Structure-Based Optimization of the Third Generation Type II Macrocycle TRK Inhibitors with Improved Activity against Solvent-Front, xDFG, and Gatekeeper Mutations.
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Ke Ding | Zhang Zhang | Zhi-Min Zhang | Yang Zhou | Jie Wang | Yongjin Wang | Xiaojuan Song | Zuqin Wang | Xiaoyun Lu | Zhengchao Tu | Shuang Xiang | Hengliang Zhou | Shukai Song