A Novel One-Pot Synthesis of N,N-Dimethylaminopyridines by Diazotization of Aminopyridines in Dimethylformamide in the Presence of Trifluoromethanesulfonic Acid

[1]  H. Gong,et al.  Amination of Aromatic Halides and Exploration of the Reactivity Sequence of Aromatic Halides. , 2018, The Journal of organic chemistry.

[2]  E. Krasnokutskaya,et al.  Pyridinyl trifluoromethanesulfonates: preparation methods and use in organic synthesis , 2016, Russian Chemical Bulletin.

[3]  Jacob P. Sorrentino,et al.  General method for nucleophilic aromatic substitution of aryl fluorides and chlorides with dimethylamine using hydroxide-assisted decomposition of N,N-dimethylforamide , 2016, Synthetic communications.

[4]  M. Mesleh,et al.  Discovery of Pyrazolopyridones as a Novel Class of Gyrase B Inhibitors Using Structure Guided Design. , 2016, ACS medicinal chemistry letters.

[5]  E. Krasnokutskaya,et al.  A Novel Convenient Synthesis of Pyridinyl and Quinolinyl Triflates and Tosylates via One-Pot Diazotization of Aminopyridines and Aminoquinolines in Solution , 2015, Synthesis.

[6]  Yao Fu,et al.  Boron-Catalyzed N-Alkylation of Amines using Carboxylic Acids. , 2015, Angewandte Chemie.

[7]  Zhu Xiaoming,et al.  Room‐Temperature Copper‐Catalyzed Arylation of Dimethylamine and Methylamine in Neat Water , 2015 .

[8]  E. Krasnokutskaya,et al.  A new synthesis of pyridinyl trifluoromethanesulfonates via one-pot diazotization of aminopyridines in the presence of trifluoromethanesulfonic acid , 2014 .

[9]  T. Kurahashi,et al.  Palladium Porphyrin Catalyzed Hydrogenation of Alkynes: Stereoselective Synthesis of cis-Alkenes , 2014, Synlett.

[10]  Jianliang Xiao,et al.  A general method for N-methylation of amines and nitro compounds with dimethylsulfoxide. , 2014, Chemistry.

[11]  T. Mita,et al.  Iridium- and rhodium-catalyzed dehydrogenative silylations of C(sp3)-H bonds adjacent to a nitrogen atom using hydrosilanes. , 2013, Chemistry, an Asian journal.

[12]  P. R. Rajamohanan,et al.  Transition-metal-free multicomponent reactions involving arynes, N-heterocycles, and isatins. , 2013, Angewandte Chemie.

[13]  A. Ritzén,et al.  Continuous flow nucleophilic aromatic substitution with dimethylamine generated in situ by decomposition of DMF. , 2013, The Journal of organic chemistry.

[14]  Lixiong Shao,et al.  N-heterocyclic carbene-palladium(II)-1-methylimidazole complex catalyzed amination between aryl chlorides and amides. , 2012, The Journal of organic chemistry.

[15]  Abdelouahid Samadi,et al.  Microwave Irradiation–Assisted Amination of 2-Chloropyridine Derivatives with Amide Solvents , 2011 .

[16]  M. Stradiotto,et al.  A highly versatile catalyst system for the cross-coupling of aryl chlorides and amines. , 2010, Chemistry.

[17]  C. E. Allen,et al.  Identification and characterisation of 2-aminopyridine inhibitors of checkpoint kinase 2. , 2010, Bioorganic & medicinal chemistry.

[18]  A. Gomtsyan,et al.  4-amino-5-aryl-6-arylethynylpyrimidines: structure-activity relationships of non-nucleoside adenosine kinase inhibitors. , 2007, Bioorganic & medicinal chemistry.

[19]  Xin-jun Liu,et al.  Design of 2,5-dimethyl-3-(6-dimethyl-4-methylpyridin-3-yl)-7-dipropylaminopyrazolo[1,5-a]pyrimidine (NBI 30775/R121919) and structure--activity relationships of a series of potent and orally active corticotropin-releasing factor receptor antagonists. , 2004, Journal of medicinal chemistry.

[20]  G. Kalayanov,et al.  Regioselective Functionalization of Guanine: Simple and Practical Synthesis of 7- and 9-Alkylated Guanines Starting from Guanosine , 2004 .

[21]  M. Sanford,et al.  Palladium-catalyzed oxygenation of unactivated sp3 C-H bonds. , 2004, Journal of the American Chemical Society.

[22]  A. Steiger,et al.  Treatment with the CRH1-receptor-antagonist R121919 improves sleep-EEG in patients with depression. , 2004, Journal of psychiatric research.

[23]  A. Agarwal,et al.  Convenient Dimethylamino Amination in Heterocycles and Aromatics with Dimethylformamide , 2004 .

[24]  J. C. Park,et al.  A very convenient dimethylamination of activated aromatic halides using N,N-dimethylformamide and ethanolamines , 1997 .

[25]  M. Jovanovic,et al.  Bromination of some pyridine and diazine N-oxides , 1983 .

[26]  I. S. Kashparov,et al.  N-anions of heteroaromatic amines , 1971 .

[27]  M. Pal,et al.  A simple synthesis of aminopyridines: use of amides as amine source , 2010 .

[28]  B. Feringa,et al.  Encyclopedia Reagents in organic synthesis , 1995 .

[29]  A. Katritzky,et al.  The kinetics and mechanism of the electrophilic substitution of heteroaromatic compounds. Part XXV. The acid-catalysed hydrogen-exchange of some 2-aminopyridine derivatives , 1971 .

[30]  W. Awe,et al.  Untersuchungen in der 2‐Aminopyridinreihe IV1,2). Untersuchungen über die Reaktionsfähigkeit der Methylgruppe im 2‐Methyl‐6‐aminopyridin , 1936 .