Reformatsky reactions with N-arylpyrrolidine-2-thiones: synthesis of tricyclic analogues of quinolone antibacterial agents
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[1] N. Osheroff,et al. Type II topoisomerases as targets for quinolone antibacterials: turning Dr. Jekyll into Mr. Hyde. , 2001, Current pharmaceutical design.
[2] M. Fujita,et al. Stereoselective synthesis of diastereomeric atropisomeric lactam with various ring sizes and their structural characterization , 2000 .
[3] P. Appelbaum,et al. The fluoroquinolone antibacterials: past, present and future perspectives. , 2000, International journal of antimicrobial agents.
[4] J. Stables,et al. Enaminones-versatile therapeutic pharmacophores. Further advances. , 2000, Current medicinal chemistry.
[5] Hasegawa,et al. Synthesis of optically active 5-substituted-2-pyrrolidinone derivatives having atropisomeric structure and 3,5-cis-selective reaction of their enolates with electrophiles , 2000, The Journal of organic chemistry.
[6] S. Pelly,et al. Enaminones: versatile intermediates for natural product synthesis , 1999 .
[7] C. Pak,et al. Reaction of thioamides with zinc enolate: Synthesis of vinylogous carbamates , 1999 .
[8] K. Lee,et al. Recent advances in the discovery and development of quinolones and analogs as antitumor agents. , 1999, Current medicinal chemistry.
[9] C. B. Koning,et al. A versatile synthesis of tricyclic analogues of quinolone antibacterial agents: Use of a novel reformatsky reaction , 1996 .
[10] T. Gootz,et al. Fluoroquinolone antibacterials: SAR, mechanism of action, resistance, and clinical aspects , 1996, Medicinal research reviews.
[11] T. Kinoshita,et al. A novel synthesis of the pyrazolo[1,5-a]quinoline ring system. New N1-C2 bridged DNA gyrase inhibitors via a novel tandem 1,4-conjugate addition-Michael [3+2] annulation process , 1996 .
[12] K. Scott,et al. Anticonvulsant enaminones: with emphasis on methyl 4-[(p-chlorophenyl)amino]-6-methyl-2-oxocyclohex-3-en-1-oate (ADD 196022) , 1994 .
[13] Guncheol Kim,et al. A synthesis of (±)-supinidine via an intramolecular carbenoid-thioimide coupling reaction , 1994 .
[14] L. Bhat,et al. Reformatsky Reaction on Thiocarbonyl Compounds : New C-C Bond Forming Reaction , 1993 .
[15] G. Schulte,et al. The total synthesis of indolizomycin , 1993 .
[16] S. Rádl,et al. Recent Advances in the Synthesis of Antibacterial Quinolones , 1993 .
[17] G. Crumplin. The 4-Quinolones: Anti Bacterial Agents in Vitro , 1990, Springer Series in Applied Biology.
[18] D. Boger,et al. Total synthesis and evaluation of (.+-.)-N-(tert-butoxycarbonyl)-CBI, (.+-.)-CBI-CDPI1, and (.+-.)-CBI-CDPI2: CC-1065 functional agents incorporating the equivalent 1,2,9,9a-tetrahydrocyclopropa[1,2-c]benz[1,2-e]indol-4-one (CBI) left-hand subunit , 1989 .
[19] J. Michael,et al. Syntheses of alkyl (E)-(1-aryl-2-pyrrolidinylidene)acetates , 1988 .
[20] D. Chu,et al. Short syntheses of 1,2,3,5‐tetrahydro‐5‐oxopyrrolo‐[1,2‐a]quinoline‐4‐carboxylic acid and 1,2,3,4‐tetrahydro‐6H‐6‐oxopyrido[1,2‐a]quinoline‐5‐carboxylic acid derivatives , 1987 .
[21] M. V. Sargent,et al. Boron trichloride as a selective demethylating agent for hindered ethers: a synthesis of the phytoalexins α- and β-pyrufuran, a synthesis of tri-O-methylleprolomin and its demethylation , 1984 .
[22] S. Raucher,et al. Ultrasound in heterogeneous organic reactions. Improved procedure for the synthesis of thioamides , 1981 .
[23] G. Coppola,et al. Novel heterocycles. 6. The condensation of ethyl o‐fluorobenzoyl acetate with cyclic imino ethers , 1980 .
[24] M. Roth,et al. Sulfidkontraktion via alkylative Kupplung: Eine methode zur darstellung von β‐dicarbonylderivaten. Über synthetische methoden, 1. Mitteilung , 1971 .
[25] M. S. Manhas,et al. Cyclization of .omega.-halo amides to lactams , 1967 .
[26] J. S. Buck,et al. Some 9-Amino-3-nitroacridine Derivatives , 1957 .
[27] R. Gould,et al. The Synthesis of Certain Substituted Quinolines and 5,6-Benzoquinolines , 1939 .