Discovery and activity of (1R,4S,6R)-N-[(1R)-2-[4-cyclohexyl-4-[[(1,1-dimethylethyl)amino]carbonyl]-1-piperidinyl]-1-[(4-fluorophenyl)methyl]-2-oxoethyl]-2-methyl-2-azabicyclo[2.2.2]octane-6-carboxamide (3, RY764), a potent and selective melanocortin subtype-4 receptor agonist.
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J. Metzger | D. Macintyre | L. V. D. van der Ploeg | C. Rosenblum | Howard Y. Chen | A. Patchett | R. Nargund | R. Tang | M. Wyvratt | C. Tamvakopoulos | R. Bakshi | W. Martin | T. Macneil | I. Sebhat | R. Kalyani | D. Weinberg | R. Stearns | Randy R Miller | D. Cashen | A. Vongs | Airu S. Chen | Z. Ye | A. Strack | K. Barakat | B. Palucki | Qianping Peng | Liangqin Guo | Patrick G Pollard | Aurawan Vongs