Studies on chalcogen-containing heterocycles. Part 38: Regio- and stereoselective tandem addition–iodocyclization of 2-ethynylphenyl isothiocyanates with N- and O-nucleophiles affording 4-(iodoalkylidene)benzo[ d ][1,3]thiazines

[1]  M. Minoura,et al.  Studies on chalcogen-containing heterocycles. Part 37: m-CPBA oxidation of isotellurochromenes and isoselenochromenes , 2012 .

[2]  Yiyuan Peng,et al.  Access to functionalized 4-benzylidene-4H-benzo[d][1,3]thiazines via tandem addition-cyclization/cross-coupling reactions , 2012 .

[3]  H. Sashida,et al.  Tandem addition–cyclization of o-ethynylphenyl isothiocyanates with N nucleophiles; difference of cyclization mode between primary and secondary amines☆ , 2012 .

[4]  H. Sashida,et al.  RAPID ONE-POT VERSATILE PREPARATION OF 2-AMINOBENZO-THIAZOLES BY HIGHLY EFFICIENT COPPER(I)-CATALYZED INORGANIC BASE-FREE INTRAMOLECULAR CYCLIZATION (Dedicated to Dr. Albert Padwa on his 75th birthday) , 2012 .

[5]  P. Zhong,et al.  Metal-free synthesis of 3-chalcogen benzo[b]furans via an iodine-mediated electrophilic cyclisation of 2-alkynylanisoles , 2011 .

[6]  H. Sashida Preparations of selenium-containing heterocycles based on an intramolecular cyclization of selenols and relatives , 2011 .

[7]  Jie Wu,et al.  Synthesis of 4-methylene-4H-benzo[d][1,3]thiazines via a tandem reaction of 1-(2-alkynylphenyl)ketoximes with Lawesson's reagent. , 2011, Chemical communications.

[8]  H. Sashida,et al.  Tandem addition–cyclization of o-ethynylphenyllithiums and isoselenocyanates: a convenient preparation of functionalized benzo[c]selenophenes , 2011 .

[9]  K. Okuma,et al.  Synthesis of 3,1-benzothiazines from 2-alkenyl- and 2-alkynylanilides and lawesson reagent , 2011 .

[10]  A. K. Banerjee,et al.  Iodocyclization: Past and Present Examples , 2011 .

[11]  Benhur Godoi,et al.  Synthesis of heterocycles via electrophilic cyclization of alkynes containing heteroatom. , 2011, Chemical reviews.

[12]  M. Minoura,et al.  One-pot copper-catalyzed tandem addition-cyclization of 2-iodoanilines with isoselenocyanates for the practical preparation of 2-aminobenzoselenazoles , 2011 .

[13]  Benhur Godoi,et al.  Electrophilic cyclization of 3-alkynyl-4-chalcogen-2-H-chromenes: synthesis of 3-halo-chalcogenophene[3,2-c]chromene derivatives , 2011 .

[14]  Huanfeng Jiang,et al.  Synthesis of 2,5-disubstituted 3-iodofurans via palladium-catalyzed coupling and iodocyclization of terminal alkynes. , 2011, The Journal of organic chemistry.

[15]  H. Sashida,et al.  Tin-tellurium exchange reaction in tin-containing heterocycles: a new entry for the preparation of tellurium heterocycles , 2010 .

[16]  C. Cho,et al.  A new approach to desketoraloxifene analogs from oxygen-bearing 3-iodobenzo[b]thiophenes prepared via iodocyclization. , 2010, Tetrahedron letters.

[17]  M. Minoura,et al.  Regioselective electrophilic cyclization of o-ethynylbenzyl phenyl selenides to (Z)-1-methylidene-2-phenyl-1,3-dihydro-1H-benzo[c]selenophenium salts ☆ , 2010 .

[18]  M. Minoura,et al.  A Facile and Practical Solvent-FreeOne-Pot Synthesis of (Z)-4-Methylene-3-selenaquinolineDerivatives from o-Ethynylanilines andIsoselenocyanates¹ , 2010 .

[19]  M. Minoura,et al.  A straightforward double intramolecular cyclization of dibenzyl dichalcogenols into a triple bond , 2010 .

[20]  Yiyuan Peng,et al.  Silica gel-promoted tandem addition-cyclization reactions of 2-alkynylbenzenamines with isothiocyanates. , 2010, Journal of combinatorial chemistry.

[21]  M. Minoura,et al.  2-substituted isotellurochromenium salt derivatives: preparations, structures, spectroscopic properties , 2010 .

[22]  H. Sashida,et al.  Novel Oxidative Ring Opening Reaction of 1H-Isotelluro-chromenes to Bis(o-formylstyryl) Ditellurides , 2010, Molecules.

[23]  M. Mphahlele Molecular Iodine-Mediated Cyclization of Tethered Heteroatom-Containing Alkenyl or Alkynyl Systems , 2009, Molecules.

[24]  A. V. Butin,et al.  Aryl Ring Migration Reactionin the Synthesis of 2,4-Diaryl-4H-3,1-benzothiazines , 2009 .

[25]  春喜 指田,et al.  1-ベンゾテルロピリリウム塩の化学:合成、構造および反応 , 2009 .

[26]  A. Vallribera,et al.  A straightforward synthesis of benzothiazines. , 2009, Organic letters.

[27]  H. Sashida,et al.  A New One-Pot Synthetic Methodfor Selenium-Containing Medium-Sized α,β-UnsaturatedCyclic Ketones , 2008 .

[28]  Jie Wu,et al.  A facile route to 2,4-dihydro-1H-benzo[d][1,3]thiazines via silver-catalyzed tandem addition-cyclization reactions. , 2008, Journal of combinatorial chemistry.

[29]  A. V. Butin,et al.  Synthesis of 2,4‐difuryl‐4H‐3,1‐benzothiazines via a furan ring migration reaction , 2008 .

[30]  J. Salminen,et al.  Novel β-lactam condensed 3-thiaquinolines: an efficient synthesis and structural characterization , 2008 .

[31]  M. S. Subhas,et al.  Copper‐Free Sonogashira Coupling of Acid Chlorides with Terminal Alkynes in the Presence of a Reusable Palladium Catalyst: An Improved Synthesis of 3‐Iodochromenones (=3‐Iodo‐4H‐1‐benzopyran‐4‐ones) , 2008 .

[32]  Takao Saito,et al.  Thiocarbonyl induced heterocumulenic Pauson-Khand type reaction: expedient synthetic method for thieno[2,3-b]indol-2-ones. , 2008, Chemical communications.

[33]  C. Luchese,et al.  Electrophilic cyclization of (Z)-selenoenynes: synthesis and reactivity of 3-iodoselenophenes. , 2007, The Journal of organic chemistry.

[34]  J. M. Babu,et al.  Regioselective construction of six-membered fused heterocyclic rings via Pd/C-mediated C–C coupling followed by iodocyclization strategy: a new entry to 2H-1,2-benzothiazine-1,1-dioxides , 2007 .

[35]  H. Sashida 1-Benzoselenopyrylium Salts and 1-Benzotelluropyrylium Salts: Preparations,Structures and Reactions , 2007 .

[36]  H. Togo,et al.  Synthetic Use of Molecular Iodine for Organic Synthesis , 2006 .

[37]  A. V. Butin,et al.  Aromatic ring transfer—a new synthesis of 2,4-diaryl-4H-3,1-benzothiazines , 2006 .

[38]  J. Matysiak Synthesis, antiproliferative and antifungal activities of some 2-(2,4-dihydroxyphenyl)-4H-3,1-benzothiazines. , 2006, Bioorganic & medicinal chemistry.

[39]  R. Larock,et al.  Synthesis of 2,3-disubstituted benzo[b]selenophenes via electrophilic cyclization. , 2006, The Journal of organic chemistry.

[40]  R. Larock,et al.  Synthesis of 3-iodoindoles by the Pd/Cu-catalyzed coupling of N,N-dialkyl-2-iodoanilines and terminal acetylenes, followed by electrophilic cyclization. , 2006, The Journal of organic chemistry.

[41]  R. Larock,et al.  Synthesis of 2,3-disubstituted benzo[b]furans by the palladium-catalyzed coupling of o-iodoanisoles and terminal alkynes, followed by electrophilic cyclization. , 2005, The Journal of organic chemistry.

[42]  F. Shibahara,et al.  Iodo-cyclization of N-Homoallyl Thioamides Leading to 2,4-Diaryl-5,6-dihydro-4H-1,3-thiazines , 2004 .

[43]  M. Schmittel,et al.  A New Facile Synthesis of exo-Methylene 3,1-Benzothiazines , 2004 .

[44]  B. Flynn,et al.  Iodine-induced reaction cascades for the rapid construction of variously substituted benzothiophenes. , 2003, Organic letters.

[45]  R. Larock,et al.  Synthesis of Isocoumarins and α-Pyrones via Electrophilic Cyclization , 2003 .

[46]  M. Trincado,et al.  IPy2BF4-promoted intramolecular addition of masked and unmasked anilines to alkynes: direct assembly of 3-iodoindole cores. , 2003, Angewandte Chemie.

[47]  G. Zanardi,et al.  Cascade radical reactions via alpha-(arylsulfanyl)imidoyl radicals: competitive [4 + 2] and [4 + 1] radical annulations of alkynyl isothiocyanates with aryl radicals. , 2003, The Journal of organic chemistry.

[48]  L. Mannina,et al.  Synthesis of 3-arylisocoumarins, including thunberginols A and B, unsymmetrical 3,4-disubstituted isocoumarins, and 3-ylidenephthalides via iodolactonization of methyl 2-ynylbenzoates or the corresponding carboxylic acids , 2003 .

[49]  R. Larock,et al.  Synthesis of isocoumarins and α-pyrones via iodocyclization , 2002 .

[50]  G. Fabrizi,et al.  Electrophilic cyclization of o-acetoxy- and o-benzyloxyalkynylpyridines: an easy entry into 2,3-disubstituted furopyridines. , 2002, Organic letters.

[51]  R. Larock,et al.  Synthesis of 2,3-disubstituted benzo[b]thiophenes via palladium-catalyzed coupling and electrophilic cyclization of terminal acetylenes. , 2002, The Journal of organic chemistry.

[52]  R. Larock,et al.  Synthesis of benzo[b]thiophenes by electrophilic cyclization , 2001 .

[53]  H. Sashida Preparations of Heterocycles by Intramolecular Cyclization of Tellurols and Related Compounds to a Triple Bond , 2001 .

[54]  L. Deck,et al.  Synthesis of derivatives of thiophene using methyl 2‐isothiocyanatobenzoate , 2001 .

[55]  E. Hamel,et al.  A novel palladium-mediated coupling approach to 2,3-disubstituted benzo(b)thiophenes and its application to the synthesis of tubulin binding agents. , 2001, Organic letters.

[56]  Hari,et al.  Rapid and efficient synthesis of 2-amino-4H-benzothiazines , 2000, Organic letters.

[57]  P. Molina,et al.  Intramolecular heteroconjugate addition of heterocumulenes to α,β-unsaturated carbonyl compounds promoted by the CS2/TBAF system , 2000 .

[58]  W. Szarek,et al.  Iodine in carbohydrate chemistry. , 2000, Advances in carbohydrate chemistry and biochemistry.

[59]  G. Fabrizi,et al.  A New Approach to 2,3-Disubstituted Benzo[b]furans from o-Alkynylphenols via 5-endo-dig-Iodocyclisation/Palladium-Catalysed Reactions , 1999 .

[60]  E. Kandeel,et al.  Synthesis and reactions of 4H‐3,1‐benzothiazines , 1999 .

[61]  A. V. Butin,et al.  o-Nitroaryl-bis(5-methylfur-2-yl)methanes as Versatile Synthons for the Synthesis of Nitrogen-Containing Heterocycles , 1997 .

[62]  T. Nishio Reaction of (1,ω)-N-Acylamino Alcohols with Lawesson's Reagent: Synthesis of Sulfur-Containing Heterocycles , 1997 .

[63]  O. Morgenstern,et al.  Untersuchungen zur Darstellung und Reaktivität c-anellierter Abkömmlinge des 1,3,4-Benzotriazepins und entsprechender Vorprodukte : N,N-verknüpfte Heterobicyclen aus Cyclischen Hydrazin-Derivaten. 12. Mitteilung , 1996 .

[64]  T. Nishio Sulfur-containing heterocycles derived by the reaction of hydroxy-amides and Lawesson's reagent , 1995 .

[65]  P. Creeke,et al.  Synthessi and elaboration of heterocycles via iodocyclisation of unsaturated thioureas , 1989 .

[66]  E. P. Papadopoulos,et al.  Synthesis of Derivatives of Pyrrole Using Methyl 2-Isothiocyanatobenzoate , 1984 .

[67]  E. P. Papadopoulos,et al.  Synthesis of 4(3H)-quinazolinones from derivatives of methyl 2-isothiocyanatobenzoate , 1982 .

[68]  F. M. Hamer,et al.  19. Thiazinocyanines. Part I. Carbocyanines containing the 2 : 4-benzthiazine nucleus , 1942 .