Diverse therapeutic potential of 3-hydroxy-4-pyranones and related compounds as kojic acid analogs
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[1] G. Karakaya,et al. Synthesis and Molecular Modeling of Some Novel Hydroxypyrone Derivatives as Antidermatophytic Agents , 2022, Journal of Heterocyclic Chemistry.
[2] L. Zhong,et al. Small molecules in targeted cancer therapy: advances, challenges, and future perspectives , 2021, Signal Transduction and Targeted Therapy.
[3] Cleison C. Lobato,et al. Molecular modification approach on kojic acid derivatives as antioxidants related to ascorbic acid , 2020, Journal of Molecular Modeling.
[4] H. Ansari,et al. An investigation of the effects of environmental and ecologic factors on cutaneous leishmaniasis in the old world: a systematic review study , 2020, Reviews on environmental health.
[5] S. Jokar,et al. Comparison of Deferoxamine, Deferiprone and Deferasirox Iron-Chelating Agents in Reducing Serum Ferritin Levels in Patients with Thalassemia Major , 2020, Journal of Clinical Care and Skills.
[6] J. Selvin,et al. Revealing antibiotic resistance in therapeutic and dietary probiotic supplements. , 2020, Journal of global antimicrobial resistance.
[7] E. Beghi. The Epidemiology of Epilepsy , 2019, Neuroepidemiology.
[8] L. Zuo,et al. Inflammaging and Oxidative Stress in Human Diseases: From Molecular Mechanisms to Novel Treatments , 2019, International journal of molecular sciences.
[9] Wei Lu,et al. Development of novel human lactate dehydrogenase A inhibitors: High-throughput screening, synthesis, and biological evaluations. , 2019, European journal of medicinal chemistry.
[10] Miri Lee,et al. Anti-inflammatory Effects of a P-coumaric Acid and Kojic Acid Derivative in LPS-stimulated RAW264.7 Macrophage Cells , 2019, Biotechnology and Bioprocess Engineering.
[11] S. Saran,et al. Consistent production of kojic acid from Aspergillus sojae SSC-3 isolated from rice husk , 2019, Molecular Biology Reports.
[12] A. Daryani,et al. In vitro and in vivo evaluation of kojic acid against Toxoplasma gondii in experimental models of acute toxoplasmosis. , 2019, Experimental parasitology.
[13] M. Peana,et al. A new tripodal kojic acid derivative for iron sequestration: Synthesis, protonation, complex formation studies with Fe3+, Al3+, Cu2+ and Zn2+, and in vivo bioassays. , 2019, Journal of inorganic biochemistry.
[14] M. Saeedi,et al. Kojic acid applications in cosmetic and pharmaceutical preparations. , 2019, Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie.
[15] Qing-Xi Chen,et al. Kinetic and computational molecular docking simulation study of novel kojic acid derivatives as anti-tyrosinase and antioxidant agents , 2019, Journal of enzyme inhibition and medicinal chemistry.
[16] D. Jun,et al. Synthesis and biological assessment of KojoTacrines as new agents for Alzheimer’s disease therapy , 2018, Journal of enzyme inhibition and medicinal chemistry.
[17] Yu-gang Shi,et al. Evaluation of antibacterial and anti-biofilm properties of kojic acid against five food-related bacteria and related subcellular mechanisms of bacterial inactivation , 2018, Food science and technology international = Ciencia y tecnologia de los alimentos internacional.
[18] E. Giovannetti,et al. Synthetic small molecules as anti-biofilm agents in the struggle against antibiotic resistance. , 2019, European journal of medicinal chemistry.
[19] Jia-hui Yu,et al. Design, synthesis and biological evaluation of 2-substituted 3-hydroxy-6-methyl-4H-pyran-4-one derivatives as Pseudomonas aeruginosa biofilm inhibitors. , 2018, European journal of medicinal chemistry.
[20] L. Peixe,et al. New fluorescent rosamine chelator showing promising antibacterial activity against Gram-positive bacteria. , 2018, Bioorganic chemistry.
[21] W. Xia,et al. One-step procedure for enhancing the antibacterial and antioxidant properties of a polysaccharide polymer: Kojic acid grafted onto chitosan. , 2018, International journal of biological macromolecules.
[22] E. Telleria,et al. Leishmania, microbiota and sand fly immunity , 2018, Parasitology.
[23] Y. Taufiq-Yap,et al. The crucial roles of inflammatory mediators in inflammation: A review , 2018, Veterinary world.
[24] Wei-Min Chen,et al. Design, synthesis and biological evaluation of novel 5-hydroxy-2-methyl-4H-pyran-4-one derivatives as antiglioma agents. , 2018, MedChemComm.
[25] B. Farhood,et al. Incidence and Mortality of Various Cancers in Iran and Compare to Other Countries: A Review Article , 2018, Iranian journal of public health.
[26] A. Fassihi,et al. Synthesis and antileishmanial activity of antimony (V) complexes of hydroxypyranone and hydroxypyridinone ligands , 2018, Research in pharmaceutical sciences.
[27] S. Emami,et al. New indole-based chalconoids as tubulin-targeting antiproliferative agents. , 2017, Bioorganic chemistry.
[28] M. Keighobadi,et al. An overview of azoles targeting sterol 14α-demethylase for antileishmanial therapy. , 2017, European journal of medicinal chemistry.
[29] Shao-Cong Sun,et al. NF-κB signaling in inflammation , 2017, Signal Transduction and Targeted Therapy.
[30] Wenjing Chu,et al. Discovery of Novel Pyridone-Conjugated Monosulfactams as Potent and Broad-Spectrum Antibiotics for Multidrug-Resistant Gram-Negative Infections. , 2017, Journal of medicinal chemistry.
[31] R. Sheng,et al. Synthesis and biological evaluation of deferiprone-resveratrol hybrids as antioxidants, Aβ1-42 aggregation inhibitors and metal-chelating agents for Alzheimer's disease. , 2017, European journal of medicinal chemistry.
[32] A. Majeed,et al. Brain biometals and Alzheimer's disease – boon or bane? , 2017, The International journal of neuroscience.
[33] Xiaole Kong,et al. Systematic comparison of the mono-, dimethyl- and trimethyl 3-hydroxy-4(1H)-pyridones - Attempted optimization of the orally active iron chelator, deferiprone. , 2016, European journal of medicinal chemistry.
[34] J. Seo,et al. Discovery of a potent enoyl-acyl carrier protein reductase (FabI) inhibitor suitable for antistaphylococcal agent. , 2015, Bioorganic & medicinal chemistry letters.
[35] M. Zirak,et al. Kojic acid in organic synthesis , 2015 .
[36] S. Ulusoy,et al. Inhibition of Pseudomonas aeruginosa biofilm formation by 2,2’-bipyridyl, lipoic, kojic and picolinic acids , 2015, Iranian journal of basic medical sciences.
[37] J. Nanubolu,et al. One-pot catalyst free synthesis of novel kojic acid tagged 2-aryl/alkyl substituted-4H-chromenes and evaluation of their antimicrobial and anti-biofilm activities. , 2015, Bioorganic & medicinal chemistry letters.
[38] S. Emami,et al. Kojic acid-derived tyrosinase inhibitors: synthesis and bioactivity , 2015 .
[39] O. Hansson,et al. β-amyloid Peptides and Amyloid Plaques in Alzheimer’s Disease , 2014, Neurotherapeutics.
[40] Shaoshan Li,et al. Ciprofloxacin containing Mannich base and its copper complex induce antitumor activity via different mechanism of action. , 2014, International journal of oncology.
[41] A. Tamrakar,et al. Synthesis of heteroaryl/aryl kojic acid conjugates as stimulators of glucose uptake by GLUT4 translocation. , 2014, European journal of medicinal chemistry.
[42] M. Faramarzi,et al. Mannich Bases of 7‐Piperazinylquinolones and Kojic Acid Derivatives: Synthesis, in vitro Antibacterial Activity and in silico Study. , 2014 .
[43] A. Santos,et al. A Novel Function for Kojic Acid, a Secondary Metabolite from Aspergillus Fungi, as Antileishmanial Agent , 2014, PloS one.
[44] Yanshun Xu,et al. Synthesis, characterization, and antimicrobial activity of kojic acid grafted chitosan oligosaccharide. , 2014, Journal of agricultural and food chemistry.
[45] M. Crespo-Alonso,et al. Searching for new aluminium chelating agents: a family of hydroxypyrone ligands. , 2014, Journal of inorganic biochemistry.
[46] M. Crespo-Alonso,et al. A family of hydroxypyrone ligands designed and synthesized as iron chelators. , 2013, Journal of inorganic biochemistry.
[47] M. Faramarzi,et al. Mannich bases of 7-piperazinylquinolones and kojic acid derivatives: synthesis, in vitro antibacterial activity and in silico study. , 2013, European journal of medicinal chemistry.
[48] O. Firuzi,et al. Cytotoxic activity assessment, QSAR and docking study of novel bis-carboxamide derivatives of 4-pyrones synthesized by Ugi four-component reaction. , 2013, European journal of medicinal chemistry.
[49] M. Jakupec,et al. Identification of the structural determinants for anticancer activity of a ruthenium arene peptide conjugate. , 2013, Chemistry.
[50] Hai-bin Luo,et al. Design, synthesis, and evaluation of multitarget-directed resveratrol derivatives for the treatment of Alzheimer's disease. , 2013, Journal of medicinal chemistry.
[51] V. Shanmugasundaram,et al. Pyridone-conjugated monobactam antibiotics with gram-negative activity. , 2013, Journal of medicinal chemistry.
[52] G. Karakaya,et al. Evaluation of bioactivities of chlorokojic acid derivatives against dermatophytes couplet with cytotoxicity. , 2013, Bioorganic & medicinal chemistry letters.
[53] P. T. Perumal,et al. Cu(OTf)2 catalyzed three component reaction: efficient synthesis of spiro[indoline-3,4'-pyrano[3,2-b]pyran derivatives and their anticancer potency towards A549 human lung cancer cell lines. , 2013, Bioorganic & medicinal chemistry letters.
[54] G. Karakaya,et al. Design, synthesis and in vivo/in vitro screening of novel chlorokojic acid derivatives , 2013, Journal of enzyme inhibition and medicinal chemistry.
[55] B. Campbell,et al. Enhancement of Commercial Antifungal Agents by Kojic Acid , 2012, International journal of molecular sciences.
[56] C. Hulme,et al. Synthesis of kojic acid-derived copper-chelating apoptosis inducing agents , 2012, Medicinal Chemistry Research.
[57] S. Shin,et al. Studies on Tyrosinase Inhibitory and Antioxidant Activities of Benzoic Acid Derivatives Containing Kojic Acid Moiety , 2011 .
[58] Xiaole Kong,et al. Synthesis, iron(III)-binding affinity and in vitro evaluation of 3-hydroxypyridin-4-one hexadentate ligands as potential antimicrobial agents. , 2011, Bioorganic & medicinal chemistry letters.
[59] J. Cho,et al. Ester Derivatives of Kojic Acid and Polyphenols Containing Adamantane Moiety with Tyrosinase Inhibitory and Anti-inflammatory Properties , 2011 .
[60] T. Gootz,et al. Preparation, gram-negative antibacterial activity, and hydrolytic stability of novel siderophore-conjugated monocarbam diols. , 2011, ACS medicinal chemistry letters.
[61] B. Özçelik,et al. Synthesis and biological activities of new Mannich bases of chlorokojic acid derivatives , 2011, Medicinal Chemistry Research.
[62] B. Reddy,et al. Indium(III) chloride catalyzed three-component coupling reaction: a novel synthesis of 2-substituted aryl(indolyl)kojic acid derivatives as potent antifungal and antibacterial agents. , 2010, Bioorganic & medicinal chemistry letters.
[63] M. Aytemir,et al. A study of cytotoxicity of novel chlorokojic acid derivatives with their antimicrobial and antiviral activities. , 2010, European journal of medicinal chemistry.
[64] J. Cho,et al. A modulatory effect of novel kojic acid derivatives on cancer cell proliferation and macrophage activation. , 2010, Die Pharmazie.
[65] M. Aytemir,et al. Anticonvulsant and Neurotoxicity Evaluation of Some Novel Kojic Acids and Allomaltol Derivatives , 2010, Archiv der Pharmazie.
[66] I. Kurnaz,et al. 4H-Pyran-4-one derivatives:; leading molecule for preparation of compounds with antimycobacterial potential , 2009 .
[67] C. Glabe,et al. Soluble fibrillar oligomer levels are elevated in Alzheimer's disease brain and correlate with cognitive dysfunction , 2009, Neurobiology of Disease.
[68] S. Hosseinimehr,et al. Radioprotective effects of kojic acid against mortality induced by gamma irradiation in mice. , 2009, Saudi medical journal.
[69] H. Waldmann,et al. Gamma-pyrone natural products--a privileged compound class provided by nature. , 2009, Bioorganic & medicinal chemistry.
[70] R. Hider,et al. Iron chelation as a potential therapy for neurodegenerative disease. , 2008, Biochemical Society transactions.
[71] J. Brtko,et al. In vitro antiproliferative and cytotoxic activities of novel kojic acid derivatives: 5‐benzyloxy‐2‐selenocyanatomethyl‐ and 5‐methoxy‐2‐selenocyanatomethyl‐4‐pyranone , 2008, Journal of applied toxicology : JAT.
[72] S. M. Taghdisi,et al. Kojic acid and its manganese and zinc complexes as potential radioprotective agents. , 2007, Bioorganic & medicinal chemistry letters.
[73] M. Camplo,et al. Novel iron-specific fluorescent probes. , 2005, Bioorganic & medicinal chemistry letters.
[74] M. Özalp,et al. Synthesis and Evaluation of Anticonvulsant and Antimicrobial Activities of 3‐Hydroxy‐6‐methyl‐2‐substituted 4H‐Pyran‐4‐one Derivatives , 2004, Archiv der Pharmazie.
[75] E. Giacobini. Cholinesterases: New Roles in Brain Function and in Alzheimer's Disease , 2003, Neurochemical Research.
[76] R. Hider,et al. Synthesis and Evaluation of Antimicrobial Activity of New 3-Hydroxy-6-methyl-4-oxo-4H -pyran-2- carboxamide Derivatives , 2003 .
[77] R. Hider,et al. Synthesis of New Antimicrobial Agents; Amide Derivatives of Pyranones and Pyridinones , 2003 .
[78] L. Novotný,et al. Antileukemic activity of 4-pyranone derivatives. , 1995, The international journal of biochemistry & cell biology.
[79] P. Watkins,et al. Hepatotoxic effects of tacrine administration in patients with Alzheimer's disease. , 1994, JAMA.
[80] J. L. Vaught,et al. An antinociceptive profile of kojic amine: an analogue of gamma-aminobutyric acid (GABA). , 1987, Neuropharmacology.
[81] J. Rokach,et al. Kojic amine--a novel gamma-aminobutyric acid analogue. , 1979, Journal of medicinal chemistry.
[82] T. Fujita,et al. Structure-activity Study of Bacteriostatic Kojic Acid Analogs , 1975 .