Synthesis of novel 2-[4-(4-substitutedbenzamido/phenylacetamido)phenyl]benzothiazoles as antimicrobial agents

[1]  Y. Komatsu,et al.  Synthesis of a Novel Dual Inhibitor of Thromboxane A2 Synthetase and 5- Lipoxygenase (E3040) via the Direct Coupling Reaction of Hydroquinone with 3-Pyridinecarboxaldehyde. , 2010 .

[2]  M. Peach,et al.  Preparation of transition metal thiosemicarbazone derivative complexes for medical imaging and therapy , 2007 .

[3]  E. Akı-Şener,et al.  3D-QSAR study on heterocyclic topoisomerase II inhibitors using CoMSIA , 2006, SAR and QSAR in environmental research.

[4]  E. Akı-Şener,et al.  3D-QSAR analysis on benzazole derivatives as eukaryotic topoisomerase II inhibitors by using comparative molecular field analysis method. , 2005, Bioorganic & medicinal chemistry.

[5]  P. Yurdakul,et al.  Some fused heterocyclic compounds as eukaryotic topoisomerase II inhibitors. , 2004, Biochemical and biophysical research communications.

[6]  E. Akı-Şener,et al.  Synthesis and structure-activity relationships of new antimicrobial active multisubstituted benzazole derivatives. , 2004, European journal of medicinal chemistry.

[7]  P Phani Kumar,et al.  Design, synthesis and biological evaluation of benzimidazole/benzothiazole and benzoxazole derivatives as cyclooxygenase inhibitors. , 2003, Bioorganic & medicinal chemistry letters.

[8]  J. Kočí,et al.  Heterocyclic benzazole derivatives with antimycobacterial in vitro activity. , 2002, Bioorganic & medicinal chemistry letters.

[9]  M. Stevens,et al.  Antitumor benzothiazoles. 16. Synthesis and pharmaceutical properties of antitumor 2-(4-aminophenyl)benzothiazole amino acid prodrugs. , 2002, Journal of medicinal chemistry.

[10]  R. Gaynes,et al.  Antimicrobial resistance in intensive care units. , 1999, Clinics in chest medicine.

[11]  M. Stevens,et al.  Antitumor benzothiazoles. 7. Synthesis of 2-(4-acylaminophenyl)benzothiazoles and investigations into the role of acetylation in the antitumor activities of the parent amines. , 1999, Journal of medicinal chemistry.

[12]  I. Yalcin,et al.  Synthesis and microbiological activity of some novel N-(2-hydroxyl-5-substitutedphenyl)benzacetamides, phenoxyacetamides and thiophenoxyacetamides as the possible metabolites of antimicrobial active benzoxazoles. , 1997, Farmaco.

[13]  H. Küçükbay,et al.  Antifungal activity of organic and organometallic derivatives of benzimidazole and benzothiazole. , 1997, Arzneimittel-Forschung.

[14]  M. Stevens,et al.  Antitumor Benzothiazoles. Part 3. Synthesis of 2‐(4‐Aminophenyl) benzothiazoles and Evaluation of Their Activities Against Breast Cancer Cell Lines in vitro and in vivo. , 1996 .

[15]  S Wrigley,et al.  Antitumor benzothiazoles. 3. Synthesis of 2-(4-aminophenyl)benzothiazoles and evaluation of their activities against breast cancer cell lines in vitro and in vivo. , 1996, Journal of medicinal chemistry.

[16]  A. Kubota,et al.  E2011 a novel, selective and reversible inhibitor of monoamine oxidase type A. , 1996, The Journal of pharmacology and experimental therapeutics.

[17]  Y. Komatsu,et al.  Synthesis of a novel dual inhibitor of thromboxane A2 synthetase and 5-lipoxygenase (E3040) via the direct coupling reaction of hydroquinone with 3-pyridinecarboxaldehyde. , 1995, Chemical & pharmaceutical bulletin.

[18]  J. Gardiner,et al.  Synthesis and HIV-1 inhibition of novel benzimidazole derivatives , 1995 .

[19]  J. Surin.  Anti-nematode activity of sixteen compounds against Trichinella spiralis in mice--a possible new screen for macrofilaricides. , 1995, The Southeast Asian journal of tropical medicine and public health.

[20]  G. Trapani,et al.  Synthesis and antimicrobial activity of some N-alkenyl-2-acylalkylidene-2,3-dihydro-1,3-benzothiazoles. , 1994, Arzneimittel-Forschung.

[21]  I. Yalcin,et al.  The Synthesis and the Structure‐Activity Relationships of Some Substituted Benzoxazoles, Oxazolo(4,5‐b)pyridines, Benzothiazoles and Benzimidazoles as Antimicrobial Agents. , 1992 .

[22]  W. R. Tully,et al.  Synthesis and Oral Antiallergic Activity of Carboxylic Acids Derived from Imidazo(2,1-c)(1,4)benzoxazines, Imidazo(1,2-a)quinolines, Imidazo(1,2-a)quinoxalines, Imidazo(1,2-a)quinoxalinones, Pyrrolo(1,2-a)quinoxalinones, Pyrrolo(2,3-a , 1988 .

[23]  R. Lewis,et al.  6-Amino-2-Benzothiazolesulfonamide , 1988 .

[24]  D. Kay,et al.  Synthesis and oral antiallergic activity of carboxylic acids derived from imidazo[2,1-c][1,4]benzoxazines, imidazo[1,2-a]quinolines, imidazo[1,2-a]quinoxalines, imidazo[1,2-a]quinoxalinones, pyrrolo[1,2-a]quinoxalinones, pyrrolo[2,3-a]quinoxalinones, and imidazo[2,1-b]benzothiazoles. , 1988, Journal of medicinal chemistry.

[25]  R. Brubaker,et al.  6-amino-2-benzothiazole-sulfonamide. The effect of a topical carbonic anhydrase inhibitor on aqueous humor formation in the normal human eye. , 1988, Ophthalmology.

[26]  D. W. Hein,et al.  The Use of Polyphosphoric Acid in the Synthesis of 2-Aryl- and 2-Alkyl-substituted Benzimidazoles, Benzoxazoles and Benzothiazoles1 , 1957 .

[27]  L. Katz.  Antituberculous Compounds. III. Benzothiazole and Benzoxazole Derivatives , 1953 .