Synthesis and evaluation of novel monosubstituted sulfonylurea derivatives as antituberculosis agents.

[1]  Chun Wu,et al.  In vitro efficacy of acetohydroxyacid synthase inhibitors against clinical strains of Mycobacterium tuberculosis isolated from a hospital in Beijing, China. , 2011, Saudi medical journal.

[2]  Alon Herschhorn,et al.  Structure--activity relationship studies of 1-(4-chloro-2,5-dimethoxyphenyl)-3-(3-propoxypropyl)thiourea, a non-nucleoside reverse transcriptase inhibitor of human immunodeficiency virus type-1. , 2011, European journal of medicinal chemistry.

[3]  Eric Arnoult,et al.  The challenge of new drug discovery for tuberculosis , 2011, Nature.

[4]  Vinayak Singh,et al.  Biochemical and transcription analysis of acetohydroxyacid synthase isoforms in Mycobacterium tuberculosis identifies these enzymes as potential targets for drug development. , 2011, Microbiology.

[5]  Jufang He,et al.  Prevalence of multidrug and extensively drug-resistant tuberculosis in Beijing, China: a hospital-based retrospective study. , 2010, Japanese journal of infectious diseases.

[6]  G. Brahmachari,et al.  A very simple and highly efficient procedure for N-formylation of primary and secondary amines at room temperature under solvent-free conditions , 2010 .

[7]  L. Guddat,et al.  Crystal structures of two novel sulfonylurea herbicides in complex with Arabidopsis thaliana acetohydroxyacid synthase , 2009, The FEBS Journal.

[8]  Zhengming Li,et al.  Synthesis and herbicidal activities of pyridyl sulfonylureas: More convenient preparation process of phenyl pyrimidylcarbamates , 2008 .

[9]  Dong-Wan Koo,et al.  In vitro and ex vivo activity of new derivatives of acetohydroxyacid synthase inhibitors against Mycobacterium tuberculosis and non-tuberculous mycobacteria. , 2008, International journal of antimicrobial agents.

[10]  Moon-Young Yoon,et al.  Characterization of acetohydroxyacid synthase from Mycobacterium tuberculosis and the identification of its new inhibitor from the screening of a chemical library , 2005, FEBS letters.

[11]  Z. Barak,et al.  Acetohydroxyacid synthase from Mycobacterium avium and its inhibition by sulfonylureas and imidazolinones. , 2003, Biochimica et biophysica acta.

[12]  J. Schloss,et al.  Inhibitors of branched-chain amino acid biosynthesis as potential antituberculosis agents. , 1998, The Journal of antimicrobial chemotherapy.

[13]  Z. Barak,et al.  Biosynthesis of 2-aceto-2-hydroxy acids: acetolactate synthases and acetohydroxyacid synthases. , 1998, Biochimica et biophysica acta.

[14]  D. Shaner,et al.  Imidazolinones: potent inhibitors of acetohydroxyacid synthase. , 1984, Plant physiology.

[15]  R S Chaleff,et al.  Acetolactate Synthase Is the Site of Action of Two Sulfonylurea Herbicides in Higher Plants , 1984, Science.

[16]  T. Mosmann.  Rapid colorimetric assay for cellular growth and survival: application to proliferation and cytotoxicity assays. , 1983, Journal of immunological methods.