Discovery of 3-[2-(imidazo[1,2-b]pyridazin-3-yl)ethynyl]-4-methyl-N-{4-[(4-methylpiperazin-1-yl)methyl]-3-(trifluoromethyl)phenyl}benzamide (AP24534), a potent, orally active pan-inhibitor of breakpoint cluster region-abelson (BCR-ABL) kinase including the T315I gatekeeper mutant.
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Wei-Sheng Huang | Jan Romero | Shuangying Liu | Tomi K Sawyer | Dong Zou | T. Clackson | V. Rivera | T. Zhou | T. Sawyer | W. Shakespeare | N. Narasimhan | Frank Y Wang | Xiaotian Zhu | Frank Wang | Yaoyu Ning | Scott Wardwell | Qurish K. Mohemmad | Yihan Wang | John Iuliucci | Tim Clackson | Tianjun Zhou | R. Sundaramoorthi | David Wen | Chester A Metcalf | Ingrid Chen | Raji Sundaramoorthi | Jiwei Qi | Lisi Cai | Lois Commodore | Qihong Xu | Jeff Keats | Joseph T Snodgrass | Marc I Broudy | Karin Russian | Victor M Rivera | David C Dalgarno | William C Shakespeare | D. Dalgarno | R Mathew Thomas | Geetha Banda | Scott P Lentini | Sasmita Das | Narayana I Narasimhan | Qurish K Mohemmad | J. Iuliucci | Jan Romero | K. Russian | M. Broudy | L. Commodore | Wei-sheng Huang | Yihan Wang | Xiaotian Zhu | C. Metcalf | Shuangying Liu | J. Keats | Scott D. Wardwell | Y. Ning | Sasmita Das | S. Lentini | R. Thomas | Qihong Xu | Jiwei Qi | D. Zou | Lisi Cai | Geetha Banda | David Wen | I. Chen | Frank Y. Wang | J. Romero | Tianjun Zhou