The utility of computed superdelocalizability for predicting the LC50 values of epoxides to guppies.
暂无分享,去创建一个
A quantitative structure-activity relationship (QSAR) was found for predicting the pseudo-first-order reaction rate constant of the alkylating chemical 4-nitrobenzylpyridine with a set of epoxides. The superdelocalizability of the unoccupied levels of the orbital along the carbon-oxygen bond of the least substituted carbon was found to be an excellent predictor. This parameter, along with the log of the octanol/water partition coefficient (log P), were found to be predictors in a QSAR for guppy (Poecilla reticulata) 14-day LC50 values.
[1] Kenichi Fukui,et al. Theory of Substitution in Conjugated Molecules , 1954 .
[2] J. Hermens,et al. A quantitative structure-activity relationship for the acute toxicity of some epoxy compounds to the guppy , 1988 .
[3] Osamu Kikuchi,et al. Systematic QSAR procedures with quantum chemical descriptors , 1987 .