Synthesis and biological evaluation studies of novel quinazolinone derivatives as antibacterial and anti-inflammatory agents.

[1]  F. Awadallah,et al.  New quinazolinone-pyrimidine hybrids: synthesis, anti-inflammatory, and ulcerogenicity studies. , 2012, European journal of medicinal chemistry.

[2]  R. Carney,et al.  Inflammation and treatment response to sertraline in patients with coronary heart disease and comorbid major depression. , 2011, Journal of psychosomatic research.

[3]  Thomas E Lane,et al.  Inflammation induced by infection potentiates tau pathological features in transgenic mice. , 2011, The American journal of pathology.

[4]  P. Mishra,et al.  Anti-inflammatory and antinociceptive evaluation of newly synthesized 4-(substituted ethanoyl) amino-3-mercapto-5-(4-methoxy) phenyl-1,2,4-triazoles , 2011, Journal of pharmacy & bioallied sciences.

[5]  Y. S. Bakhle,et al.  Is the sulphonamide radical in the celecoxib molecule essential for its analgesic activity? , 2010, Pharmacological research.

[6]  K. El-Bayouki,et al.  Synthesis of some new 4(3H)-quinazolinone-2-carboxaldehyde thiosemicarbazones and their metal complexes and a study on their anticonvulsant, analgesic, cytotoxic and antimicrobial activities - part-1. , 2010, European journal of medicinal chemistry.

[7]  M. Khedr,et al.  Synthesis, biological evaluation and molecular docking of novel series of spiro [(2H,3H) quinazoline-2,1'- cyclohexan]-4(1H)- one derivatives as anti-inflammatory and analgesic agents. , 2010, European journal of medicinal chemistry.

[8]  T. Giordano,et al.  Design, synthesis and evaluation of novel 2-thiophen-5-yl-3H-quinazolin-4-one analogues as inhibitors of transcription factors NF-kappaB and AP-1 mediated transcriptional activation: Their possible utilization as anti-inflammatory and anti-cancer agents. , 2010, Bioorganic & medicinal chemistry.

[9]  B. Rather,et al.  Synthesis and anti-microbial screening of some Schiff bases of 3-amino-6,8-dibromo-2-phenylquinazolin-4(3H)-ones. , 2009, European journal of medicinal chemistry.

[10]  William E. Klunk,et al.  Effects of lipophilicity on the affinity and nonspecific binding of iodinated benzothiazole derivatives , 2007, Journal of Molecular Neuroscience.

[11]  A. Mishra,et al.  Synthesis and pharmacological study of novel pyrido-quinazolone analogues as anti-fungal, antibacterial, and anticancer agents. , 2006, Bioorganic & medicinal chemistry letters.

[12]  Christopher J. Wilson,et al.  Privileged structure-based quinazolinone natural product-templated libraries: identification of novel tubulin polymerization inhibitors. , 2006, Bioorganic & medicinal chemistry letters.

[13]  S. Kini,et al.  Synthesis and evaluation of new quinazolone derivatives of nalidixic acid as potential antibacterial and antifungal agents. , 2006, European journal of medicinal chemistry.

[14]  P. Guiry,et al.  Synthesis of Quinazolinones and Quinazolines , 2005 .

[15]  P. Khadikar,et al.  Topological modeling of lipophilicity, diuretic activity, and carbonic inhibition activity of benzene sulfonamides: a molecular connectivity approach. , 2004, Bioorganic & medicinal chemistry letters.

[16]  S. Sridhar,et al.  Synthesis, antiviral and cytotoxic activity of 6-bromo-2,3-disubstituted-4(3H)-quinazolinones. , 2003, Biological & pharmaceutical bulletin.

[17]  V. Ram,et al.  Synthesis and antihyperglycemic activity of suitably functionalized 3H-quinazolin-4-ones. , 2003, Bioorganic & medicinal chemistry.

[18]  Ola Sköld,et al.  Sulfonamide resistance: mechanisms and trends. , 2000, Drug resistance updates : reviews and commentaries in antimicrobial and anticancer chemotherapy.

[19]  H. G. Vogel.  Drug Discovery and Evaluation: Pharmacological Assays , 1997 .

[20]  P. Gounon,et al.  Inflammation: Patterns and new concepts , 1996, Research in Immunology.

[21]  K. Yoshikawa,et al.  Microbial bioassay of acute toxicity by the pH inhibition method and comparison of IC50 (pHI) with LD50 for rats and mice , 1993 .

[22]  T. Saito,et al.  Bioisosteric transformation of H1-antihistaminic benzimidazole derivatives. , 1989, Chemical & pharmaceutical bulletin.

[23]  C A WINTER,et al.  Carrageenin-Induced Edema in Hind Paw of the Rat as an Assay for Antiinflammatory Drugs , 1962, Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine.