Solvent-free synthesis of penta-substituted pyrroles: one-pot reaction of amine, alkyl acetoacetate, and fumaryl chloride
暂无分享,去创建一个
[1] A. Alizadeh,et al. Synthesis of Highly Functionalized Pyrrole Derivatives via a Four-Component Reaction of Two Primary Amines and Diketene in the Presence of Nitrostyrene , 2008 .
[2] A. Alizadeh,et al. One-Pot Synthesis of Pyrrolo[2,1-a]isoquinoline-1-carboxamide Derivatives via a Four-Component Reaction , 2008 .
[3] A. Alizadeh,et al. One-pot synthesis of 4,5-dihydro-1H-pyrrol-3-carboxamide derivatives via a four-component reaction , 2008 .
[4] J. Yadav,et al. PMA/SiO2 as efficient, cost-effective and recyclable catalytic system for the synthesis of highly substituted pyrroles , 2007 .
[5] A. Alizadeh,et al. One-pot synthesis of functionalized furamide derivatives via a three-component reaction between an amine, diketene and dibenzoylacetylene in the presence of triphenylphosphine , 2007 .
[6] A. Alizadeh,et al. A Novel Synthesis of Aminofurans Using a Four-Component Reaction , 2007 .
[7] C. Bruneau,et al. Tertiary 3-Aminopropenones and 3-Aminopropenoates: Their Preparation, with and without Lewis Acids, from Secondary Amines and 1,3-Diketo Compounds , 2007 .
[8] A. J. Whitehead,et al. A convenient one-pot aza-annulation of primary amines, acryloyl chloride and electron-deficient allenes , 2007 .
[9] A. Alizadeh,et al. A new method for the synthesis of functionalized 5-hydroxy-1,5-dihydro-2H-pyrrol-2-one : Reaction of an enamine, derived from addition of a secondary amine to dibenzoylacetylene, with an arylsulfonyl isocyanate , 2006 .
[10] A. Alizadeh,et al. A new method for the synthesis of functionalized maleimides , 2006 .
[11] Mao‐Lin Hu,et al. A Novel Four-Component Reaction for the Synthesis of 2,5-Diaminofuran Derivatives , 2006 .
[12] Mohammed Abid,et al. Organofluorine inhibitors of amyloid fibrillogenesis. , 2006, Biochemistry.
[13] Matthew D. Wessel,et al. Estrogen receptor beta selective ligands: discovery and SAR of novel heterocyclic ligands. , 2005, Bioorganic & medicinal chemistry letters.
[14] P. Baran,et al. Direct coupling of pyrroles with carbonyl compounds: short enantioselective synthesis of (S)-ketorolac. , 2005, Angewandte Chemie.
[15] D. Boger,et al. Multidrug resistance reversal activity of permethyl ningalin B amide derivatives. , 2004, Bioorganic & medicinal chemistry letters.
[16] G. Balme,et al. Pyrrole syntheses by multicomponent coupling reactions. , 2004, Angewandte Chemie.
[17] P. Dervan,et al. Expanding the repertoire of heterocycle ring pairs for programmable minor groove DNA recognition. , 2004, Journal of the American Chemical Society.
[18] D. Tejedor,et al. A diversity-oriented strategy for the construction of tetrasubstituted pyrroles via coupled domino processes. , 2004, Journal of the American Chemical Society.
[19] K. Scheidt,et al. Catalytic multicomponent synthesis of highly substituted pyrroles utilizing a one-pot sila-Stetter/Paal-Knorr strategy. , 2004, Organic letters.
[20] R. Bürli,et al. DNA binding ligands targeting drug-resistant Gram-positive bacteria. Part 2: C-terminal benzimidazoles and derivatives. , 2004, Bioorganic & medicinal chemistry letters.
[21] Jie Zhang,et al. Design and synthesis of poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors. Part 4: biological evaluation of imidazobenzodiazepines as potent PARP-1 inhibitors for treatment of ischemic injuries. , 2003, Bioorganic & medicinal chemistry.
[22] Dorte Renneberg,et al. Imidazopyridine/Pyrrole and hydroxybenzimidazole/pyrrole pairs for DNA minor groove recognition. , 2003, Journal of the American Chemical Society.
[23] V. Nair,et al. A novel synthesis of 2-aminopyrroles using a three-component reaction. , 2001, The Journal of organic chemistry.
[24] L. Barrier,et al. Synthesis and antioxidant activity of new tetraarylpyrroles. , 1999, European journal of medicinal chemistry.
[25] T. Tamaoki,et al. Synthesis and antitumor activity of duocarmycin derivatives: modification of segment-A of A-ring pyrrole compounds. , 1999, Journal of Medicinal Chemistry.
[26] D. Boger,et al. Total Syntheses of Ningalin A, Lamellarin O, Lukianol A, and Permethyl Storniamide A Utilizing Heterocyclic Azadiene Diels−Alder Reactions , 1999 .
[27] M. Maccoss,et al. Pyrroles and other heterocycles as inhibitors of p38 kinase. , 1998, Bioorganic & medicinal chemistry letters.
[28] M. Del Poeta,et al. Structure-In Vitro Activity Relationships of Pentamidine Analogues and Dication-Substituted Bis-Benzimidazoles as New Antifungal Agents , 1998, Antimicrobial Agents and Chemotherapy.
[29] M. Baumgarten,et al. Nonclassical Conducting Polymers: New Approaches to Organic Metals? , 1998 .
[30] Alan R. Katritzky,et al. Comprehensive Heterocyclic Chemistry IV , 1996 .
[31] A. Fürstner,et al. A New, Titanium-Mediated Approach to Pyrroles: First Synthesis of Lukianol A and Lamellarin 0 Dimethyl Ether , 1995 .
[32] V. Demopoulos,et al. Isomeric benzoylpyrroleacetic acids: some structural aspects for aldose reductase inhibitory and anti-inflammatory activities. , 1995, Journal of pharmaceutical sciences.
[33] G. Gribble. Recent developments in indole ring synthesis—methodology and applications , 2010 .
[34] G. Pagani. Heterocycle-Based Electric Conductors , 1994 .
[35] A. Katritzky,et al. 1-Aza-1,3-bis(triphenylphosphoranylidene)propane: A Novel :CHCH2N: Synthon , 1994 .
[36] E G McMahon,et al. Nonpeptide angiotensin II antagonists: N-phenyl-1H-pyrrole derivatives are angiotensin II receptor antagonists. , 1993, Journal of medicinal chemistry.
[37] R. Dowell,et al. Novel inhibitors of prolyl 4-hydroxylase. Part 4 pyridine-2-carboxylic acid analogues with alternative 2-substituents , 1993 .
[38] H. Wurziger,et al. Synthesis and biological activities of meribendan and related heterocyclic benzimidazolo-pyridazinones , 1993 .
[39] F. Berrée,et al. Base mediated reactions in solid-liquid media. A 1,3-dipolar cycloaddition route to pyrrolines and pyrroles from imino chlorosulfides , 1992 .
[40] W. Denny,et al. Potential antitumor agents. 59. Structure-activity relationships for 2-phenylbenzimidazole-4-carboxamides, a new class of "minimal" DNA-intercalating agents which may not act via topoisomerase II. , 1990, Journal of medicinal chemistry.
[41] A. Mertens,et al. Nonsteroidal cardiotonics. 2. The inotropic activity of linear, tricyclic 5-6-5 fused heterocycles. , 1989, Journal of medicinal chemistry.
[42] P. Schiatti,et al. 3-Alkyl-2-aryl-3H-naphth[1,2-d]imidazoles, a novel class of nonacidic antiinflammatory agents. , 1984, Journal of medicinal chemistry.
[43] A. Hantzsch. Neue Bildungsweise von Pyrrolderivaten , 1890 .
[44] C. Paal. Synthese von Thiophen- und Pyrrolderivaten , 1885 .
[45] L. Knorr. Synthese von Pyrrolderivaten , 1884 .