An efficient and highly stereoselective synthesis of novel trifluoromethylated trans-dihydrofuro[2,3-c]pyrazoles using arsonium ylides

[1]  Jianwei Han,et al.  Facile synthesis of novel CF3-substituted ring-fused furo[2,3-c]pyrazoles through Rh2(OAc)4 catalyzed [3+2] cycloaddition of 4-diazo-1-phenyl-3-(trifluoromethyl)-1H-pyrazol-5(4H)-one with aromatic alkynes , 2011 .

[2]  Xiaolan Fu,et al.  Divergent synthesis of fully substituted isoxazoles and spiro-fused pyrazolin-5-ones from cyclopropyl oximes , 2011 .

[3]  K. Atta,et al.  Annulation and evaluation of antibacterial activity of the new fused tricyclic (5,5,6) ring system of pyrazolo〔1,5-c〕-1,2,4-triazolo〔4,3-a〕pyrimidines , 2011 .

[4]  S. Bondock,et al.  Synthesis and antimicrobial activity of some new 4-hetarylpyrazole and furo[2,3-c]pyrazole derivatives. , 2011, European journal of medicinal chemistry.

[5]  Masaharu Nakayama,et al.  Synthesis of a novel series of tricyclic dihydrofuran derivatives: discovery of 8,9-dihydrofuro[3,2-c]pyrazolo[1,5-a]pyridines as melatonin receptor (MT1/MT2) ligands. , 2011, Journal of medicinal chemistry.

[6]  W. Cao,et al.  First one-pot stereoselective synthesis of cis-2,3-dihydro-4-perfluoroalkyl-1H-1,5-benzodiazepines via a catalyst-free three-component reaction. , 2011, Chemical communications.

[7]  Hyunik Shin,et al.  Recent Advances in the Regioselective Synthesis of Pyrazoles , 2011 .

[8]  M. Franchini,et al.  Regiocontrolled Synthesis of Ring‐Fused Thieno[2,3‐c]pyrazoles through 1,3‐Dipolar Cycloaddition of Nitrile Imines with Sulfur‐Based Acetylenes , 2010 .

[9]  M. Christodoulou,et al.  Novel pyrazole derivatives: synthesis and evaluation of anti-angiogenic activity. , 2010, Bioorganic & medicinal chemistry.

[10]  J. Mousseau,et al.  Synthesis of 2-substituted pyrazolo[1,5-a]pyridines through cascade direct alkenylation/cyclization reactions. , 2010, Organic letters.

[11]  H. Amada,et al.  Ring-fused pyrazole derivatives as potent inhibitors of lymphocyte-specific kinase (Lck): Structure, synthesis, and SAR. , 2010, Bioorganic & medicinal chemistry letters.

[12]  W. Cao,et al.  A simple and convenient synthesis of 2-(perfluoroalkyl)-4H-chromenes from salicyl N-tosylimines or salicylaldehydes and methyl 2-perfluoroalkynoates , 2009 .

[13]  H. Alper,et al.  Synthesis of ring-fused oxazolo- and pyrazoloisoquinolinones by a one-pot Pd-catalyzed carboxamidation and aldol-type condensation cascade process. , 2009, The Journal of organic chemistry.

[14]  W. Cao,et al.  A facile stereoselective synthesis of 2-perfluoroalkyl-3a,4,5, 6-tetrahydroimidazo[ 1,5-b]isoxazoles , 2009 .

[15]  A. Ponti,et al.  Enantiopure furo[3,4-c]pyrazole derivatives by intramolecular nitrilimine cycloaddition: a stereoselectivity rationale based upon MP2 calculations , 2008 .

[16]  P. Pohlhaus,et al.  Scope and mechanism for lewis acid-catalyzed cycloadditions of aldehydes and donor-acceptor cyclopropanes: evidence for a stereospecific intimate ion pair pathway. , 2008, Journal of the American Chemical Society.

[17]  Zhongjiao Ren,et al.  Highly stereoselective construction of spiro[cyclopropane-1,4′-pyrazolin-5′-one]with 4-arylidene-3-methyl-1-phenyl-pyrazolin-5-one and arsonium ylide , 2008 .

[18]  S. Laufer,et al.  Three-component combinatorial synthesis of novel dihydropyrano[2,3-c]pyrazoles. , 2008, Journal of combinatorial chemistry.

[19]  S. Kim,et al.  A novel and efficient one-pot synthesis of furo[3′,4′:5,6]pyrido[2,3-c]pyrazole derivatives using organocatalysts , 2008 .

[20]  W. Cao,et al.  Highly stereoselective synthesis of cyclopropyl heterocycles via cyclopropanation of olefin with arsonium salt , 2008 .

[21]  W. Cao,et al.  Stereoselective synthesis of highly substituted trans -2,3-dihydrofuran and trans -1,2-cyclopropane derivatives containing sulfonyl groups , 2008 .

[22]  S. Rogelj,et al.  Discovery and investigation of antiproliferative and apoptosis-inducing properties of new heterocyclic podophyllotoxin analogues accessible by a one-step multicomponent synthesis. , 2007, Journal of medicinal chemistry.

[23]  S. Ji,et al.  Synthesis of pyrazolo[1,5-a]indoles via copper(I)-catalyzed intramolecular amination , 2007 .

[24]  Shizheng Zhu,et al.  A novel and facile synthesis of 2,3-dihydrofuran derivatives containing trifluoromethyl group , 2007 .

[25]  S. Gogoi,et al.  A facile two-step chemoenzymatic access to natural germination inhibitor (+)-erigeronic acid A , 2006 .

[26]  P. Toy,et al.  Polystyrene-supported triphenylarsines: useful ligands in palladium-catalyzed aryl halide homocoupling reactions and a catalyst for alkene epoxidation using hydrogen peroxide , 2005 .

[27]  P. Toy,et al.  Arsonium ylides in organic synthesis , 2005 .

[28]  Ming‐Shiuan Yu,et al.  Recent advances in donor-acceptor (DA) cyclopropanes , 2005 .

[29]  Shizheng Zhu,et al.  Unexpected formation of tetrasubstituted 2,3-dihydrofurans from the reactions of beta-keto polyfluoroalkanesulfones with aldehydes. , 2004, The Journal of organic chemistry.

[30]  L. Toupet,et al.  Synthesis of trifluoromethylated pyrazoles from trifluoromethylenaminones and monosubstituted hydrazines , 2004 .

[31]  W. Cao,et al.  Stereoselective Synthesis of cis‐1‐Aryl‐2‐benzoyl‐3,3‐dicyanocyclopropanes in the Presence of KF·2H2O , 2004 .

[32]  A. IJzerman,et al.  Pyrazole derivatives as partial agonists for the nicotinic acid receptor. , 2003, Journal of medicinal chemistry.

[33]  R. Zimmer,et al.  Donor-acceptor-substituted cyclopropane derivatives and their application in organic synthesis. , 2003, Chemical reviews.

[34]  A. Skaltsounis,et al.  Design, synthesis, and antiproliferative activity of some new pyrazole-fused amino derivatives of the pyranoxanthenone, pyranothioxanthenone, and pyranoacridone ring systems: a new class of cytotoxic agents. , 2002, Journal of medicinal chemistry.

[35]  Toshio Suzuki,et al.  Domino Michael–O-alkylation reaction: one-pot synthesis of 2,4-diacylhydrofuran derivatives and its application to antitumor naphthofuran synthesis , 2001 .

[36]  J. Garrido,et al.  One-Step Palladium-Catalyzed Synthesis of Substituted Dihydrofurans from the Carbonate Derivatives of γ-Hydroxy-α,β-unsaturated Sulfones , 1998 .

[37]  S. Schabbert,et al.  Palladium-Catalyzed Cyclization of Silyl-Substituted Bis(homo)propargylic Alcohols to 2,3-Dihydrofurans , 1998 .

[38]  Alan R. Katritzky,et al.  Comprehensive Heterocyclic Chemistry IV , 1996 .

[39]  M. Rizzacasa,et al.  Convergent synthesis of polyether ionophore antibiotics: protective manipulation and synthesis of monensin A , 1993 .

[40]  K. Nicolaou,et al.  Total synthesis of hemibrevetoxin B and (7a.alpha.)-epi-hemibrevetoxin B , 1993 .

[41]  R. K. Boeckman,et al.  The chemistry of cyclic vinyl ethers. 6. Total synthesis of polyether ionophore antibiotics of the calcimycin (A-23187) class , 1991 .

[42]  T. Hudlický,et al.  Use of cyclopropanes and their derivatives in organic synthesis , 1989 .

[43]  H. Reissig Donor-acceptor-substituted cyclopropanes: versatile building blocks in organic synthesis , 1988 .

[44]  D. Lloyd,et al.  Arsonium ylides (with some mention also of arsinimines, stibonium and bismuthonium ylides) , 1987 .

[45]  B. Lipshutz Five-membered heteroaromatic rings as intermediates in organic synthesis , 1986 .

[46]  P. Schuda Aflatoxin chemistry and syntheses , 1980 .