Visible light-induced one-pot three-component synthesis of quinazolines under catalyst-free condition

[1]  G. Psomas,et al.  Transition metal(II) complexes of halogenated derivatives of (E)-4-(2-(pyridin-2-ylmethylene)hydrazinyl)quinazoline: structure, antioxidant activity, DNA-binding DNA photocleavage, interaction with albumin and in silico studies. , 2022, Dalton Transactions.

[2]  R. Tuxworth,et al.  Inhibition of Chk2 promotes neuroprotection, axon regeneration, and functional recovery after CNS injury , 2022, Science advances.

[3]  Q. Fan,et al.  Straightforward synthesis of quinazolin-4(3H)-ones via visible light-induced condensation cyclization , 2022, RSC advances.

[4]  Neelima Mahato,et al.  Recent Advances on Quinazoline Derivatives: A Potential Bioactive Scaffold in Medicinal Chemistry , 2021, ChemEngineering.

[5]  Q. Fan,et al.  Catalyst-free visible-light mediated selective oxidation of sulfides into sulfoxides under clean conditions , 2021, Green Chemistry.

[6]  Xue-Meng Wang,et al.  Synthesis of benzothiazoles using fluorescein as an efficient photocatalyst under visible light , 2021, Molecular Catalysis.

[7]  Xiao‐Feng Wu,et al.  Palladium-catalyzed carbonylative synthesis of quinazolines: Silane act as better nucleophile than amidine , 2021, Molecular Catalysis.

[8]  Jorge Quintero-Saumeth,et al.  Biologically Active Quinoline‐Hydrazone Conjugates as Potential Trypanosoma cruzi DHFR‐TS Inhibitors: Docking, Molecular Dynamics, MM/PBSA and Drug‐Likeness Studies , 2021 .

[9]  Cheng‐Chung Wang,et al.  TMSOTf-catalyzed synthesis of substituted quinazolines using hexamethyldisilazane as a nitrogen source under neat and microwave irradiation conditions. , 2020, Organic & biomolecular chemistry.

[10]  N. Azas,et al.  Synthesis and Antiplasmodial Evaluation of 4-Carboxamido- and 4-Alkoxy-2-Trichloromethyl Quinazolines , 2020, Molecules.

[11]  N. Curtin,et al.  DNA damage checkpoint kinases in cancer , 2020, Expert Reviews in Molecular Medicine.

[12]  D. S. Bose,et al.  A convenient access to 2,4-disubstituted quinazolines via one-pot three-component reaction under mild conditions† , 2020, Synthetic Communications.

[13]  Bo Xu,et al.  A two-dimensional quinazoline based covalent organic framework with a suitable direct gap and superior optical absorption for photovoltaic applications , 2020 .

[14]  Qingbin Meng,et al.  Direct C–H difluoromethylation of heterocycles via organic photoredox catalysis , 2020, Nature Communications.

[15]  A. Gemma,et al.  Gefitinib Alone Versus Gefitinib Plus Chemotherapy for Non-Small-Cell Lung Cancer With Mutated Epidermal Growth Factor Receptor: NEJ009 Study. , 2020, Journal of clinical oncology : official journal of the American Society of Clinical Oncology.

[16]  A. Gemma,et al.  Erlotinib plus bevacizumab versus erlotinib alone in patients with EGFR-positive advanced non-squamous non-small-cell lung cancer (NEJ026): interim analysis of an open-label, randomised, multicentre, phase 3 trial. , 2019, The Lancet. Oncology.

[17]  Chae S. Yi,et al.  Synthesis of Quinazoline and Quinazolinone Derivatives via Ligand-Promoted Ruthenium-Catalyzed Dehydrogenative and Deaminative Coupling Reaction of 2-Aminophenyl Ketones and 2-Aminobenzamides with Amines. , 2019, Organic letters.

[18]  S. Sinha,et al.  Dehydrogenative Synthesis of Quinolines, 2-Aminoquinolines, and Quinazolines Using Singlet Diradical Ni(II)-Catalysts. , 2019, The Journal of organic chemistry.

[19]  O. Chupakhin,et al.  Functionalized Quinazolines and Pyrimidines for Optoelectronic Materials , 2018, Current Organic Synthesis.

[20]  A. Lei,et al.  Electrochemical Acceptorless Dehydrogenation of N-Heterocycles Utilizing TEMPO as Organo-Electrocatalyst , 2018 .

[21]  T. Mohamed,et al.  2,4-Disubstituted quinazolines as amyloid-β aggregation inhibitors with dual cholinesterase inhibition and antioxidant properties: Development and structure-activity relationship (SAR) studies. , 2017, European journal of medicinal chemistry.

[22]  Yang Fan,et al.  Heterogeneous Palladium‐Catalyzed Hydrogen‐Transfer Cyclization of Nitroacetophenones with Benzylamines: Access to C−N Bonds , 2016 .

[23]  G. Deng,et al.  Lewis acid-catalyzed 2-arylquinazoline formation from N′-arylbenzimidamides and paraformaldehyde , 2016 .

[24]  N. Azas,et al.  Looking for new antiplasmodial quinazolines: DMAP-catalyzed synthesis of 4-benzyloxy- and 4-aryloxy-2-trichloromethylquinazolines and their in vitro evaluation toward Plasmodium falciparum. , 2016, European journal of medicinal chemistry.

[25]  K. Skubi,et al.  Dual Catalysis Strategies in Photochemical Synthesis , 2016, Chemical reviews.

[26]  G. Khodarahmi,et al.  Quinazolinone and quinazoline derivatives: recent structures with potent antimicrobial and cytotoxic activities , 2016, Research in pharmaceutical sciences.

[27]  Jieping Zhu,et al.  Cross-Coupling Hydrogen Evolution by Visible Light Photocatalysis Toward C(sp(2))-P Formation: Metal-Free C-H Functionalization of Thiazole Derivatives with Diarylphosphine Oxides. , 2016, Organic letters.

[28]  Yanmei Zhang,et al.  Synthesis and Evaluation of Novel Erlotinib-NSAID Conjugates as More Comprehensive Anticancer Agents. , 2015, ACS medicinal chemistry letters.

[29]  S. Saad,et al.  A new and facile CuCl2·2H2O-catalyzed one-pot three-component synthesis for quinazolines , 2015, Monatshefte für Chemie - Chemical Monthly.

[30]  B. Green Prazosin in the Treatment of PTSD , 2014, Journal of psychiatric practice.

[31]  S. Bari,et al.  Quinazolines: new horizons in anticonvulsant therapy. , 2014, European journal of medicinal chemistry.

[32]  A. Saeed,et al.  Recent advances in the structural library of functionalized quinazoline and quinazolinone scaffolds: synthetic approaches and multifarious applications. , 2014, European journal of medicinal chemistry.

[33]  L. Shaw,et al.  Antibacterial activity of a series of N2,N4-disubstituted quinazoline-2,4-diamines. , 2014, Journal of medicinal chemistry.

[34]  S. Saha,et al.  I2-Catalyzed three-component protocol for the synthesis of quinazolines , 2012 .

[35]  P. Pratap,et al.  DDQ/TBHP-Induced Oxidative Cyclization Process: A Metal-Free Approach for the Synthesis of 2-Phenylquinazolines , 2012 .

[36]  Xiao‐Nan Zhang,et al.  Catalyst-free synthesis of quinazoline derivatives using low melting sugar–urea–salt mixture as a solvent , 2012 .

[37]  A. Thangamani Regiospecific synthesis and biological evaluation of spirooxindolopyrrolizidines via [3+2] cycloaddition of azomethine ylide. , 2010, European journal of medicinal chemistry.

[38]  A. Kadi,et al.  Synthesis, analgesic and anti-inflammatory evaluation of some novel quinazoline derivatives. , 2010, European journal of medicinal chemistry.

[39]  N. Fujii,et al.  Direct synthesis of quinazolines through copper-catalyzed reaction of aniline-derived benzamidines. , 2010, Organic letters.

[40]  Anren Hu,et al.  Antimicrobial study of newly synthesized 6-substituted indolo[1,2-c]quinazolines. , 2010, European journal of medicinal chemistry.

[41]  U. Murthy,et al.  Synthesis of multisubstituted quinolines from Baylis-Hillman adducts obtained from substituted 2-chloronicotinaldehydes and their antimicrobial activity. , 2006, Bioorganic & medicinal chemistry.

[42]  P. Guiry,et al.  Synthesis of Quinazolinones and Quinazolines , 2005 .

[43]  E. Peskind,et al.  Reduction of nightmares and other PTSD symptoms in combat veterans by prazosin: a placebo-controlled study. , 2003, The American journal of psychiatry.

[44]  Corey R J Stephenson,et al.  Visible light photoredox catalysis: applications in organic synthesis. , 2011, Chemical Society reviews.

[45]  J. Michael Quinoline, quinazoline and acridone alkaloids. , 2008, Natural product reports.