O-Ethyl 1-azidoalkylphosphonic acids—versatile reagents for the synthesis of protected phosphonamidate peptides
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[1] D. Sikora,et al. A New Synthesis of Protected Phosphonodipeptides with an N-Terminal Amino Acid , 2000 .
[2] D. Sikora,et al. A FACILE SYNTHESIS OF DIETHYL 1- ISOTHIOCYANO)ALKYLPHOSPHONATES[1] , 2000 .
[3] F. Hammerschmidt,et al. Enzymes in organic chemistry. Part 9:Chemo-enzymatic synthesis of phosphonic acid analogues of l-valine, l-leucine, l-isoleucine, l-methionine and l-α-aminobutyric acid of high enantiomeric excess , 1999 .
[4] H. Kakinuma,et al. Comparison of phosphonate transition state analogs for inducing catalytic antibodies and evaluation of key structural factors by an ab initio study , 1999 .
[5] M. Chelliah,et al. Synthesis of a Model Bicyclic CDE Ring System of Ristocetin A and Observation of a Facile Inversion of Configuration in a 16-Membered DE Ring Model , 1998 .
[6] Carol M. Taylor,et al. Phosphonate Diester and Phosphonamide Synthesis. Reaction Coordinate Analysis by 31P NMR Spectroscopy: Identification of Pyrophosphonate Anhydrides and Highly Reactive Phosphonylammonium Salts1 , 1997 .
[7] H. Krawczyk. A Convenient Route for Monodealkylation of Diethyl Phosphonates , 1997 .
[8] M. Meldal,et al. Azido Acids in a Novel Method of Solid-Phase Peptide Synthesis. , 1997 .
[9] Davidr . Evans,et al. Synthesis of the orienticin C M(2–4) macrocycle utilizing a nucleophilic aromatic substitution strategy , 1996 .
[10] K. Reddy,et al. SYNTHETIC STUDIES TOWARDS GLYCOPEPTIDE ANTIBIOTICS : SYNTHESIS OF THE 16-MEMBERED CYCLIC TRIPEPTIDE (DOEG RING) SYSTEM OF TEICOPLANIN , 1996 .
[11] Carol M. Taylor,et al. PHOSPHONYLTRIETHYLAMMONIUM SALTS : NOVEL REACTIVE SPECIES FOR THE SYNTHESIS OF PHOSPHONATE ESTERS AND PHOSPHONONAMIDES , 1995 .
[12] P. Savignac,et al. PREPARATION DE L'ACIDE AMINOMETHYLPHOSPHONIQUE α-DIDEUTERIE , 1995 .
[13] C. Mioskowski,et al. Selective Monodeprotection of Phosphate, Phosphite, Phosphonate, and Phosphoramide Benzyl Esters , 1995 .
[14] R. Crouch,et al. [[(Guaninylalkyl)phosphinico]methyl]phosphonic acids. Multisubstrate analogue inhibitors of human erythrocyte purine nucleoside phosphorylase. , 1995, Journal of medicinal chemistry.
[15] S. Shibuya,et al. Stereoselective Synthesis of .beta.-Oxygenated .alpha.-Hydroxyphosphonates by Lewis Acid-Mediated Stereoselective Hydrophosphonylation of .alpha.-Benzyloxy Aldehydes. An Application to the Synthesis of Phosphonic Acid Analogs of Oxyamino Acids , 1994 .
[16] W. Malachowski,et al. The Chemistry of Phosphapeptides: Investigations on the Synthesis of Phosphonamidate, Phosphonate, and Phosphinate Analogs of Glutamyl-.gamma.-glutamate , 1994 .
[17] W. Malachowski,et al. The Chemistry of Phosphapeptides: Formation of Functionalized Phosphonochloridates under Mild Conditions and Their Reaction with Alcohols and Amines , 1994 .
[18] L. Moroder,et al. On the Synthesis of Phosphonamidate Peptides , 1994 .
[19] D. Payne,et al. The synthesis and serine β-lactamase inhibitory activity of some phosphonamidate analogues of dipeptides , 1994 .
[20] A. J. Pearson,et al. Synthesis of a 14-Membered Cyclic Peptide Model of the CFG Rings of Ristocetin A and Observations on Atropdiastereoisomerism , 1994 .
[21] H. Cristau,et al. The preparation of phosphono peptides containing a phosphonamidate bond , 1994 .
[22] P. Hawkins,et al. Synthesis of stereochemically defined phosphonamidate-containing peptides: Inhibitors for the HIV-1 proteinase , 1992 .
[23] R. Hoffman,et al. Preparation of (R)-2-azidoesters from 2-((p-nitrobenzene)sulfonyl)oxy esters and their use as protected amino acid equivalents for the synthesis of di- and tripeptides containing d-amino acid constituents , 1992 .
[24] A. J. Pearson,et al. Model studies on the synthesis of carboxylate-binding pocket analogs of vancomycin using arene-ruthenium chemistry , 1992 .
[25] S. Shibuya,et al. Enantioselective synthesis of α-amino phosphonic acids by an application of stereoselective opening of homochiral dioxane acetals with triethyl phosphite , 1992 .
[26] P. Wirsching,et al. Phosphonamidates and phosphonamidate esters as HIV-1 protease inhibitors , 1991 .
[27] J. Hanson,et al. Potent inhibition of pepsin and penicillopepsin by phosphorus-containing peptide analogues , 1990 .
[28] Davidr . Evans,et al. The asymmetric synthesis of .alpha.-amino acids. Electrophilic azidation of chiral imide enolates, a practical approach to the synthesis of (R)- and (S)-.alpha.-azido carboxylic acids , 1990 .
[29] Davidr . Evans,et al. The total syntheses of the isodityrosine-derived cyclic tripeptides OF4949-III and K-13. Determination of the absolute configuration of K-13 , 1989 .
[30] N. Sampson,et al. Synthesis of phosphonic acid derivatives by oxidative activation of phosphinate esters , 1988 .
[31] P. Bartlett,et al. Phosphorus amino acid analogues as inhibitors of leucine aminopeptidase. , 1987, Journal of medicinal chemistry.
[32] F. Goffic,et al. Towards new inhibitors of D-alanine:D-alanine ligase: The synthesis of 3-amino butenylphosphonic and aminophosphonamidic acids. , 1987 .
[33] P. Portoghese,et al. Synthesis and biological evaluation of phosphonamidate peptide inhibitors of enkephalinase and angiotensin-converting enzyme. , 1985, Journal of medicinal chemistry.
[34] D. C. Roberts,et al. A new synthesis of peptides from azides and unactivated carboxylic acids , 1985 .
[35] I. Ojima,et al. Synthesis of chiral oligopeptides by means of catalytic asymmetric hydrogenation of dehydropeptides , 1984 .
[36] P. Bartlett,et al. A phosphonamidate dipeptide analog as an inhibitor of carboxypeptidase A , 1981 .
[37] J. Jacques,et al. La formation de sels augmente-t-elle la fréquence des dédoublements spontanés? , 1981 .
[38] M. D. Gray,et al. Selective demethylation of phosphorus esters , 1980 .
[39] K. Yamauchi,et al. Peptides Containing Aminophosphonic Acids. III. The Synthesis of Tripeptide Analogs Containing Aminomethylphosphonic Acid , 1975 .
[40] M. Hariharan,et al. Synthesis of Phosphonopeptide Derivatives , 1974 .
[41] K. Yamauchi,et al. Peptides Containing Aminophosphonic Acids. II. The Synthesis of Tripeptide Analogs , 1972 .
[42] K. Yamauchi,et al. Peptides Containing Aminophosphonic Acids. I. Reactivity of α-Aminobenzylphosphonic Acid , 1972 .