An efficient NaHSO3-promoted protocol for chemoselective synthesis of 2-substituted benzimidazoles in water
暂无分享,去创建一个
Shu-Shan Jia | Wei Li | Weiwei Zhang | Yu-qin Jiang | Gui-qing Xu | Yamin Sun | Xi-yong Li
[1] H. Chiang,et al. The New Synthesis , 2019, Creatures of Cain.
[2] D. Wunderlin,et al. Selective and eco-friendly procedures for the synthesis of benzimidazole derivatives. The role of the Er(OTf)3 catalyst in the reaction selectivity , 2016, Beilstein journal of organic chemistry.
[3] Yao Tong,et al. An efficient route for the synthesis of benzimidazoles via a hydrogen-transfer strategy between o-nitroanilines and alcohols , 2016 .
[4] Youngsoo Kim,et al. Exploration of 2-benzylbenzimidazole scaffold as novel inhibitor of NF-κB. , 2016, Bioorganic & medicinal chemistry.
[5] Saratchandra Babu Mukkamala,et al. Simple and Efficient One-Pot Synthesis of 2-Substituted Benzimidazoles from o-Diaminoarene and Aryl Aldehydes. , 2016 .
[6] Monika Gupta,et al. 1,3,5-Trimethylpyrazolium chloride based ionogel as an efficient and reusable heterogeneous catalyst for the synthesis of benzimidazoles , 2016, Journal of Chemical Sciences.
[7] Ming Lu,et al. Synthesis of Benzimidazoles via Iron‐Catalyzed Aerobic Oxidation Reaction of Imine Derivatives with O‐Phenylenediamine. , 2015 .
[8] Ming Lu,et al. Green and Efficient Methods for One-Pot Aerobic Oxidative Synthesis of Benzimidazoles from Alcohols with TEMPO-PEG4000-NHC-Cu(II) Complex in Water. , 2015 .
[9] Saratchandra Babu Mukkamala,et al. Simple and Efficient One-Pot Synthesis of 2-Substituted Benzimidazoles from θ-Diaminoarene and Aryl Aldehydes , 2015 .
[10] N. Kaur,et al. Synergetic catalytic effect of ionic liquids and ZnO nanoparticles on the selective synthesis of 1,2-disubstituted benzimidazoles using a ball-milling technique , 2015 .
[11] Ming Lu,et al. Synthesis of Benzimidazoles via Iron-Catalyzed Aerobic Oxidation Reaction of Imine Derivatives with o-Phenylenediamine , 2015 .
[12] P. Verma,et al. Highly efficient water-mediated approach to access benzazoles: metal catalyst and base-free synthesis of 2-substituted benzimidazoles, benzoxazoles, and benzothiazoles , 2015, Molecular Diversity.
[13] Ming Lu,et al. Green and Efficient Methods for One-Pot Aerobic Oxidative Synthesis of Benzimidazoles from Alcohols with TEMPO-PEG4000-NHC-Cu(II) Complex in Water , 2015 .
[14] T. Punniyamurthy,et al. Copper(I)-catalyzed regioselective amination of N-aryl imines using TMSN3 and TBHP: a route to substituted benzimidazoles. , 2015, The Journal of organic chemistry.
[15] G. Bai,et al. An Ammonium Molybdate Deposited Amorphous Silica Coated Iron Oxide Magnetic Core—Shell Nanocomposite for the Efficient Synthesis of 2‐Benzimidazoles Using Hydrogen Peroxide. , 2014 .
[16] Sehyun Park,et al. Visible-Light-Promoted Synthesis of Benzimidazoles , 2014 .
[17] Hui-wang Ai,et al. A highly efficient oxidative condensation reaction for selective protein conjugation. , 2014, Chemical communications.
[18] G. Marconi,et al. A Scalable Route to the SMO Receptor Antagonist SEN826: Benzimidazole Synthesis via Enhanced in Situ Formation of the Bisulfite–Aldehyde Complex , 2014 .
[19] Gunaganti Naresh,et al. Molecular iodine promoted divergent synthesis of benzimidazoles, benzothiazoles, and 2-benzyl-3-phenyl-3,4-dihydro-2H-benzo[e][1,2,4]thiadiazines. , 2014, The Journal of organic chemistry.
[20] Radheshyam S. Shelkar,et al. Nano Ceria Catalyzed Synthesis of Substituted Benzimidazole, Benzothiazole, and Benzoxazole in Aqueous Media. , 2014 .
[21] A. Bamoniri,et al. One-Pot Synthesis of Benzimidazoles in Water in the Presence of SiO2–OPO3H , 2014, Chemistry of Heterocyclic Compounds.
[22] Dipratn G. Khandare,et al. DBSA Mediated Chemoselective Synthesis of 2-Substituted Benzimidazoles in Aqueous Media. , 2014 .
[23] R. Yousefi,et al. Magnetic nanoparticles-supported tungstosilicic acid: as an efficient magnetically separable solid acid for the synthesis of benzoazoles in water , 2014, Journal of the Iranian Chemical Society.
[24] Hidemasa Hikawa,et al. Benzoyl methyl phosphates as efficient reagents in the one-pot tandem approach for the synthesis of 2-phenylbenzimidazoles in water , 2014 .
[25] Radheshyam S. Shelkar,et al. Nano ceria catalyzed synthesis of substituted benzimidazole, benzothiazole, and benzoxazole in aqueous media , 2013 .
[26] S. Buchwald,et al. Suzuki-Miyaura cross-coupling of unprotected, nitrogen-rich heterocycles: substrate scope and mechanistic investigation. , 2013, Journal of the American Chemical Society.
[27] Ryosuke Ijuin,et al. Novel strategy for synthesis of substituted benzimidazo[1,2-a]quinolines. , 2013, Organic letters.
[28] L. Zhang,et al. Catalyst Free Approach to Benzimidazoles Using Air as the Oxidant at Room Temperature. , 2013 .
[29] Ji-tai Li,et al. Eco-Friendly Synthesis of 2-Substituted Benzimidazoles Using Air as the Oxidant , 2013 .
[30] M. Abdollahi-Alibeik,et al. Nanosized sulfated zirconia as solid acid catalyst for the synthesis of 2-substituted benzimidazoles , 2013, Chemical Papers.
[31] Dinesh Kumar,et al. Selectivity control during the solid supported protic acids catalysed synthesis of 1,2-disubstituted benzimidazoles and mechanistic insight to rationalize selectivity , 2013 .
[32] L. Zhang,et al. Catalyst free approach to benzimidazoles using air as the oxidant at room temperature , 2012 .
[33] William A. Dean,et al. Benzazoles from aliphatic amines and o-amino/mercaptan/hydroxyanilines: elemental sulfur as a highly efficient and traceless oxidizing agent. , 2012, Organic letters.
[34] A. Dandia,et al. Synthesis and characterization of CdS and Mn doped CdS nanoparticles and their catalytic application for chemoselective synthesis of benzimidazoles and benzothiazoles in aqueous medium , 2012 .
[35] P. Sahu,et al. Mild and highly efficient copper (II) sulfate catalyzed one pot synthesis of 2-aryl benzimidazole using atmospheric air as an oxidant and its antibacterial study , 2012, Medicinal Chemistry Research.
[36] M. Kočevar,et al. Boric Acid‐Catalyzed Direct Condensation of Carboxylic Acids with Benzene‐1,2‐diamine into Benzimidazoles. , 2012 .
[37] Manian Rajesh Kumar,et al. Copper-catalyzed, one-pot, three-component synthesis of benzimidazoles by condensation and C-N bond formation. , 2011, The Journal of organic chemistry.
[38] Chenjie Zhu,et al. An inorganic iodine-catalyzed oxidative system for the synthesis of benzimidazoles using hydrogen peroxide under ambient conditions. , 2011, ChemSusChem.
[39] Subhash C. Jain,et al. Synthesis of 2‐Arylbenzimidazoles in Water. , 2011 .
[40] M. Constantin,et al. A New Laccase-Catalyzed Domino Process and Its Application to the Efficient Synthesis of 2-Aryl-1H-benzimidazoles. , 2011 .
[41] R. Aryan,et al. Aqueous 1 M Glucose Solution as a Novel and Fully Green Reaction Medium and Catalyst for the Oxidant-Free Synthesis of 2-Arylbenzimidazoles , 2011 .
[42] L. Du,et al. Efficient One‐Pot Synthesis of Benzimidazoles under Solvent‐Free Conditions. , 2011 .
[43] Fangyun Hu,et al. Copper-catalyzed intramolecular C-N bond formation: a straightforward synthesis of benzimidazole derivatives in water. , 2011, The Journal of organic chemistry.
[44] S. Paul,et al. Nanosized Mn(acac)3 Anchored on Amino Functionalized Silica for the Selective Oxidative Synthesis of 2-arylbenzimidazoles, 2-arylbenzothiazoles and Aerobic Oxidation of Benzoins in Water , 2011 .
[45] P. Gong,et al. Synthesis and biological evaluation of 1H-benzimidazol-5-ols as potent HBV inhibitors. , 2010, Bioorganic & medicinal chemistry letters.
[46] K. Bahrami,et al. Synthesis of 1,2-disubstituted benzimidazoles, 2-substituted benzimidazoles and 2-substituted benzothiazoles in SDS micelles , 2010 .
[47] Nahid M. Yazdani,et al. Discovery of dual inducible/neuronal nitric oxide synthase (iNOS/nNOS) inhibitor development candidate 4-((2-cyclobutyl-1H-imidazo[4,5-b]pyrazin-1-yl)methyl)-7,8-difluoroquinolin-2(1H)-one (KD7332) part 2: identification of a novel, potent, and selective series of benzimidazole-quinolinone iNOS/nNOS , 2010, Journal of medicinal chemistry.
[48] Atul Kumar,et al. Diversity‐Oriented Synthesis of Benzimidazole, Benzoxazole, Benzothiazole and Quinazolin‐4(3H)‐one Libraries via Potassium Persulfate—CuSO4‐Mediated Oxidative Coupling Reactions of Aldehydes in Aqueous Micelles. , 2010 .
[49] Zhao‐Yang Wang,et al. Rapid and Cheap Synthesis of Benzimidazoles via Intermittent Microwave Promotion: A Simple and Potential Industrial Application of Air as Oxidant , 2010 .
[50] T. Yamashita,et al. New Procedure for the Synthesis of 2‐Alkylbenzimidazoles. , 2010 .
[51] Anna Wilhelmsson,et al. 1-(3-Aryloxyaryl)benzimidazole sulfones are liver X receptor agonists. , 2010, Bioorganic & medicinal chemistry letters.
[52] B. Pérez,et al. One‐Pot Microwave Promoted Synthesis of 2‐Aryl‐1H‐benzimidazoles Using Sodium Hydrogen Sulfite. , 2009 .
[53] Jie‐Ping Wan,et al. Water mediated chemoselective synthesis of 1,2-disubstituted benzimidazoles using o-phenylenediamine and the extended synthesis of quinoxalines , 2009 .
[54] A. Amani,et al. Very fast and efficient synthesis of some novel substituted 2-arylbenzimidazoles in water using ZrOCl2·nH2O on montmorillonite K10 as catalyst , 2009 .
[55] G. Coppola. N-Hydroxyphthalimide/Cobalt Acetate, a New Catalytic Oxidative System for the Synthesis of Benzimidazoles. , 2009 .
[56] L. Goossen,et al. Concise synthesis of telmisartan via decarboxylative cross-coupling. , 2008, The Journal of organic chemistry.
[57] H. Sharghi,et al. Reusable Cobalt(III)‐Salen Complex Supported on Activated Carbon as an Efficient Heterogeneous Catalyst for Synthesis of 2‐Arylbenzimidazole Derivatives , 2008 .
[58] Y. Bansal,et al. Angiotensin II--AT1 receptor antagonists: design, synthesis and evaluation of substituted carboxamido benzimidazole derivatives. , 2008, European journal of medicinal chemistry.
[59] K. Bahrami,et al. Mild and highly efficient method for the synthesis of 2-arylbenzimidazoles and 2-arylbenzothiazoles. , 2008, The Journal of organic chemistry.
[60] Huiqiang Ma,et al. A simple and efficient synthesis of 2-aryl-substituted benzimidazoles , 2008 .
[61] G. Navarrete-Vázquez,et al. Microwave‐Assisted One‐Pot Synthesis of 2‐(Substituted phenyl)‐1H‐benzimidazole Derivatives. , 2008 .
[62] C. Aakeröy,et al. Structural competition between hydrogen bonds and halogen bonds. , 2007, Journal of the American Chemical Society.
[63] Yanguang Wang,et al. A Rapid and Efficient Synthesis of Benzimidazoles Using Hypervalent Iodine as Oxidant , 2007 .
[64] A. Mavrova,et al. Antihelminthic activity of some newly synthesized 5(6)-(un)substituted-1H-benzimidazol-2-ylthioacetylpiperazine derivatives. , 2006, European journal of medicinal chemistry.
[65] Chinpiao Chen,et al. Synthesis and anticancer evaluation of bis(benzimidazoles), bis(benzoxazoles), and benzothiazoles. , 2006, Bioorganic & medicinal chemistry.
[66] Libing Yu,et al. Microwave-Assisted One-Step High-Throughput Synthesis of Benzimidazoles. , 2006 .
[67] M. Heravi,et al. Zeolites. Efficient and Eco-friendly Catalysts for the Synthesis of Benzimidazoles , 2006 .
[68] P. Gogoi,et al. An efficient and one-pot synthesis of imidazolines and benzimidazoles via anaerobic oxidation of carbon–nitrogen bonds in water , 2006 .
[69] Lihu Yang,et al. A Simple and Efficient Procedure for the Synthesis of Benzimidazoles Using Air as the Oxidant. , 2005 .
[70] S. Anzali,et al. Halothiophene benzimidazoles as P1 surrogates of inhibitors of blood coagulation factor Xa. , 2004, Bioorganic & medicinal chemistry letters.
[71] Douglas A. Horton,et al. The Combinatorial Synthesis of Bicyclic Privileged Structures or Privileged Substructures , 2003 .
[72] M. Stevens,et al. Antitumor Benzothiazoles. Part 20. 3′-Cyano and 3′-Alkynyl-Substituted 2-(4′-Aminophenyl)benzothiazoles as New Potent and Selective Analogues. , 2003 .
[73] A. J. Blake,et al. Synthesis of benzimidazoles in high-temperature water , 2003 .
[74] M. Stevens,et al. Antitumour benzothiazoles. Part 20: 3'-cyano and 3'-alkynyl-substituted 2-(4'-aminophenyl)benzothiazoles as new potent and selective analogues. , 2003, Bioorganic & medicinal chemistry letters.
[75] S. Servi. The efficient synthesis of 2-arylamino-2-imidazolines, 2-heteroaryl-substituted benzimidazoles, and their morpholin-4-ylmethyl derivatives , 2002 .
[76] J. Kane,et al. A Short Synthesis of the PARP Inhibitor 2‐(4‐Trifluoromethylphenyl)benzimidazole‐4‐carboxamide (NU1077) (V). , 2001 .
[77] B. Foleno,et al. Amidino Benzimidazole Inhibitors of Bacterial Two-Component Systems , 2001 .
[78] John A. Walker,et al. Design, Synthesis, and Antiviral Activity of α‐Nucleosides: D‐ and L‐Isomers of Lyxofuranosyl‐ and (5‐Deoxylyxofuranosyl)benzimidazoles. , 1998 .
[79] P. Boyer,et al. Synthesis and Biological Activity of Novel Nonnucleoside Inhibitors of HIV‐1 Reverse Transcriptase. 2‐Aryl‐Substituted Benzimidazoles. , 1998 .
[80] L. Kucera,et al. Design, synthesis, and antiviral evaluations of 1-(substituted benzyl)-2-substituted-5,6-dichlorobenzimidazoles as nonnucleoside analogues of 2,5,6-trichloro-1-(beta-D-ribofuranosyl)benzimidazole. , 1998, Journal of medicinal chemistry.
[81] L. Braverman,et al. Ammonium persulfate: a safe alternative oxidizing reagent for measuring urinary iodine. , 1996, Clinical chemistry.
[82] J. V. Eynde,et al. 2,3-Dichloro-5,6-dicyano-1,4-benzoquinone, a Mild Catalyst for the Formation of Carbon-Nitrogen Bonds. , 1995 .
[83] J. V. Eynde,et al. 2,3-Dichloro-5,6-dicyano-1,4-benzoquinone, a mild catalyst for the formation of carbon-nitrogen bonds , 1995 .
[84] E. Bouwman,et al. Model systems for type I copper proteins: structures of copper coordination compounds with thioether and azole-containing ligands , 1990 .
[85] J. B. Hendrickson,et al. Reactions of Carboxylic Acids with “Phosphonium Anhydrides”. , 1989 .
[86] M. A. Pujar,et al. Cobalt(II), nickel(II) and copper(II) complexes of bidentate bibenzimidazoles , 1988 .
[87] G. M. Timmis,et al. A new synthesis of benzimidazoles and aza‐analogs , 1965 .
[88] W. Hartung,et al. α-Aminoalkanesulfonic Acids1,2 , 1959 .