Novel nicotine analogues with potential anti-mycobacterial activity.
暂无分享,去创建一个
[1] J. Sacchettini,et al. The identification of novel Mycobacterium tuberculosis DHFR inhibitors and the investigation of their binding preferences by using molecular modelling , 2015, Scientific Reports.
[2] M. Files,et al. Synthesis and anti-tubercular activity of 3-substituted benzo[b]thiophene-1,1-dioxides , 2014, PeerJ.
[3] Marvin J. Miller,et al. Bactericidal Activity of an Imidazo[1, 2-a]pyridine Using a Mouse M. tuberculosis Infection Model , 2014, PloS one.
[4] V. Bernardes-Génisson,et al. Isoniazid: an update on the multiple mechanisms for a singular action. , 2013, Current medicinal chemistry.
[5] D. Sherman,et al. Identification of New Drug Targets and Resistance Mechanisms in Mycobacterium tuberculosis , 2013, PloS one.
[6] P. Yogeeswari,et al. Design, synthesis, and structure-activity correlations of novel dibenzo[b,d]furan, dibenzo[b,d]thiophene, and N-methylcarbazole clubbed 1,2,3-triazoles as potent inhibitors of Mycobacterium tuberculosis. , 2012, Journal of medicinal chemistry.
[7] S. Loewenberg. India reports cases of totally drug-resistant tuberculosis , 2012, The Lancet.
[8] C. Evans,et al. A new era for global tuberculosis control , 2011, The Lancet.
[9] J. Maurice. WHO framework targets tuberculosis–diabetes link , 2011, The Lancet.
[10] L. Dover,et al. Current status and research strategies in tuberculosis drug development. , 2011, Journal of medicinal chemistry.
[11] A. Tyagi,et al. Identification of Inhibitors against Mycobacterium tuberculosis Thiamin Phosphate Synthase, an Important Target for the Development of Anti-TB Drugs , 2011, PloS one.
[12] A. Ginsberg. Drugs in Development for Tuberculosis , 2010, Drugs.
[13] Antoine Taly,et al. Nicotinic receptors: allosteric transitions and therapeutic targets in the nervous system , 2009, Nature Reviews Drug Discovery.
[14] Lynn Rasmussen,et al. High-throughput screening for inhibitors of Mycobacterium tuberculosis H37Rv. , 2009, Tuberculosis.
[15] Sandeep Jain,et al. Synthesis and in-vitro antibacterial activity of some novel N-nicotinoyl-1-ethyl-6-fluoro-1,4-dihydro-7-piperazin-1-yl-4-oxoquinoline-3-carboxylates. , 2008, Acta poloniae pharmaceutica.
[16] W. Denny,et al. A roadmap for drug discovery and its translation to small molecule agents in clinical development for tuberculosis treatment. , 2008, Tuberculosis.
[17] Mohamed M. Abdulla,et al. Anti-inflammatory and analgesic activities of some newly synthesized pyridinedicarbonitrile and benzopyranopyridine derivatives , 2008, Acta pharmaceutica.
[18] V. Choubey,et al. Antiplasmodial Activity of [(Aryl)arylsulfanylmethyl]Pyridine , 2007, Antimicrobial Agents and Chemotherapy.
[19] Yves L Janin,et al. Antituberculosis drugs: ten years of research. , 2007, Bioorganic & medicinal chemistry.
[20] J. Nowakowski,et al. Antimicrobial activity of nicotine against a spectrum of bacterial and fungal pathogens. , 2000, Journal of medical microbiology.
[21] I. Sinha,et al. Differentiation of non-pathogenic (biotype 1A) Yersinia enterocolitica from pathogenic bioserotypes by sodium acetate utilisation. , 2000, Journal of medical microbiology.
[22] L. Collins,et al. Microplate alamar blue assay versus BACTEC 460 system for high-throughput screening of compounds against Mycobacterium tuberculosis and Mycobacterium avium , 1997, Antimicrobial agents and chemotherapy.
[23] N. Benowitz,et al. Metabolism of nicotine to cotinine studied by a dual stable isotope method , 1994, Clinical pharmacology and therapeutics.
[24] M. Shigenaga,et al. Metabolism-dependent covalent binding of (S)-[5-3H]nicotine to liver and lung microsomal macromolecules. , 1988, Drug metabolism and disposition: the biological fate of chemicals.
[25] James C. Sacchettini,et al. Drugs versus bugs: in pursuit of the persistent predator Mycobacterium tuberculosis , 2008, Nature Reviews Microbiology.
[26] D. Donnelly-roberts,et al. Stable expression, pharmacologic properties and regulation of the human neuronal nicotinic acetylcholine alpha 4 beta 2 receptor. , 1996, The Journal of pharmacology and experimental therapeutics.