Preparation of a bromine-76 labelled analogue of epibatidine: a potent ligand for nicotinic acetylcholine receptor studies.
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C. Crouzel | R. Dannals | M. Kassiou | F. Dollé | B. Maziére | J. Musachio | C. Loc'h | L. Dolci
[1] D. Comar,et al. Nicotine-11C: Synthesis and distribution kinetics in animals , 1976, European Journal of Nuclear Medicine.
[2] D. Gündisch. Nicotinic acetylcholine receptors and imaging. , 2000, Current pharmaceutical design.
[3] N. Volkow,et al. Dopamine Receptor‐Mediated Regulation of Striatal Cholinergic Activity , 2000, Journal of neurochemistry.
[4] N. Volkow,et al. Occupancy of brain nicotinic acetylcholine receptors by nicotine doses equivalent to those obtained when smoking a cigarette , 2000, Synapse.
[5] C. Crouzel,et al. Synthesis of a fluorine-18 labeled derivative of epibatidine for in vivo nicotinic acetylcholine receptor PET imaging. , 1999, Bioorganic & medicinal chemistry.
[6] E. London,et al. Synthesis and evaluation of N-[11C]methylated analogues of epibatidine as tracers for positron emission tomographic studies of nicotinic acetylcholine receptors. , 1998, Journal of medicinal chemistry.
[7] J S Fowler,et al. Fluoro-norchloroepibatidine: preclinical assessment of acute toxicity. , 1997, Nuclear Medicine and Biology.
[8] E. London,et al. [125/123I]IPH: A radioiodinated analog of epibatidine for in vivo studies of nicotinic acetylcholine receptors , 1997, Synapse.
[9] Y. Yonekura,et al. Synthesis and characterization of radioiodinated (S)-5-iodonicotine: a new ligand for potential imaging of brain nicotinic cholinergic receptors by single photon emission computed tomography. , 1997, Chemical & pharmaceutical bulletin.
[10] H Lundqvist,et al. Imaging of nicotinic and muscarinic receptors in Alzheimer's disease: effect of tacrine treatment. , 1997, Dementia and geriatric cognitive disorders.
[11] E. London,et al. Synthesis of a radioiodinated analog of epibatidine : (±)-exo-2-(2-iodo-5-pyridyl)-7-azabicyclo[2.2.1]heptane for in vitro and in vivo studies of nicotinic acetylcholine receptors , 1997 .
[12] N. Volkow,et al. Mapping nicotinic acetylcholine receptors with PET , 1996, Synapse.
[13] E. London,et al. Synthesis of a radiotracer for studying nicotinic acetylcholine receptors : (+/−)-exo-2-(2-[18F]fluoro-5-pyridyl)-7-azabicyclo[2.2.1]heptane , 1996 .
[14] J. Krystal,et al. Continuous intravenous infusion of iodine-123-IBZM for SPECT determination of human brain dopamine receptor occupancy by antipsychotic agent RWJ-37796. , 1996, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[15] R Anand,et al. Comparative pharmacology of epibatidine: a potent agonist for neuronal nicotinic acetylcholine receptors. , 1995, Molecular pharmacology.
[16] E. London,et al. In vivo labeling of nicotinic acetylcholine receptors in brain with [3H]epibatidine. , 1995, European journal of pharmacology.
[17] B. Långström,et al. Kinetic Analysis of Regional (S)(-)11C‐Nicotine Binding in Normal and Alzheimer Brains In Vivo Assessment Using Positron Emission Tomography , 1995, Alzheimer disease and associated disorders.
[18] E. Wong,et al. Characterization of the electrophysiological, biochemical and behavioral actions of epibatidine. , 1995, The Journal of pharmacology and experimental therapeutics.
[19] M. Maziére. Cholinergic neurotransmission studied in vivo using positron emission tomography or single photon emission computerized tomography. , 1995, Pharmacology & therapeutics.
[20] M. Damaj,et al. Pharmacological effects of epibatidine optical enantiomers , 1994, Brain Research.
[21] A. Nordberg. Human nicotinic receptors—Their role in aging and dementia , 1994, Neurochemistry International.
[22] J. Daly,et al. Epibatidine, a potent analgetic and nicotinic agonist. , 1994, Molecular pharmacology.
[23] P. Merlet,et al. Preparation and pharmacological characterization of [76Br]-meta-bromobenzylguanidine ([76Br]MBBG). , 1994, Nuclear medicine and biology.
[24] J. Eckman,et al. Epibatidine is a nicotinic analgesic. , 1993, European journal of pharmacology.
[25] A. Nordberg. Clinical studies in Alzheimer patients with positron emission tomography , 1993, Behavioural Brain Research.
[26] A. Regan,et al. A total synthesis of (±)-epibatidine , 1993 .
[27] B. Winblad,et al. Tacrine restores cholinergic nicotinic receptors and glucose metabolism in alzheimer patients as visualized by positron emission tomography , 1992, Neurobiology of Aging.
[28] Y. Yonekura,et al. Synthesis of (S)-N-[methyl-11C]nicotine and its regional distribution in the mouse brain: a potential tracer for visualization of brain nicotinic receptors by positron emission tomography. , 1992, Chemical & pharmaceutical bulletin.
[29] E. Vogel,et al. Small and Medium Rings, 74. Syntheses and Photoelectron Spectra of 7‐Azanorbornadiene and Related Compounds An Analysis with Fragment Orbitals , 1991 .
[30] S. Moerlein,et al. No-Carrier-Added Radiohalogenation Methods with Heavy Halogens , 1983 .
[31] G. Antoni,et al. Synthesis of some 11C-labelled alkaloids , 1982 .