Radiolabeled CCK/gastrin peptides for imaging and therapy of CCK2 receptor-expressing tumors
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Otto C. Boerman | Peter Laverman | O. Boerman | F. V. van Delft | P. Laverman | S. Roosenburg | Susan Roosenburg | Floris L. van Delft
[1] E. Krenning,et al. Cholecystokinin receptor imaging using an octapeptide DTPA-CCK analogue in patients with medullary thyroid carcinoma , 2000, European Journal of Nuclear Medicine.
[2] R. Valkema,et al. Preclinical and initial clinical evaluation of 111In-labeled nonsulfated CCK8 analog: a peptide for CCK-B receptor-targeted scintigraphy and radionuclide therapy. , 1999, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[3] J. Erion,et al. Unsulfated DTPA- and DOTA-CCK analogs as specific high-affinity ligands for CCK-B receptor-expressing human and rat tissues in vitro and in vivo , 1998, European Journal of Nuclear Medicine.
[4] W. Oyen,et al. Improved tumour detection by gastrin receptor scintigraphy in patients with metastasised medullary thyroid carcinoma , 2006, European Journal of Nuclear Medicine and Molecular Imaging.
[5] W. Oyen,et al. Stabilized (111)in-labeled sCCK8 analogues for targeting CCK2-receptor positive tumors: synthesis and evaluation. , 2010, Bioconjugate chemistry.
[6] W. Oyen,et al. Targeting of a CCK(2) receptor splice variant with (111)In-labelled cholecystokinin-8 (CCK8) and (111)In-labelled minigastrin. , 2008, European journal of nuclear medicine and molecular imaging.
[7] H. Hellmich,et al. Human Colorectal Cancers Express a Constitutively Active Cholecystokinin-B/Gastrin Receptor That Stimulates Cell Growth* , 2000, The Journal of Biological Chemistry.
[8] W. Oyen,et al. Synthesis and biological evaluation of potent alphavbeta3-integrin receptor antagonists. , 2006, Nuclear medicine and biology.
[9] S. Snyder,et al. Distinct cholecystokinin receptors in brain and pancreas. , 1980, Proceedings of the National Academy of Sciences of the United States of America.
[10] N. Iwata,et al. Cholecystokinin-B/gastrin receptor: a novel molecular probe for human small cell lung cancer. , 1995, Cancer research.
[11] L. F. Kolakowski,et al. Expression cloning and characterization of the canine parietal cell gastrin receptor. , 1992, Proceedings of the National Academy of Sciences of the United States of America.
[12] J. Vanderhaeghen,et al. New peptide in the vertebrate CNS reacting with antigastrin antibodies , 1975, Nature.
[13] J C Reubi,et al. Cholecystokinin(CCK)-A and CCK-B/gastrin receptors in human tumors. , 1997, Cancer research.
[14] I. Zagon,et al. Characterization of the CCK-C (cancer) receptor in human pancreatic cancer. , 2002, International journal of molecular medicine.
[15] T. Wheldon,et al. Relationships between tumor size and curability for uniformly targeted therapy with beta-emitting radionuclides. , 1995, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[16] M. Béhé,et al. Cholecystokinin-B/Gastrin receptor-targeting peptides for staging and therapy of medullary thyroid cancer and other cholecystokinin-B receptor-expressing malignancies. , 2002, Seminars in nuclear medicine.
[17] B. Roques,et al. CCK-B receptor: chemistry, molecular biology, biochemistry and pharmacology , 1999, Progress in Neurobiology.
[18] E. Krenning,et al. Comparison of three radiolabelled peptide analogues for CCK-2 receptor scintigraphy in medullary thyroid carcinoma , 2009, European Journal of Nuclear Medicine and Molecular Imaging.
[19] M. Béhé,et al. CCK-2/gastrin receptor-targeted tumor imaging with (99m)Tc-labeled minigastrin analogs. , 2005, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[20] M. Ocak,et al. Cyclic minigastrin analogues for gastrin receptor scintigraphy with technetium-99m: preclinical evaluation. , 2009, Journal of medicinal chemistry.
[21] J C Reubi,et al. Unexpected high incidence of cholecystokinin‐B/gastrin receptors in human medullary thyroid carcinomas , 1996, International journal of cancer.
[22] U. Haberkorn,et al. (68)Ga-labeled peptides in tumor imaging. , 2005, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[23] W. Oyen,et al. Targeting of a CCK2 receptor splice variant with 111In-labelled cholecystokinin-8 (CCK8) and 111In-labelled minigastrin , 2008, European Journal of Nuclear Medicine and Molecular Imaging.
[24] Roland Haubner,et al. αvβ3-integrin imaging: a new approach to characterise angiogenesis? , 2006, European Journal of Nuclear Medicine and Molecular Imaging.
[25] J. Fichna,et al. Synthesis of target-specific radiolabeled peptides for diagnostic imaging. , 2003, Bioconjugate chemistry.
[26] Michele Saviano,et al. Conformationally Constrained CCK8 Analogues Obtained from a Rationally Designed Peptide Library as Ligands for Cholecystokinin Type B Receptor , 2006, ChemMedChem.
[27] Pomila Singh,et al. Clinical significance of gastrin receptors in human colon cancers. , 1989, Cancer research.
[28] W. Oyen,et al. Two technetium-99m-labeled cholecystokinin-8 (CCK8) peptides for scintigraphic imaging of CCK receptors. , 2004, Bioconjugate chemistry.
[29] A. Ivy,et al. A HORMONE MECHANISM FOR GALL-BLADDER CONTRACTION AND EVACUATION , 1928 .
[30] M. Walter,et al. Macrocyclic chelator-coupled gastrin-based radiopharmaceuticals for targeting of gastrin receptor-expressing tumours , 2008, European Journal of Nuclear Medicine and Molecular Imaging.
[31] J. Hughes,et al. Cholecystokinin receptors , 2005, Cellular and Molecular Neurobiology.
[32] L. Miller,et al. CCK2 receptor splice variant with intron 4 retention in human gastrointestinal and lung tumours , 2009, Journal of cellular and molecular medicine.
[33] M. Salvatore,et al. In vitro and in vivo evaluation of 111In-DTPAGlu-G-CCK8 for cholecystokinin-B receptor imaging. , 2004, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[34] M. Béhé,et al. Targeting of cholecystokinin-B/gastrin receptors in vivo: preclinical and initial clinical evaluation of the diagnostic and therapeutic potential of radiolabelled gastrin , 1998, European Journal of Nuclear Medicine.
[35] J Nucl Med , 2010 .
[36] J. Williams,et al. Binding of cholecystokinin to high affinity receptors on isolated rat pancreatic acini. , 1980, The Journal of biological chemistry.
[37] S. Wank,et al. G protein-coupled receptors in gastrointestinal physiology. I. CCK receptors: an exemplary family. , 1998, The American journal of physiology.
[38] M. Salvatore,et al. In vitro and in vivo characterization of Indium-111 and Technetium-99m labeled CCK-8 derivatives for CCK-B receptor imaging. , 2004, Cancer biotherapy & radiopharmaceuticals.
[39] M. Béhé,et al. Radiolabeled peptides for targeting cholecystokinin-B/gastrin receptor-expressing tumors. , 1999, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[40] M. Béhé,et al. Cholecystokinin-B (CCK-B)/gastrin receptor targeting peptides for staging and therapy of medullary thyroid cancer and other CCK-B receptor expressing malignancies. , 2002, Biopolymers.
[41] M. Béhé,et al. Use of polyglutamic acids to reduce uptake of radiometal-labeled minigastrin in the kidneys. , 2005, Journal of nuclear medicine : official publication, Society of Nuclear Medicine.
[42] S. Wank. I. CCK receptors: an exemplary family. , 1998, American journal of physiology. Gastrointestinal and liver physiology.
[43] O. Boerman,et al. Synthesis and biological evaluation of potent a v h 3 -integrin receptor antagonists , 2006 .
[44] S. Watson,et al. Selection of Radiolabeled Gastrin Analogs for Peptide Receptor–Targeted Radionuclide Therapy , 2007, Journal of Nuclear Medicine.
[45] G. Baldwin,et al. Expression of gastrin, gastrin/CCK-B and gastrin/CCK-C receptors in human colorectal carcinomas , 2005, Journal of Cancer Research and Clinical Oncology.
[46] E. Krenning,et al. Optimised labeling, preclinical and initial clinical aspects of CCK-2 receptor-targeting with 3 radiolabeled peptides. , 2008, Nuclear medicine and biology.
[47] R. Haubner. Alphavbeta3-integrin imaging: a new approach to characterise angiogenesis? , 2006, European journal of nuclear medicine and molecular imaging.
[48] J. Crawley,et al. International Union of Pharmacology. XXI. Structure, distribution, and functions of cholecystokinin receptors. , 1999, Pharmacological reviews.
[49] B. Maigret,et al. Insights into the binding and activation sites of the receptors for cholecystokinin and gastrin , 2008, Regulatory Peptides.
[50] M. Béhé,et al. Improved kinetic stability of DTPA-dGlu as compared with conventional monofunctional DTPA in chelating indium and yttrium: preclinical and initial clinical evaluation of radiometal labelled minigastrin derivatives , 2003, European Journal of Nuclear Medicine and Molecular Imaging.