Sulfate esters of morphine derivatives: synthesis and characterization.
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S. Béni | B. Noszál | A. Váradi | A. Gergely | S. Hosztafi | P. Jankovics
[1] U. Desai,et al. Chemical Sulfation of Small Molecules - Advances and Challenges. , 2010, Tetrahedron.
[2] Weihong Zheng. Activation of mu opioid receptor inhibits the excitatory glutamatergic transmission in the anterior cingulate cortex of the rats with peripheral inflammation. , 2010, European journal of pharmacology.
[3] B. Noszál,et al. Structural and physicochemical profiling of morphine and related compounds of therapeutic interest. , 2009, Mini-Reviews in Medical Chemistry.
[4] M. Korostyński,et al. Local peripheral opioid effects and expression of opioid genes in the spinal cord and dorsal root ganglia in neuropathic and inflammatory pain , 2009, PAIN.
[5] A. Somogyi,et al. Role of active metabolites in the use of opioids , 2009, European Journal of Clinical Pharmacology.
[6] P. García-Nogales,et al. Tolerance to the antinociceptive effects of peripherally administered opioids Expression of β-arrestins , 2009, Brain Research.
[7] R. Meyer,et al. Peripherally acting mu-opioid receptor agonist attenuates neuropathic pain in rats after L5 spinal nerve injury , 2008, PAIN.
[8] Howard S. Smith,et al. Peripherally-acting opioids. , 2008, Pain physician.
[9] D. Butterfield,et al. Opiate receptor binding properties of morphine-, dihydromorphine-, and codeine 6-O-sulfate ester congeners. , 2006, Bioorganic & medicinal chemistry letters.
[10] Steven Edward Kern,et al. Role of morphine's metabolites in analgesia: Concepts and controversies , 2006, The AAPS Journal.
[11] A. Gergely,et al. 6-oxo-morphinane oximes: pharmacology, chemistry and analytical application. , 2004, Current medicinal chemistry.
[12] M. Eguchi. Recent advances in selective opioid receptor agonists and antagonists , 2004, Medicinal research reviews.
[13] T. Lis,et al. Synthesis and X-ray structures of sulfate esters of fructose and its isopropylidene derivatives. Part 1: 2,3:4,5-di-O-isopropylidene-beta-D-fructopyranose 1-sulfate and 4,5-O-isopropylidene-beta-D-fructopyranose 1-sulfate. , 2002, Carbohydrate research.
[14] Amy Zuckerman,et al. Pharmacological characterization of morphine-6-sulfate and codeine-6-sulfate , 1999, Brain Research.
[15] R. Prankerd,et al. Investigation of the antinociceptive efficacy and relative potency of extended duration injectable 3-acylmorphine-6-sulfate prodrugs in rats , 1998 .
[16] R. Prankerd,et al. Ester prodrugs of a potent analgesic, morphine-6-sulfate: syntheses, spectroscopic and physicochemical properties , 1998 .
[17] A. Somogyi,et al. The disposition of morphine and its 3- and 6-glucuronide metabolites in humans and animals, and the importance of the metabolites to the pharmacological effects of morphine. , 1996, Drug metabolism reviews.
[18] S. Hosztafi,et al. Application of the Mitsunobu Reaction for the Preparation of Isomorphine and Isocodeine Derivatives , 1991 .
[19] F. Kaspersen,et al. A review of the methods of chemical synthesis of sulphate and glucuronide conjugates. , 1987, Xenobiotica; the fate of foreign compounds in biological systems.
[20] J. Fujimoto,et al. Analgesic potencies of morphine 3- and 6-sulfates after intracerebroventricular administration in mice: relationship to structural characteristics defined by mass spectrometry and nuclear magnetic resonance. , 1985, Journal of pharmaceutical sciences.
[21] A. DiSciullo,et al. Diastereoisomeric quaternary morphinium salts: synthesis, stereochemistry and analgesic properties , 1984 .
[22] J. Bowen,et al. Circular dichroism spectra of opium alkaloids in the solid state , 1980 .
[23] H. Krebs,et al. Isolation and identification of morphine 3- and 6-glucuronides, morphine 3,6-diglucuronide, morphine 3-ethereal sulfate, normorphine, and normorphine 6-glucuronide as morphine metabolites in humans. , 1977, Journal of pharmaceutical sciences.
[24] J. Fishman,et al. Narcotic antagonists. 1. Isomeric sulfate and acetate esters of naloxone (N-allylnoroxymorphone). , 1973, Journal of medicinal chemistry.
[25] K. Oguri,et al. Chemical synthesis and analgesic effect of morphine ethereal sulfates. , 1972, Life sciences. Pt. 1: Physiology and pharmacology.
[26] J. Fujimoto,et al. Isolation of Naloxone–3–Ethereal Sulfate from Urine of the Cat 1 , 1972, Proceedings of the Society for Experimental Biology and Medicine. Society for Experimental Biology and Medicine.
[27] C. I. Wright. THE ENZYMATIC DEACETYLATION OF HEROIN AND RELATED MORPHINE DERIVATIVES BY BLOOD SERUM , 1941 .
[28] B. Noszál,et al. HPCE analysis of hydrolysing morphine derivatives. Quantitation of decomposition rate and mobility , 2000 .
[29] R. Purdie,et al. Analytical applications of circular dichroism. , 1989, Journal of pharmaceutical and biomedical analysis.
[30] W. Purdie. Analytical application of circular dichroism , 1987 .
[31] N. Purdie,et al. Simultaneous determination of opiates by circular dichroism. , 1986, Analytical chemistry.
[32] N. Purdie,et al. Circular dichroism spectra of opium alkaloids in aqueous media , 1981 .
[33] J. Norymberski,et al. 773. Steroid sulphates. Part I. Some solvolytic reactions of the salts of steroid sulphates , 1957 .