Automated Optimized Synthesis of [18F]FLT Using Non-Basic Phase-Transfer Catalyst with Reduced Precursor Amount
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[1] V. Goh,et al. Role of 3'-Deoxy-3'-[18F] Fluorothymidine Positron Emission Tomography-Computed Tomography as a Predictive Biomarker in Argininosuccinate Synthetase 1-Deficient Thoracic Cancers Treated With Pegargiminase , 2022, JTO clinical and research reports.
[2] M. Ray,et al. Automated Radiochemical Synthesis of Pharmaceutical Grade [18 F]FLT using 3-N-Boc-5'-O-dimethoxytrityl-3'-O-nosyl-thymidine precursor and its Sep-Pak® Purification employing Selective Elution from Reversed Phase. , 2022, Journal of labelled compounds & radiopharmaceuticals.
[3] R. Krasikova,et al. Automated synthesis of the 16α-[18F]fluoroestradiol ([18F]FES): minimization of precursor amount and resulting benefits , 2020 .
[4] O. Fedorova,et al. Tetrabutylammonium tosylate as inert phase-transfer catalyst: The key to high efficiency SN2 radiofluorinations. , 2020, Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.
[5] R. Krasikova,et al. A fully automated azeotropic drying free synthesis of O-(2-[18F]fluoroethyl)-l-tyrosine ([18F]FET) using tetrabutylammonium tosylate. , 2019, Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.
[6] R. Krasikova,et al. Automated SPE-based synthesis of 16α-[18F]fluoroestradiol without HPLC purification step. , 2018, Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.
[7] S. G. Patching,et al. Nucleoside transporters in PET imaging of proliferating cancer cells using 3ꞌ-deoxy-3ꞌ-[18F]fluoro-L-thymidine , 2018 .
[8] G. Shen,et al. Correlations of 18F-FDG and 18F-FLT uptake on PET with Ki-67 expression in patients with lung cancer: a meta-analysis , 2018, Acta radiologica.
[9] I. Tsougos,et al. 18F-fluorothymidine PET imaging in gliomas: an update , 2017, Annals of Nuclear Medicine.
[10] A. Ouadi,et al. Automated and efficient radiosynthesis of [(18)F]FLT using a low amount of precursor. , 2016, Nuclear medicine and biology.
[11] W. Oyen,et al. A systematic review on [(18)F]FLT-PET uptake as a measure of treatment response in cancer patients. , 2016, European journal of cancer.
[12] E. McKinley,et al. High-yielding, automated production of 3'-deoxy-3'-[(18)F]fluorothymidine using a modified Bioscan Coincidence FDG reaction module. , 2015, Applied radiation and isotopes : including data, instrumentation and methods for use in agriculture, industry and medicine.
[13] M. Muzi,et al. Applications of PET imaging with the proliferation marker [18F]-FLT. , 2015, The quarterly journal of nuclear medicine and molecular imaging : official publication of the Italian Association of Nuclear Medicine (AIMN) [and] the International Association of Radiopharmacology (IAR), [and] Section of the Society of....
[14] B. Solomon,et al. Effect of Platinum-Based Chemoradiotherapy on Cellular Proliferation in Bone Marrow and Spleen, Estimated by 18F-FLT PET/CT in Patients with Locally Advanced Non–Small Cell Lung Cancer , 2014, The Journal of Nuclear Medicine.
[15] F. Bertagna,et al. The role of F-18-fluorothymidine PET in oncology , 2013, Clinical and Translational Imaging.
[16] Yuka Yamamoto,et al. Usefulness of 3′-Deoxy-3′-18F-Fluorothymidine PET for Predicting Early Response to Chemoradiotherapy in Head and Neck Cancer , 2012, The Journal of Nuclear Medicine.
[17] A. Bogni,et al. Simple preparation and purification of ethanol-free solutions of 3'-deoxy-3'-[18F]fluorothymidine by means of disposable solid-phase extraction cartridges. , 2012, Nuclear medicine and biology.
[18] Federico Turkheimer,et al. [18F]-3′Deoxy-3′-Fluorothymidine Positron Emission Tomography and Breast Cancer Response to Docetaxel , 2011, Clinical Cancer Research.
[19] T. Saga,et al. PET/CT with 3′-deoxy-3′-[18F]fluorothymidine for lung cancer patients receiving carbon-ion radiotherapy , 2011, Nuclear medicine communications.
[20] S. Oh,et al. Simple and highly efficient synthesis of 3′-deoxy-3′-[18F]fluorothymidine using nucleophilic fluorination catalyzed by protic solvent , 2007, European Journal of Nuclear Medicine and Molecular Imaging.
[21] Dong Wook Kim,et al. A new class of SN2 reactions catalyzed by protic solvents: Facile fluorination for isotopic labeling of diagnostic molecules. , 2006, Journal of the American Chemical Society.
[22] J. Yeo,et al. Fully automated synthesis system of 3'-deoxy-3'-[18F]fluorothymidine. , 2004, Nuclear medicine and biology.
[23] Dae Hyuk Moon,et al. High radiochemical yield synthesis of 3'-deoxy-3'-[18F]fluorothymidine using (5'-O-dimethoxytrityl-2'-deoxy-3'-O-nosyl-beta-D-threo pentofuranosyl)thymine and its 3-N-BOC-protected analogue as a labeling precursor. , 2003, Nuclear medicine and biology.
[24] U. Haberkorn,et al. A new precursor for the radiosynthesis of [18F]FLT. , 2002, Nuclear medicine and biology.
[25] Otto Muzik,et al. Imaging proliferation in vivo with [F-18]FLT and positron emission tomography , 1998, Nature Medicine.
[26] L. T. C. Nascimento,et al. Comparison between Two Ethanolic Solutions for 3’-Deoxy-3’-[ 18 F]Fluorothymidine Elution , 2017 .