systematic Review Of Genetic Polymorphisms and Breast Cancer Risk 1 , 2000 .
[83] K E Carlson,et al. Estrogen receptor subtype-selective ligands: asymmetric synthesis and biological evaluation of cis- and trans-5,11-dialkyl- 5,6,11, 12-tetrahydrochrysenes. , 1999, Journal of medicinal chemistry.
[84] B. Katzenellenbogen,et al. Novel ligands that function as selective estrogens or antiestrogens for estrogen receptor-alpha or estrogen receptor-beta. , 1999, Endocrinology.
[85] J. Hebebrand,et al. Systematic mutation screening of the estrogen receptor beta gene in probands of different weight extremes: identification of several genetic variants. , 1998, The Journal of clinical endocrinology and metabolism.
[86] Helmut Dotzlaw,et al. Estrogen receptor beta: mine is longer than yours? , 1998, The Journal of clinical endocrinology and metabolism.
[87] J. Corton,et al. Interaction of Estrogenic Chemicals and Phytoestrogens with Estrogen Receptor β. , 1998, Endocrinology.
[88] Y. Ouchi,et al. Molecular cloning and characterization of human estrogen receptor βcx: A potential inhibitor of estrogen action in human , 1998 .
[89] J. Gustafsson,et al. Differential response of estrogen receptor alpha and estrogen receptor beta to partial estrogen agonists/antagonists. , 1998, Molecular pharmacology.
[90] J. Lehmann,et al. Cloning and Characterization of Human Estrogen Receptor β Isoforms , 1998 .
[91] Interaction and dissociation by ligands of estrogen receptor and Hsp90: the antiestrogen RU 58668 induces a protein synthesis-dependent clustering of the receptor in the cytoplasm. , 1998, Molecular endocrinology.
[92] S. Kato,et al. A novel isoform of rat estrogen receptor beta with 18 amino acid insertion in the ligand binding domain as a putative dominant negative regular of estrogen action. , 1998, Biochemical and biophysical research communications.
[93] Y. Ouchi,et al. The complete primary structure of human estrogen receptor beta (hER beta) and its heterodimerization with ER alpha in vivo and in vitro. , 1998, Biochemical and biophysical research communications.
[94] J. Corton,et al. Interaction of estrogenic chemicals and phytoestrogens with estrogen receptor beta. , 1998, Endocrinology.
[95] Y. Ouchi,et al. Molecular cloning and characterization of human estrogen receptor betacx: a potential inhibitor ofestrogen action in human. , 1998, Nucleic acids research.
[96] Zbigniew Dauter,et al. Molecular basis of agonism and antagonism in the oestrogen receptor , 1997, Nature.
[97] S. Chu,et al. Identification of a splice variant of the rat estrogen receptor β gene , 1997, Molecular and Cellular Endocrinology.
[98] S. Safe,et al. Identification of a functional imperfect estrogen-responsive element in the 5'-promoter region of the human cathepsin D gene. , 1997, Biochemistry.
[99] N. Copeland,et al. Cloning, chromosomal localization, and functional analysis of the murine estrogen receptor beta. , 1997, Molecular endocrinology.
[100] J. Gustafsson,et al. Comparison of the ligand binding specificity and transcript tissue distribution of estrogen receptors alpha and beta. , 1997, Endocrinology.
[101] S. Chu,et al. Identification of a splice variant of the rat estrogen receptor beta gene. , 1997, Molecular and Cellular Endocrinology.
[102] J. Gustafsson,et al. Cloning of a novel receptor expressed in rat prostate and ovary. , 1996, Proceedings of the National Academy of Sciences of the United States of America.
[103] E. May,et al. Human estrogen receptor messenger RNA variants in both normal and tumor breast tissues , 1995, Molecular and Cellular Endocrinology.
[104] K. Korach,et al. Estrogen resistance caused by a mutation in the estrogen-receptor gene in a man. , 1994, The New England journal of medicine.
[105] M. Tzukerman,et al. Human estrogen receptor transactivational capacity is determined by both cellular and promoter context and mediated by two functionally distinct intramolecular regions. , 1994, Molecular endocrinology.
[106] G. Aguiari,et al. Dinucleotide repeat polymorphism in the human estrogen receptor (ESR) gene. , 1992, Human molecular genetics.
[107] Y. Edwards,et al. Two TaqI polymorphisms at the human PGM1 locus. , 1992, Human molecular genetics.
[108] J. Ham,et al. Structural organization and expression of the mouse estrogen receptor. , 1987, Molecular endocrinology.
[109] S. Koike,et al. Molecular cloning and characterization of rat estrogen receptor cDNA. , 1987, Nucleic acids research.
[110] P. Argos,et al. Human oestrogen receptor cDNA: sequence, expression and homology to v-erb-A , 1986, Nature.
[111] J. Shine,et al. Sequence and expression of human estrogen receptor complementary DNA. , 1986, Science.
[112] C. Bailey,et al. Role of ovarian hormones in the long-term control of glucose homeostasis. Effects of insulin secretion. , 1980, Diabetologia.